RSC Publishing Logo
Perkin Transactions 1 1972-2002 logo

Year 2001
Main Index

Issue 1


Perkin 1 Abstracts: Solid Phase Organic Synthesis
Catherine McCusker Tanya Wildman and Fiona McKerlie
pg 1-ix; DOI:
10.1039/b009122g
PDF
Applications of stoichiometric transition metal complexes in organic synthesis
Anthony J. Fletcher and Steven D. R. Christie
pg 1; DOI:
10.1039/b002281k
PDF
A new synthetic approach to porphyrin--diones and a -2,3,12,13-tetraone: building blocks for laterally conjugated porphyrin arrays
Vinich Promarak and Paul L. Burn
pg 14; DOI:
10.1039/b007389j
PDF
An approach to the synthesis of 5,5-trans-fused lactam analogues of -lactam antibiotics
Paul W. Smith Andrew R. Whittington Kevin N. Cobley Albert Jaxa-Chamiec and Harry Finch
pg 21; DOI:
10.1039/b007286i
PDF
Organophosphorus chemistry. Part 1. The synthesis of alkyl methylphosphonic acids
Christopher M. Timperley Michael Bird Ian Holden and Robin M. Black
pg 26; DOI:
10.1039/b007077g
PDF
Picolyl-armed 1,3-alternate calix[4]areneazacrown ethers
Jong Seung Kim Ok Jae Shon Wonbo Sim Sun Kyu Kim Moon Hwan Cho Jin-Gyu Kim Il-Hwan Suh and Dong Won Kim
pg 31; DOI:
10.1039/b006801m
PDF
Studies on the reactivity of N-(3-thienyl)carbamates
Delphine Brugier Francis Outurquin and Claude Paulmier
pg 37; DOI:
10.1039/b003580g
PDF
Unexpected products from the formylation of N,N-dimethylanilines with 2-formamidopyridine in POCl3
Ying Cheng Peng Jiao David J. Williams and Otto-Meth Cohn
pg 44; DOI:
10.1039/b006148o
PDF
Cross-coupling reactions in Cinchona alkaloid chemistry: aryl-substituted and dimeric quinine, quinidine, as well as quincorine and quincoridine derivatives
Jens Frackenpohl Wilfried M. Braje and H. Martin R. Hoffmann
pg 47; DOI:
10.1039/b004693k
PDF
TFA-catalyzed ring transformation of 4-hydroxycyclobutenone: A simple and general route for preparation of 3-substituted 4-aminofuran-2(5H)-ones
Jie Wang Xin Jiang Ming Chen Zongming Ge Yuefei Hu and Hongwen Hu
pg 66; DOI:
10.1039/b004654j
PDF
Parasite glycoconjugates. Part 11. Preparation of phosphodisaccharide synthetic probes, substrate analogues for the elongating -D-mannopyranosylphosphate transferase in the Leishmania
Andrew J. Ross Irina A. Ivanova Michael A. J. Ferguson and Andrei V. Nikolaev
pg 72; DOI:
10.1039/b004653l
PDF
-Chymotrypsin-catalysed peptide synthesis via the kinetically controlled approach using activated esters as acyl donors in organic solvents with low water content: incorporation of non-protein amino acids into peptides
Toshifumi Miyazawa Shinichi Nakajo Miyako Nishikawa Kazumi Hamahara Kiwamu Imagawa Eiichi Ensatsu Ryoji Yanagihara and Takashi Yamada
pg 82; DOI:
10.1039/b004183l
PDF
Broadening of the substrate tolerance of -chymotrypsin by using the carbamoylmethyl ester as an acyl donor in kinetically controlled peptide synthesis
Toshifumi Miyazawa Kayoko Tanaka Eiichi Ensatsu Ryoji Yanagihara and Takashi Yamada
pg 87; DOI:
10.1039/b004180g
PDF

Issue 2


Perkin 1 Abstracts: Biocatalysis in Organic Synthesis
Gideon Grogan Alexis Carstairs Ian Jackson Denise McIntyre Alan Watt Sabine Flitsch and Nicholas Turner
pg 2-ix; DOI:
10.1039/b010107i
PDF
Perkin 1 Abstracts: Natural Product Synthesis
Jacqueline E. Milne Marcel de Puit and Duncan McAurthur
pg 2-xv; DOI:
10.1039/b010200h
PDF
Stoichiometric asymmetric processes
Peter OBrien
pg 95; DOI:
10.1039/a907926b
PDF
Ring-fused gem-dibromocyclopropanes as precursors to enantiomerically pure D- and L-series 3-deoxy- and 2-amino-2,3-dideoxyaldohexose derivatives
Martin G. Banwell Wolfgang Ebenbeck and Alison J. Edwards
pg 114; DOI:
10.1039/b008146i
PDF
The chemistry of lithiated phosphine oxides: the stereoselective synthesis of alkene-4,5-diols
Thomas Boesen Neil Feeder Martin D. Eastgate David J. Fox Jonathan A. Medlock Charles R. Tyzack and Stuart Warren
pg 118; DOI:
10.1039/b008500f
PDF
Cyclodimerization of indol-2-ylacetylenes. An example of intermolecular enyne–alkyne cycloaddition
Daniele Passarella Alessandra Giardini Marisa Martinelli and Alessandra Silvani
pg 127; DOI:
10.1039/b009154p
PDF
General syntheses of 1-alkyltoxoflavin and 8-alkylfervenulin derivatives of biological significance by the regioselective alkylation of reumycin derivatives and the rates of transalkylation from 1-alkyltoxoflavins into nucleophiles
Tomohisa Nagamatsu and Hirofumi Yamasaki
pg 130; DOI:
10.1039/b007302o
PDF
Scope and limitations of the [1,2]-alkylsulfanyl (SMe, SEt and SCH2Ph) and sulfanyl (SH) migration in the stereospecific synthesis of substituted tetrahydrofurans
Jason Eames Nikolai Kuhnert and Stuart Warren
pg 138; DOI:
10.1039/b007284m
PDF
Synthesis of 3-deazathiamine
Daniel Hawksley David A. Griffin and Finian J. Leeper
pg 144; DOI:
10.1039/b006962k
PDF
Juli–Colonna stereoselective epoxidation of some ,-unsaturated enones possessing a stereogenic centre at the -position: synthesis of a protected galactonic acid derivative
Peter C. Ray and Stanley M. Roberts
pg 149; DOI:
10.1039/b007100p
PDF
Synthesis of thieno[2,3-b]quinoxalines from 2-haloquinoxalines
Montserrat Armengol and John A. Joule
pg 154; DOI:
10.1039/b008459j
PDF
Synthesis of biphenylenes and tetraphenylenes using copper-catalyzed coupling of arylzinc intermediates
S. M. Humayun Kabir Masashi Hasegawa Yoshiyuki Kuwatani Masato Yoshida Haruo Matsuyama and Masahiko Iyoda
pg 159; DOI:
10.1039/b006375o
PDF
Approaches to the synthesis of (+)- and (–)-epibatidine
M. Teresa Barros Christopher D. Maycock and M. Rita Ventura
pg 166; DOI:
10.1039/b002980g
PDF
Stereoselective synthesis of 24-alkyl-22-hydroxysterols based on chelation-controlled radical reactions
Hajime Nagano Mikako Matsuda and Tomoko Yajima
pg 174; DOI:
10.1039/b007139k
PDF
Photoinduced [2+2] cycloadditions (the Paterno–Bchi reaction) of 1H-1-acetylindole-2,3-dione with alkenes
Jie Xue Yan Zhang Tao Wu Hoong-Kun Fun and Jian-Hua Xu
pg 183; DOI:
10.1039/b005576j
PDF
Synthesis of naturally occurring phosphatidylinositol 3,4,5-trisphosphate [PtdIns(3,4,5)P3] and its diastereoisomers
Piers R. J. Gaffney and Colin B. Reese
pg 192; DOI:
10.1039/b007267m
PDF
A conjugate addition–radical cyclisation approach to sesquiterpene-phenol natural products
Barry S. Crombie Colin Smith Christalla Z. Varnavas and Timothy W. Wallace
pg 206; DOI:
10.1039/b005617k
PDF

Issue 3


Professor Christopher J. Moody Recipient of the RSC 2000–2001 Tilden Medal and Lectureship

pg 3-vii; DOI:
10.1039/b009213o
PDF
Perkin 1 Abstracts: Solid Phase Organic Synthesis
Catherine McCusker Tanya Wildman Fiona McKerlie Andrew Gunn Hassan Mamdani Jennifer Delaney and Sabrice Anizon
pg 3-ix; DOI:
10.1039/b100469g
PDF
Unusual chemoselective addition of diisopropylzinc to 2,2-bipyridine-5,5-dicarbonyl compounds in the 2-position and autoxidative reconversion with carbon–carbon bond cleavage
Shigehisa Tanji Takanori Shibata Itaru Sato and Kenso Soai
pg 217; DOI:
10.1039/b009474i
PDF
Observations on the samarium diiodide-promoted C–C fragmentation/ring expansion chemistry of some aliphatic 1,4-diketones
D. Bradley G. Williams Kevin Blann and Cedric W. Holzapfel
pg 219; DOI:
10.1039/b008110h
PDF
A first synthesis of a phosphatidylcholine bearing docosahexaenoic and tetracosahexaenoic acids
Naomichi Baba Md. Khorshed Alam Yoshihiro Mori Syed S. Haider Masatoshi Tanaka Shuhei Nakajima and Sakayu Shimizu
pg 221; DOI:
10.1039/b007923p
PDF
Selenium catalysed oxidations with aqueous hydrogen peroxide. Part I: epoxidation reactions in homogeneous solution
Gerd-Jan ten Brink Bruno C. M. Fernandes Michiel C. A. van Vliet Isabel W. C. E. Arends and Roger A. Sheldon
pg 224; DOI:
10.1039/b008198l
PDF
Synthesis of espicufolin based on 6-endo ring closure of o-alkynoylnaphthols
Hidemitsu Uno Katsuji Sakamoto Erina Honda Kaori Fukuhara Noboru Ono Junya Tanaka and Masahiro Sakanaka
pg 229; DOI:
10.1039/b007859j
PDF
Synthesis and reactivity of -sulfonylvinylselenonium salts: a simple stereoselective synthesis of -functionalized (Z)-vinyl sulfones
Shin-ichi Watanabe Keiichirou Yamamoto Yukiko Itagaki Tatsunori Iwamura Tetsuo Iwama Tadashi Kataoka Genzoh Tanabe and Osamu Muraoka
pg 239; DOI:
10.1039/b007715l
PDF
Studies on the preparation of camphorylidene derivatives of -amino acids
David L. Gamble William P. Hems and Brian Ridge
pg 248; DOI:
10.1039/b007659g
PDF
Spirostanic analogues of teasterone. Synthesis, characterisation and biological activity of laxogenin, (23S)-hydroxylaxogenin and 23-ketolaxogenin (23-oxolaxogenin)
Martín A. Iglesias-Arteaga Roxana Pérez Gil Carlos S. Pérez Martínez and Francisco Coll Manchado
pg 261; DOI:
10.1039/b007656m
PDF
Stereocontrolled synthesis of (2S*,3R*,4R*)-4-hydroxy-3-methylproline using a silicon assisted aza-[2,3]-Wittig sigmatropic rearrangement
James C. Anderson and Alice Flaherty
pg 267; DOI:
10.1039/b007586h
PDF
Regio- and stereoselectivity in the solvomercuriation and intramolecular alkoxymercuriation of cyclic unsaturated alcohols
Yasuhisa Senda Satomi Takayanagi Tomomi Sudo and Hiroki Itoh
pg 270; DOI:
10.1039/b006963i
PDF
Synthesis, X-ray structures and chemistry of enantiomerically pure 10,11-dihydro-5-phenyl-5H-dibenzo[b,f]phosphepine 5-oxides
Paul Wyatt Stuart Warren Mary McPartlin and Tom Woodroffe
pg 279; DOI:
10.1039/b006883g
PDF
Synthesis of sugar-modified derivatives of the unusual nucleoside oxanosine and its carbocyclic analogs as potential inhibitors of HIV
Yoshio Saito Mariko Nakamura Tsuneya Ohno Chanya Chaicharoenpong Eiko Ichikawa Shosuke Yamamura Kuniki Kato and Kazuo Umezawa
pg 298; DOI:
10.1039/b006763f
PDF
Synthesis of novel analogues of the calicheamicin 1I and esperamicin A1B oligosaccharides
Stéphane Moutel and Jacques Prandi
pg 305; DOI:
10.1039/b006113l
PDF
Diethylamino(trimethyl)silane-mediated direct 1,4-addition of naked aldehydes to electron-deficient olefins
Hisahiro Hagiwara Nao Komatsubara Hiroki Ono Tomoyuki Okabe Takashi Hoshi Toshio Suzuki Masayoshi Ando and Michiharu Kato
pg 316; DOI:
10.1039/b005728m
PDF
The thionophosphate–thiolophosphate photoisomerization proceeds predominantly through a non-chain radical pathway. Synthetically viable benzylation of tetrahydrofuran, propan-2-ol and olefins
Veejendra K. Yadav Rengarajan Balamurugan Masood Parvez and Raghav Yamdagni
pg 323; DOI:
10.1039/b003501g
PDF

Issue 4


Perkin 1 Abstracts: Natural Product Synthesis
Jacqueline E. Milne Marcel de Puit Andrew Gunn and Duncan McAurthur
pg 4-xiii; DOI:
10.1039/b100677k
PDF
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis
Gideon Grogan Alexis Carstairs Ian Jackson Denise McIntyre Alan Watt Sabine Flitsch and Nicholas Turner
pg 4-ix; DOI:
10.1039/b100781p
PDF
The synthesis of thiols, selenols, sulfides, selenides, sulfoxides, selenoxides, sulfones and selenones
David J. Procter
pg 335; DOI:
10.1039/b002081h
PDF
Indium triiodide catalysed one-step conversion of tetrahydropyranyl ethers to acetates with high selectivity
Brindaban C. Ranu and Alakananda Hajra
pg 355; DOI:
10.1039/b100014b
PDF
A polymer-supported thionating reagent
Steven V. Ley Andrew G. Leach and R. Ian Storer
pg 358; DOI:
10.1039/b008814p
PDF
Enantiospecific enzyme-catalysed resolution of novel N,N-disubstituted -amino acid phenolic ester derivatives using pig liver esterase
D. Jonathan Bennett Kirsteen I. Buchanan Andrew Cooke Ola Epemolu Niall M. Hamilton Edward J. Hutchinson and Ann Mitchell
pg 362; DOI:
10.1039/b008000o
PDF
The preparation and use of polyHIPE-grafted reactants to reduce alkyl halides under free-radical conditions
Alexandre Chemin Anthony Mercier Hervé Deleuze Bernard Maillard and Olivier Mondain-Monval
pg 366; DOI:
10.1039/b009318l
PDF
Asymmetric synthesis of enantiomerically enriched atropisomeric amides by desymmetrisation of N,N-dialkylmesitamides
Jonathan Clayden Paul Johnson and Jennifer H. Pink
pg 371; DOI:
10.1039/b008678i
PDF
Selective vicarious nucleophilic amination of 3-nitropyridines
Jan M. Bakke Harald Svensen and Raffaela Trevisan
pg 376; DOI:
10.1039/b008660f
PDF
Synthesis of the bis-spiroacetal moiety of the polyether antibiotic CP44,161
Paul R. Allen Margaret A. Brimble and Hishani Prabaharan
pg 379; DOI:
10.1039/b008159k
PDF
Titanium(IV) chloride, zirconium(IV) chloride or boron trichloride and phosphine-promoted Baylis–Hillman reaction of aldehydes with ,-unsaturated ketone
Min Shi Jian-Kang Jiang Shi-Cong Cui and Yan-Shu Feng
pg 390; DOI:
10.1039/b008105l
PDF
Transformations of selenadiazoliumyl-N-unsubstituted methanides (ylides) to new divinyl selenide derivatives and substituted 1,3,5-selenadiazines. Organoselenium systems from azolium 1,3-dipoles
Richard N. Butler and Anthony Fox
pg 394; DOI:
10.1039/b007974j
PDF
Reactions involving fluoride ion. Part 47. Reactions of perfluorobicycloalkenes
Richard D. Chambers and Takayuki Nakamura
pg 398; DOI:
10.1039/b007825p
PDF
Novel organosulfur donors containing hydroxy functionalities: synthesis of bis[2,2-bis(hydroxymethyl)propane-1,3-diyldithio]tetrathiafulvalene and related materials
Turan Ozturk Nezire Saygili Serife Ozkara Melanie Pilkington Craig R. Rice Deborah A. Tranter Figen Turksoy and John D. Wallis
pg 407; DOI:
10.1039/b007660k
PDF
Carbocyclic ring closure of hex-5-enopyranosides and pent-4-enofuranosides: a nitrile oxide approach
John K. Gallos and Theocharis V. Koftis
pg 415; DOI:
10.1039/b007654f
PDF
Gas-phase pyrolysis of 4-amino-3-allylthio-1,2,4-triazoles: a new route to [1,3]thiazolo[3,2-b][1,2,4]triazoles
Dale D. J. Cartwright Bernard A. J. Clark and Hamish McNab
pg 424; DOI:
10.1039/b007638o
PDF
Synthesis of a regio-isomer of kealiiquinone, a marine benzimidazole alkaloid
Seikou Nakamura Naoki Tsuno Masayuki Yamashita Ikuo Kawasaki Shunsaku Ohta and Yoshitaka Ohishi
pg 429; DOI:
10.1039/b007560o
PDF
Alkoxydienylstannanes via metalation of ,-unsaturated and -phenyl acetals: preparation and synthetic uses in the Stille cross-coupling reaction
Paolo Balma Tivola Anna Deagostino Cristina Prandi and Paolo Venturello
pg 437; DOI:
10.1039/b007500k
PDF
Selective metallation of thiophene and thiazole rings with magnesium amide base
Manabu Shilai Yoshinori Kondo and Takao Sakamoto
pg 442; DOI:
10.1039/b007376h
PDF
The role of the ester group in determining the regiochemistry of selected -amino and -ammonio radical cyclisations: generation of 1-azabicyclo[3.2.1]octyl- and -[2.2.2]octyl systems
Ernest W. Della and Paul A. Smith
pg 445; DOI:
10.1039/b006691p
PDF
Microwave-induced 1,3-dipolar intramolecular cycloadditions of N-substituted oximes, nitrones, and azomethine ylides for the chiral synthesis of functionalized nitrogen heterocycles
Qian Cheng Wen Zhang Yoshimichi Tagami and Takayuki Oritani
pg 452; DOI:
10.1039/b006000n
PDF
Heterocycles of biological importance. Part 5. The formation of novel biologically active pyrimido[1,2-a]benzimidazoles from allenic nitriles and aminobenzimidazoles
Peter Forche Asobo Helene Wahe Joseph Tanyi Mbafor Augustin Ephraim Nkengfack Zacharias Tanee Fomum Emmanuel Fondjo Sopbue and Dietrich Döpp
pg 457; DOI:
10.1039/b005511p
PDF
Investigation of arene–arene interaction in stereoselective MCPBA epoxidation
Keiki Kishikawa Mamoru Naruse Shigeo Kohmoto Makoto Yamamoto and Kentaro Yamaguchi
pg 462; DOI:
10.1039/b004098n
PDF

Issue 5


The synthesis of cyclic peptides
John N. Lambert Jeffrey P. Mitchell and Kade D. Roberts
pg 471; DOI:
10.1039/b001942i
PDF
Synthesis of novel 5-amino-6-ethoxy-2-alkylpyrimidine-4-carbonitriles
Amal Al-Azmi Brian L. Booth Robin G. Pritchard and Fernanda J. R. P. Proença
pg 485; DOI:
10.1039/b009804n
PDF
Diastereoselective SmI2 mediated cascade radical cyclisations of methylenecyclopropane derivatives—syntheses of paeonilactone B and 6-epi-paeonilactone A
Raymond J. Boffey William G. Whittingham and Jeremy D. Kilburn
pg 487; DOI:
10.1039/b009513n
PDF
Regiochemistry in alkylation, acylation and methoxycarbonylation of alkali salts from 2-substituted alkenylpropanedinitriles
Hege Karlsen Pål H. Songe Lise Kristin Sunsby Lise Cathrine Hagen Per Kolsaker and Christian Rømming
pg 497; DOI:
10.1039/b009175h
PDF
Synthesis of novel pipecolic acid derivatives. Part 2. Addition of trimethylsilyl cyanide to 3,4,5,6-tetrahydropyridines
Ole Westerhoff Arne Lützen Wolfgang Maison Marc Kosten and Jürgen Martens
pg 508; DOI:
10.1039/b009112j
PDF
Microchip-based synthesis and total analysis systems (SYNTAS): chemical microprocessing for generation and analysis of compound libraries
Michael C. Mitchell Valerie Spikmans Andreas Manz and Andrew J. de Mello
pg 514; DOI:
10.1039/b009037i
PDF
Stereocontrolled synthesis of trifluoromethylated (E)- or (Z)-ynenyl sulfones via sequential transformations
Yanchang Shen Guoping Wang and Jie Sun
pg 519; DOI:
10.1039/b008849h
PDF
Synthesis of trisphaeridine and norchelerythrine through palladium-catalyzed aryl–aryl coupling reactions
Takashi Harayama Hisashi Akamatsu Kana Okamura Taeko Miyagoe Toshihiko Akiyama Hotoshi Abe and Yasuo Takeuchi
pg 523; DOI:
10.1039/b008683p
PDF
Synthesis and structure of 1-methyl-2,6-bis(electron-withdrawing group)-substituted selenabenzenes
Eiji Honda Tatsunori Iwamura Shin-ichi Watanabe Tadashi Kataoka Osamu Muraoka and Genzoh Tanabe
pg 529; DOI:
10.1039/b008562f
PDF
Metabolites of the higher fungi. Part 32. Rosnecatrone, a phytotoxic bicyclo[4.1.0]hept-3-en-2-one from the fungus Rosellinia necatrix Prill
Raymond L. Edwards Derek J. Maitland Ian J. Scowen Antonio J. T. De Sousa and Anthony J. S. Whalley
pg 537; DOI:
10.1039/b008195g
PDF
A strategy for chemical synthesis of selectively methyl-esterified oligomers of galacturonic acid
Mads H. Clausen Malene R. Jørgensen Jesper Thorsen and Robert Madsen
pg 543; DOI:
10.1039/b006981g
PDF
Reaction of tetrafluoroethene oligomers. Part 17. Some reactions of (E/Z)-perfluoro-2,3-dimethylpenta-1,3-diene
Graham D. Burns Paul L. Coe and Colan L. Andrews
pg 552; DOI:
10.1039/b006825j
PDF
Preparation of pyrimido[2,1-a]phthalazines and an aminopyrimido[2,1-a]isoindole by retro Diels–Alder reaction
Pál Sohár Ferenc Miklós Antal Csámpai and Géza Stájer
pg 558; DOI:
10.1039/b005008n
PDF

Issue 6


Perkin 1 Abstracts: Natural Product Synthesis
Andrew Gunn Jaqueline E. Milne Marcel de Puit and Duncan McArthur
pg 6-xvii; DOI:
10.1039/b101363g
PDF
Perkin 1 Abstracts: Solid Phase Organic Synthesis
Fabrice Anizon Jennifer Delaney Andrew Gunn Hassan Mamdani Catherine McCusker Fiona McKerlie and Tanya Wildman
pg 6-vii; DOI:
10.1039/b101365n
PDF
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis
Gideon Grogan Alexis Carstairs Ian Jackson Denise McIntyre Alan Watt Sabine Flitsch and Nicholas Turner
pg 6-xii; DOI:
10.1039/b101581h
PDF
Versatile route to 2,6-dideoxyamino sugars from non-sugar materials: Syntheses of vicenisamine and kedarosamine
Yoshitaka Matsushima Takuya Nakayama Shigehiro Tohyama Tadashi Eguchi and Katsumi Kakinuma
pg 569; DOI:
10.1039/b008878l
PDF
Benzylic oxidation of aromatics with cerium(IV) triflate; synthetic scope and mechanistic insight
Kenneth K. Laali Mark Herbert Brad Cushnyr Anand Bhatt and David Terrano
pg 578; DOI:
10.1039/b008843i
PDF
Cyclodextrins to limit substrate inhibition and alter substrate selectivity displayed by enzymes
Christopher J. Easton Jason B. Harper Sarah J. Head Kitty Lee and Stephen F. Lincoln
pg 584; DOI:
10.1039/b008339i
PDF
Attempts to find a solution to the problem of atropisomer interconversion in 1,8-diarylnaphthalenes and 5,6-diarylacenaphthenes
Melanie Steele Michael Watkinson and Andrew Whiting
pg 588; DOI:
10.1039/b008319o
PDF
The bisected s-trans conformation-controlled highly stereoselective addition of Grignard reagents to C-cyclopropylaldonitrone. An efficient synthesis of 1-phenyl-2-[(S)-1-aminoalkyl]-N,N-diethylcyclopropanecarboxamides, a new class of potent NMDA receptor antagonists
Yuji Kazuta Satoshi Shuto Hiroshi Abe and Akira Matsuda
pg 599; DOI:
10.1039/b008230i
PDF
Further evidence for the participation of primary carbon-centered free radicals in the antimalarial action of the qinghaosu (artemisinin) series of compounds
Dong-Ye Wang Yu-Lin Wu Yikang Wu Jie Liang and Ying Li
pg 605; DOI:
10.1039/b008145k
PDF
Secondary mould metabolites. Part 59. Sesquiterpene illudanes: semi-synthesis of new illudins, structures and biological activity
Alberto Arnone Lucio Merlini Gianluca Nasini Orso Vajna de Pava and Franco Zunino
pg 610; DOI:
10.1039/b007633n
PDF
Steroid-fullerene adducts from Diels–Alder reactions: characterization and the effect on the activity of Ca2+-ATPase
Lian-Sheng Li Yun-Jin Hu Yikang Wu Yu-Lin Wu Jiachang Yue and Fuyu Yang
pg 617; DOI:
10.1039/b007498p
PDF
Pyrimidine annelated heterocycles—synthesis and cycloaddition of the first pyrimido[1,4]diazepine N-oxides
Frances Heaney Cathriona Burke Desmond Cunningham and Patrick McArdle
pg 622; DOI:
10.1039/b007163n
PDF

Issue 7


Perkin 1 Abstracts: Solid Phase Organic Synthesis
Fabrice Anizon Jennifer Delaney Andrew Gunn Hassan Mamdani Catherine McCusker Fiona McKerlie and Tanya Wildman
pg 7-vii; DOI:
10.1039/b102280f
PDF
Enantioselective synthesis of hydroxy ketones through cleavage and formation of acyloin linkage. Enzymatic kinetic resolution via C–C bond cleavage
Ayhan S. Demir Martina Pohl Elena Janzen and Michael Müller
pg 633; DOI:
10.1039/b100341k
PDF
Multiple substitutions on (6-arene)tricarbonylchromium(0) complexes
Susan E. Gibson (née Thomas) Jonathan W. Steed and Surojit Sur
pg 636; DOI:
10.1039/b009639n
PDF
Regioselectivity of methylation of O-demethylangolensin [1-(2,4-dihydroxyphenyl)-2-(4-hydroxyphenyl)propan-1-one]. An expedient synthesis of angolensin
Kristiina Wähälä Tuija Jokela Auli Salakka Seppo Kaltia and Markku Mesilaakso
pg 642; DOI:
10.1039/b100778p
PDF
Efficient 1,8- and 1,9-asymmetric inductions in the Grignard reaction of - and ?-keto esters of 1,1-binaphthalen-2-ols with an oligoether tether as the 2-substituent: application to the synthesis of (–)-malyngolide
Masamitsu Date Yasufumi Tamai Tetsutaro Hattori Hideki Takayama Yoshinori Kamikubo and Sotaro Miyano
pg 645; DOI:
10.1039/b100497m
PDF
The pyridinium reduction route to alkaloids: a synthesis of ()-tashiromine
Roderick W. Bates and Jutatip Boonsombat
pg 654; DOI:
10.1039/b100407g
PDF
Synthesis and absolute configuration of stellettadine A, a bisguanidinium alkaloid isolated from a marine sponge Stelletta sp.
Hirosato Takikawa Dai Nozawa and Kenji Mori
pg 657; DOI:
10.1039/b100206f
PDF
Conversion of enamines, enamides and triazoles by trithiazyl trichloride into 1,2,5-thiadiazoles
Charles W. Rees and Tai-Yuen Yue
pg 662; DOI:
10.1039/b010140k
PDF
The efficient, enantioselective synthesis of quinoxaline, pyrazine and 1,2,4-triazine substituted -amino acids from vicinal tricarbonyls
Robert M. Adlington Jack E. Baldwin David Catterick and Gareth J. Pritchard
pg 668; DOI:
10.1039/b010134f
PDF
The oxidative rearrangement of furan-2-carboximidamides: preparation and properties of 2-acylaminofurans
Mária Boboíková William Clegg Simon J. Coles Miloslava Dandárová Michael B. Hursthouse Tibor Kiss Albeta Krutoíková Tibor Liptaj Nada Prónayová and Christopher A. Ramsden
pg 680; DOI:
10.1039/b010010m
PDF
Total synthesis and radiolabelling of an efficient rt-PA inhibitor: [11C] (Z,Z)-BABCH. A first route to [11C] labelled amidines
Fabrice Siméon Franck Sobrio Fabienne Gourand and Louisa Barré
pg 690; DOI:
10.1039/b009850g
PDF
Novel bis(tetrahydropyrrolo[3,4-b]carbazoles) linked with aliphatic chains: synthesis and structural aspects
Kerstin U. Meyer and Ulf Pindur
pg 695; DOI:
10.1039/b009731o
PDF
Attempts at asymmetric electrosynthesis of -fluorinated cyclopropylphosphonamides
Sophie Goumain Hassan Oulyadi Philippe Jubault Christian Feasson and Jean-Charles Quirion
pg 701; DOI:
10.1039/b008906k
PDF
Utilization of industrial waste materials. Part 20. Stereoselective cycloaddition of silylenes and a disilene to an enantiomerically pure cyclic ketimine derived from an industrial waste material
Nikolai Graf von Keyserlingk Jürgen Martens Detlev Ostendorf Wolfgang Saak and Manfred Weidenbruch
pg 706; DOI:
10.1039/b008708o
PDF
Synthesis and NMR characterisation of novel highly cyclised polyprenoid hydrocarbons from sediments
Emmanuelle Grosjean Jacques Poinsot Armelle Charrié-Duhaut Stéphanie Tabuteau Pierre Adam Jean Trendel Philippe Schaeffer Jacques Connan Daniel Dessort and Pierre Albrecht
pg 711; DOI:
10.1039/b008104n
PDF
Aromatic azapentalenes: 1H- and (mesoionic) 2H-pyrrolotetrazoles. Part 1. Synthesis and spectral characteristics
Dietrich Moderhack Dirk Decker and Bernhard Holtmann
pg 720; DOI:
10.1039/b007873p
PDF
Aromatic azapentalenes: 1H- and (mesoionic) 2H-pyrrolotetrazoles. Part 2. Reaction with electrophiles
Dietrich Moderhack Dirk Decker and Bernhard Holtmann
pg 729; DOI:
10.1039/b007874n
PDF
Pd(0)–Cu(I)-catalyzed cross-coupling of alkynylsilanes with triarylantimony(V) diacetates
Suk-Ku Kang Hyung-Chul Ryu and Young-Taek Hong
pg 736; DOI:
10.1039/b007800j
PDF
Synthesis, characterization, and electrogenerated chemiluminescence of phenyl-substituted, phenyl-annulated, and spirofluorenyl-bridged oligothiophenes
Ullrich Mitschke and Peter Bäuerle
pg 740; DOI:
10.1039/b006553f
PDF
Carbohydrate-derived dienes for intramolecular and asymmetric Diels–Alder reactions
Pilar Areces José Luis Jiménez Maria de la Cruz Pozo Emilio Román and José Antonio Serrano
pg 754; DOI:
10.1039/b006078j
PDF

Issue 8


Gran Magnusson
Jan Kihlberg
pg 767; DOI:
10.1039/b009690n
PDF
Iodine and its interhalogen compounds: versatile reagents in carbohydrate chemistry. XIV. Glycosylated amino acid synthesis
K. P. Ravindranathan Kartha Lluis Ballell Julia Bilke Michael McNeil and Robert A. Field
pg 770; DOI:
10.1039/b009682m
PDF
Synthesis of clustered xenotransplantation antagonists using palladium-catalyzed cross-coupling of prop-2-ynyl -D-galactopyranoside
Bingcan Liu and René Roy
pg 773; DOI:
10.1039/b101234g
PDF
Synthesis of carba sugars from aldonolactones. Part IV. Stereospecific synthesis of carbaheptopyranoses by radical-induced carbocyclisation of 2,3-unsaturated octonolactones
Sussi Holstein Wagner and Inge Lundt
pg 780; DOI:
10.1039/b100708o
PDF
Cyclizations versus rearrangements in the reactions of some epoxyolefins with Lewis acids
Lars Pettersson and Torbjörn Frejd
pg 789; DOI:
10.1039/b010101j
PDF
Stereoselective photochemical transformations of hexopyranosyl imides to highly functionalised heterocycles
Swantje Thiering Carsten E. Sowa and Joachim Thiem
pg 801; DOI:
10.1039/b010020j
PDF
Carbopeptoids: peptides and diketopiperazines incorporating the anomeric centre of mannopyranose
Daniel D. Long Richard J. Tennant-Eyles Juan C. Estevez Mark R. Wormald Raymond A. Dwek Martin D. Smith and George W. J. Fleet
pg 807; DOI:
10.1039/b009940f
PDF
Towards a modular approach for heparin synthesis
Michael Haller and Geert-Jan Boons
pg 814; DOI:
10.1039/b009845k
PDF
Trivalent -D-mannoside clusters as inhibitors of type-1 fimbriae-mediated adhesion of Escherichia coli: structural variation and biotinylation
Thisbe K. Lindhorst Sven Kötter Ulrike Krallmann-Wenzel and Stefan Ehlers
pg 823; DOI:
10.1039/b009786l
PDF
Efficient stereoselective synthesis of 1-thio--mannopyranosides
Henry N. Yu Chang-Chun Ling and David R. Bundle
pg 832; DOI:
10.1039/b009626l
PDF
Synthesis and structure–activity relationships of di- and trisaccharide inhibitors for Shiga-like toxin Type 1
Pavel I. Kitov and David R. Bundle
pg 838; DOI:
10.1039/b009685g
PDF
Studies on aluminium mediated asymmetric Friedel–Crafts hydroxyalkylation reactions of pyridinecarbaldehydes
Aase Sejr Gothelf Tore Hansen and Karl Anker Jørgensen
pg 854; DOI:
10.1039/b009669p
PDF
Halogenation of pyrazoloquinolines and pyrazoloisoquinolines. Theoretical analysis of the regioreactivity and cross-coupling of 3-halogen derivatives
Jan Pawlas Jeremy Greenwood Per Vedsø Tommy Liljefors Palle Jakobsen Per Olaf Huusfeldt and Mikael Begtrup
pg 861; DOI:
10.1039/b006435l
PDF
Conformational selection of non-hydrolyzable glycomimetics: the conformation of N,N-diacetylthiochitobiose bound to wheat germ agglutinin
José Luis Muñoz Alicia García-Herrero Juan Luis Asensio F.-Isabelle Auzennaeau F. Javier Cañada and Jesús Jiménez-Barbero
pg 867; DOI:
10.1039/b006965p
PDF
Synthesis of uronic acid-containing xylans found in wood and pulp
Stefan Oscarson and Pär Svahnberg
pg 873; DOI:
10.1039/b009670a
PDF
Chemoenzymatic synthesis of derivatives of a T-cell-stimulating peptide which carry tumor-associated carbohydrate antigens
Shaji K. George Björn Holm Celso A. Reis Tilo Schwientek Henrik Clausen and Jan Kihlberg
pg 880; DOI:
10.1039/b009567m
PDF
The p-methoxybenzyl ether as an in situ-removable carbohydrate-protecting group: a simple one-pot synthesis of the globotetraose tetrasaccharide
Sumita Bhattacharyya Bengt G. Magnusson Ulf Wellmar and Ulf J. Nilsson
pg 886; DOI:
10.1039/b009448j
PDF
Investigation of the Lewis acid mediated stereoselective cyclization of cationic aminyl radicals leading to substituted pyrrolidines
Åsa Sjöholm Martin Hemmerling Nicolas Pradeille and Peter Somfai
pg 891; DOI:
10.1039/b009391m
PDF
Synthesis and evaluation of anti-HIV activity of 3-azido-4-(hydroxymethyl)tetrahydrofuran derivatives containing 2-(thymin-1-yl)methyl, 2-(cytosin-1-yl)methyl or 2-(adenin-9-yl)methyl substituents – a new series of AZT analogues
Anne G. Olsen Claus Nielsen and Jesper Wengel
pg 900; DOI:
10.1039/b009109j
PDF
Synthesis of 1-azagalactofagomine, a potent galactosidase inhibitor
Henrik Helligsø Jensen and Mikael Bols
pg 905; DOI:
10.1039/b007973l
PDF
Studies on the C-alkylation and C-allylation of small peptides employing glycyl radical intermediates
Peter Blakskjær Lone Pedersen and Troels Skrydstrup
pg 910; DOI:
10.1039/b005468m
PDF

Issue 9


Professor Ei-ichi Negishi
Professor Ei-ichi Negishi
pg 9-xi; DOI:
10.1039/b009326m
PDF
Perkin 1 Abstracts: Natural Product Synthesis
Andrew Gunn Jacqueline E. Milne Marcel de Puit and Duncan McArthur
pg 9-xxi; DOI:
10.1039/b102281b
PDF
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis
Gideon Grogan Alexis Carstairs Ian Jackson Denise McIntyre Alan Watt Sabine Flitsch and Nicholas Turner
pg 9-xiii; DOI:
10.1039/b102587m
PDF
Perkin 1 Abstracts: Solid Phase Organic Synthesis
Fabrice Anizon Jennifer Delaney Andrew Gunn Hassan Mamdani Catherine McCusker Fiona McKerlie and Tanya Wildman
pg 9-xxvi; DOI:
10.1039/b103258p
PDF
The use of supercritical fluids in synthetic organic chemistry
R. Scott Oakes Anthony A. Clifford and Christopher M. Rayner
pg 917; DOI:
10.1039/b101219n
PDF
exo-Glycals from glycosyl cyanides. First generation of C-glycosylmethylene carbenes from 2,5- and 2,6-anhydroaldose tosylhydrazones
Marietta Tóth and László Somsák
pg 942; DOI:
10.1039/b102963k
PDF
Synthesis of N-acylaziridines from -amido selenides
Virginia R. Ward Matthew A. Cooper and A. David Ward
pg 944; DOI:
10.1039/b102468j
PDF
Indium-mediated allylation reactions of -chlorocarbonyl compounds and preparation of allylic epoxides
Jeong Ah Shin Kyung Il Choi Ae Nim Pae Hun Yeong Koh Han-Young Kang and Yong Seo Cho
pg 946; DOI:
10.1039/b101111l
PDF
Unusually facile palladium catalysed oxidation of imidazolidines and oxazolidines
Alexandre Alexakis Isabelle Aujard Julien Pytkowicz Sylvain Roland and Pierre Mangeney
pg 949; DOI:
10.1039/b010089g
PDF
Synthesis and characterisation of -aminophosphine ligands on a solid support
Amal Mansour and Moshe Portnoy
pg 952; DOI:
10.1039/b009640g
PDF
Indium metal as a reducing agent in organic synthesis
Michael R. Pitts Justin R. Harrison and Christopher J. Moody
pg 955; DOI:
10.1039/b101712h
PDF
Synthesis of thieno[2,3-b]quinoxalines and pyrrolo[1,2-a]quinoxalines from 2-haloquinoxalines
Montserrat Armengol and John A. Joule
pg 978; DOI:
10.1039/b101458g
PDF
Synthesis of bicyclic nucleosides by ring-closing metathesis
Jacob Ravn and Poul Nielsen
pg 985; DOI:
10.1039/b101364p
PDF
Development and application of allyl, 2-sulfonylethyl and 2-thioethyl carbamate linkers for solid phase N-acyliminium ion chemistry
Jan H. van Maarseveen Wim J. N. Meester Johan J. N. Veerman Chris G. Kruse Pedro H. H. Hermkens Floris P. J. T. Rutjes and Henk Hiemstra
pg 994; DOI:
10.1039/b100998m
PDF
Asymmetric cycloaddition of anthrone and maleimides catalyzed by C2-chiral pyrrolidines
Kouhei Uemae Satoshi Masuda and Yukio Yamamoto
pg 1002; DOI:
10.1039/b100961n
PDF
Triterpenoid total synthesis. Part 6. Synthesis of testudinariols A and B, triterpene metabolites of the marine mollusc Pleurobrancus testudinarius
Masao Yoshida Hirosato Takikawa and Kenji Mori
pg 1007; DOI:
10.1039/b100777g
PDF
Synthesis of trans-3,4-dihydroxy-3,4-dihydrophenanthro[3,2-b][1]benzothiophene, a potentially carcinogenic metabolite of sulfur heterocycle phenanthro[3,2-b][1]benzothiophene
Subodh Kumar
pg 1018; DOI:
10.1039/b100345n
PDF
Rhodium(II)-carbenoid C–H insertion reactions in the synthesis of ,-dioxospirane systems
Pompiliu S. Aburel Christian Rømming and Kjell Undheim
pg 1024; DOI:
10.1039/b100179p
PDF
An efficient synthesis of highly functionalized asymmetric porphyrins with organolithium reagents
Xiangdong Feng and Mathias O. Senge
pg 1030; DOI:
10.1039/b100012h
PDF
Solvent and ligand effects on selective mono- and dilithiation of 1-(chlorophenyl)pyrroles and 1-(methoxyphenyl)pyrroles
Katalin Fogassy Krisztina Kovács György M. Keser László Tke and Ferenc Faigl
pg 1039; DOI:
10.1039/b100008j
PDF
Synthesis and nicotinic acetylcholine-binding properties of epibatidine homologues: homoepibatidine and dihomoepibatidine
John R. Malpass David A. Hemmings Anna L. Wallis Stephen R. Fletcher and Shailendra Patel
pg 1044; DOI:
10.1039/b010178h
PDF
Stereocontrol in a one-pot procedure for anionic oxy-Cope rearrangement followed by intramolecular aldol reaction
Alistair P. Rutherford Cameron S. Gibb Richard C. Hartley and Jonathan M. Goodman
pg 1051; DOI:
10.1039/b010138i
PDF
The reaction of 1-(2,4,6-trimethylphenyl)-1,2-dihydrophosphinine 1-oxides with dimethyl acetylenedicarboxylate; a [4+2] or a [2+2] cycloaddition?
György Keglevich Ágnes GyöngyvérVaskó András Dobó Krisztina Ludányi and László Tke
pg 1062; DOI:
10.1039/b010080n
PDF
[2+2] Heterodimers of methyl phenanthrene-9-carboxylate and benzene
Taehee Noh Hyun Yu Youngmee Jeong Kyungmoon Jeon and Sukjin Kang
pg 1066; DOI:
10.1039/b009846i
PDF
Thermal decomposition of tert-butyl ortho-(phenylsulfanyl)- and ortho-(phenylsulfonyl)phenyliminoxyperacetates: The reactivity of thio-substituted iminyl radicals
Rino Leardini Hamish McNab Matteo Minozzi and Daniele Nanni
pg 1072; DOI:
10.1039/b009843o
PDF
Gas-phase cyclisation reactions of 1-(2-arylthiophenyl)alkaniminyl and 2-(aryliminomethyl)thiophenoxyl radicals
Tim Creed Rino Leardini Hamish McNab Daniele Nanni Iain S. Nicolson and David Reed
pg 1079; DOI:
10.1039/b009844m
PDF
Synthesis of multifunctionalized phosphonic acid esters via opening of oxiranes and azetidinium salts with phosphoryl-substituted carbanions
Agata Bakalarz-Jeziorna Jan Heliski and Boena Krawiecka
pg 1086; DOI:
10.1039/b009720i
PDF
Synthesis and isomerization of arene oxide metabolites of phenanthrene, triphenylene, dibenz[a,c]anthracene and dibenz[a,h]anthracene
Suresh K. Balani I. N. Brannigan Derek R. Boyd Narain D. Sharma Francis Hempenstall and Allison Smith
pg 1091; DOI:
10.1039/b009712h
PDF
Phenylboronic acid as a labile protective agent: the selective derivatisation of 1,2,3-triols
Vijaya Bhaskar K. Peter J. Duggan David G. Humphrey Guy Y. Krippner Victoria McCarl and Daniel A. Offermann
pg 1098; DOI:
10.1039/b009450l
PDF
Substituted triazines and pyrimidines from 1,3,5-triazine and a lithium amidinate, alkyl- or 1-azaallyl
W. Marco Boesveld Peter B. Hitchcock and Michael F. Lappert
pg 1103; DOI:
10.1039/b008681i
PDF
Synthesis and reactions of some optically active epoxides formally derived from tertiary allylic alcohols
Jamie F. Bickley Adam T. Gillmore Stanley M. Roberts John Skidmore and Alexander Steiner
pg 1109; DOI:
10.1039/b008275i
PDF
Cryptoregiochemistry of a Brassica napus fatty acid desaturase (FAD3): a kinetic isotope effect study
Christopher K. Savile Darwin W. Reed Dauenpen Meesapyodsuk Patrick S. Covello and Peter H. Buist
pg 1116; DOI:
10.1039/b008111f
PDF
Clavulanic acid biosynthesis; the final steps
M. Fulston M. Davison S. W. Elson N. H. Nicholson J. W. Tyler and S. R. Woroniecki
pg 1122; DOI:
10.1039/b007009m
PDF
The reaction of 2-(tetrazol-5-yl)alkyl ketones and of 2-(tetrazol-5-yl)alkanoic acid derivatives with lead tetraacetate. A novel method of preparation of alk-2-ynyl ketones and alk-2-ynoic acid derivatives
József Fetter Ildikó Nagy Le Thanh Giang Mária Kajtár-Peredy Antal Rockenbauer László Korecz and Gábor Czira
pg 1131; DOI:
10.1039/b005286h
PDF
Synthesis of phosphorus- and selenium-containing macrocycles and their complexation with Pd(II)Cl2
J. L. Li J. B. Meng Y. M. Wang J. T. Wang and T. Matsuura
pg 1140; DOI:
10.1039/b005045h
PDF

Issue 10


Perkin 1 Abstracts: Natural Product Synthesis
Andrew Gunn Jacqueline E. Milne Marcel de Puit and Duncan McArthur
pg 10-xv; DOI:
10.1039/b103457j
PDF
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis
Gideon Grogan Alexis Carstairs Ian Jackson Denise McIntyre Alan Watt Sabine Flitsch and Nicholas Turner
pg 10-ix; DOI:
10.1039/b103527b
PDF
A simple entry into enantiopure hydrindanes, hydroisoquinolones and diquinanes from 3,10-dioxygenated dicyclopentadienes: Application to the synthesis of (+)-coronafacic acid and a formal synthesis of (+)-coriolin
Goverdhan Mehta and D. Srinivasa Reddy
pg 1153; DOI:
10.1039/b009307f
PDF
Conversion of homochiral amines, -amino alcohols and -amino acids to their chiral 2-substituted pyrrole derivatives
Ayhan S. Demir Idris M. Akhmedov Özge eenoglu Onur Alptürk Sinem Apaydn Zuhal Gerçek and Nezire Ibrahimzade
pg 1162; DOI:
10.1039/b008317h
PDF
Electrochemical and yeast-catalysed ring-opening of isoxazoles in the synthesis of analogues of the herbicide Grasp
Christopher J. Easton Graham A. Heath C. Merrîcc M. Hughes Connie K. Y. Lee G. Paul Savage Gregory W. Simpson Edward R. T. Tiekink George J. Vuckovic and Richard D. Webster
pg 1168; DOI:
10.1039/b008081k
PDF
Syntheses and X-ray crystal structures of derivatives of 2,2,4,4,6,6-hexaiodobiphenyl
Pier Lucio Anelli Marino Brocchetta (the late) Costantino Maffezzoni Paola Paoli Patrizia Rossi Fulvio Uggeri and Massimo Visigalli
pg 1175; DOI:
10.1039/b009666k
PDF
A stereochemically flexible approach to pyrrolidines based on 5-endo-trig iodocyclisations of homoallylic sulfonamides
Andrew D. Jones David W. Knight and David E. Hibbs
pg 1182; DOI:
10.1039/b008537p
PDF
Convenient synthesis of optically active 1,2-diol monosulfonates and terminal epoxides via oxazaborolidine-catalyzed asymmetric borane reduction of -sulfonyloxy ketones
Byung Tae Cho Weon Ki Yang and Ok Kyung Choi
pg 1204; DOI:
10.1039/b010155i
PDF
1,2-Bis[(2-dimethylamino-2-thioxo-1-phenylethylidene)hydrazino]ethane: a new tetradentate ligand for Ni2+
Jean-Damien Charrier David Deniaud Alain Reliquet and Jean-Claude Meslin
pg 1212; DOI:
10.1039/b101030l
PDF
A multinuclear NMR study of the restricted rotation in a bi-imidazole nucleoside
Jukka Mäki Karel D. Klika Rainer Sjöholm and Leif Kronberg
pg 1216; DOI:
10.1039/b010182f
PDF
Solvent-free bentonite-catalyzed condensation of malonic acid and aromatic aldehydes under microwave irradiation
André Loupy Suk-Jin Song Sun-Mee Sohn Young-Mee Lee and Tae-Woo Kwon
pg 1220; DOI:
10.1039/b009803p
PDF
A novel and convenient method for synthesizing unsymmetrical N-benzyloxycarbonyl-protected 1-amino-1-arylalkylphosphonate mixed diesters
Jiaxi Xu and Nanyan Fu
pg 1223; DOI:
10.1039/b008340m
PDF
Synthesis and reactions of N-(azulen-1-ylmethylene)arylamines
Alexandru C. Razus Carmen Nitu Simona Carvaci Liviu Birzan Stefan A. Razus Mihaela Pop and Laszlo Tarko
pg 1227; DOI:
10.1039/b100007l
PDF
Molybdenum(0) and tungsten(0) catalysts with enhanced reactivity for allylic substitution: regioselectivity and solvent effects
Andrei V. Malkov Ian R. Baxendale Darren J. Mansfield and Pavel Koovský
pg 1234; DOI:
10.1039/b100903f
PDF
A new and efficient approach to the synthesis of 6-amidino-2-oxopurines
Brian L. Booth Isabel M. Cabral Alice M. Dias A. Paula Freitas Ana M. Matos Beja M. Fernanda Proença and Manuela Ramos Silva
pg 1241; DOI:
10.1039/b010224p
PDF

Issue 11


The semi-pinacol rearrangement of homochiral epoxyalcohols catalysed by rare earth triflates
Jamie F. Bickley Bernhardt Hauer Paula C. A. Pena Stanley M. Roberts and John Skidmore
pg 1253; DOI:
10.1039/b101838h
PDF
A novel utilization of trifluoromethanide as a base: a convenient synthesis of trimethylsilylacetylene
Mitsuhiro Yoshimatsu and Masako Kuribayashi
pg 1256; DOI:
10.1039/b101537k
PDF
Enantioselective amino acid recognition using acyclic thiourea receptors
Graham M. Kyne Mark E. Light Mike B. Hursthouse Javier de Mendoza and Jeremy D. Kilburn
pg 1258; DOI:
10.1039/b102298a
PDF
Regio- and stereo-selective dioxygenase-catalysed cis-dihydroxylation of fjord-region polycyclic arenes
Derek R. Boyd Narain D. Sharma John S. Harrison Martina A. Kennedy Christopher C. R. Allen and David T. Gibson
pg 1264; DOI:
10.1039/b101833g
PDF
The azomethine ylide strategy for -lactam synthesis. A comprehensive mechanistic evaluation
David Brown Giles A. Brown Sarah R. Martel Denis Planchenault Evelyn Turmes Kenneth E. Walsh Richard Wisedale Neil J. Hales Colin W. G. Fishwick and Timothy Gallagher
pg 1270; DOI:
10.1039/b010046n
PDF
The azomethine ylide strategy for -lactam synthesis. An evaluation of alternative pathways for azomethine ylide generation
Giles A. Brown Sarah R. Martel Richard Wisedale Jonathan P. H. Charmant Neil J. Hales Colin W. G. Fishwick and Timothy Gallagher
pg 1281; DOI:
10.1039/b010050l
PDF
Intermolecular addition of alkyl radicals to imines in the absence and in the presence of a Lewis acid
Nis Halland and Karl Anker Jørgensen
pg 1290; DOI:
10.1039/b101762o
PDF
Metabolites of the higher fungi. Part 33. Grammicin, a novel bicyclic C7H6O4 furanopyranol from the fungus Xylariagrammica (Mont.) Fr.
Raymond L. Edwards Derek J. Maitland Pattama Pittayakhajonwut and Anthony J. S. Whalley
pg 1296; DOI:
10.1039/b101708j
PDF
Synthesis of substituted hexa-3,5-dienoic acid methyl esters from conjugated dienones
Rishan Lang Nongkhlaw Ridaphun Nongrum and Bekington Myrboh
pg 1300; DOI:
10.1039/b101242h
PDF
One-step synthesis of 5-acylisothiazoles from furans
Jérôme Guillard Christelle Lamazzi Otto Meth-Cohn Charles W. Rees Andrew J. P. White and David J. Williams
pg 1304; DOI:
10.1039/b101157j
PDF
An efficient procedure for cleavage of aziridines with various thiols promoted by ZnCl2
Jie Wu Xue-Long Hou and Li-Xin Dai
pg 1314; DOI:
10.1039/b100591j
PDF
Ebenaceae extractives. Part 11. The synthesis of 7-methyljuglone. A re-examination
Oliver C. Musgrave and Douglas Skoyles
pg 1318; DOI:
10.1039/b009531l
PDF
Binding interactions between 3-aryl-1,2,4-oxadiazol-5-ones and a trisimidazoline base
Anja Reichert Roland Fröhlich Roderick Ferguson and Arno Kraft
pg 1321; DOI:
10.1039/b009451j
PDF
Steroidal guanidines as enantioselective receptors for N-acyl -amino acids. Part 1. 3-Guanylated carbamates derived from cholic acid
Laurence J. Lawless Adrian G. Blackburn Alan J. Ayling M. Nieves Pérez-Payán and Anthony P. Davis
pg 1329; DOI:
10.1039/b009215k
PDF

Issue 12


Perkin 1 Abstracts: Natural Product Synthesis
Andrew Gunn Jacqueline E. Milne Marcel de Puit and Duncan McArthur
pg 12-xvi; DOI:
10.1039/b104270j
PDF
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis
Gideon Grogan Alexis Carstairs Ian Jackson Denise McIntyre Alan Watt Sabine Flitsch and Nicholas Turner
pg 12-ix; DOI:
10.1039/b104422m
PDF
An operationally simple and fully regiocontrolled formal total synthesis of the montanine-type Amaryllidaceae alkaloid ()-pancracine
Martin G. Banwell Alison J. Edwards Katrina A. Jolliffe and Michael Kemmler
pg 1345; DOI:
10.1039/b102252k
PDF
Improved catalytic procedures for the copper(I)-promoted reactions of -amido zinc reagents
Christopher Hunter Richard F. W. Jackson and Harshad K. Rami
pg 1349; DOI:
10.1039/b102446a
PDF
Synthesis and some properties of 7H-naphth[3,2,1-cd]azulen-7-ones and related compounds
Noritaka Abe Hiroyuki Fujii Kahei Takase and Tadayoshi Morita
pg 1353; DOI:
10.1039/b101333p
PDF
Reactions of 7H-naphth[3,2,1-cd]azulen-7-ones
Noritaka Abe Hiroyuki Fujii Kahei Takase and Tadayoshi Morita
pg 1359; DOI:
10.1039/b101332g
PDF
Synthesis of novel Hg2+ receptors based on N-benzyloxyamide derivatives and their application to anion-selective electrodes
Shin-ichi Sasaki Tsuyoshi Amano Satoru Ozawa Tomomi Masuyama Daniel Citterio Hideaki Hisamoto Hisao Hori and Koji Suzuki
pg 1366; DOI:
10.1039/b008978h
PDF
Neighboring group effect of pyridazine and pyrazine rings for -facial selectivity in the reactions of fused isopropylidenenorbornene systems with electrophilic reagents
Tomoshige Kobayashi Kiyomi Miki Behrooz Nikaeen and Akira Ohta
pg 1372; DOI:
10.1039/b101330k
PDF
Dimethyl sulfoxide as a co-solvent dramatically enhances the enantioselectivity in lipase-catalysed resolutions of 2-phenoxypropionic acyl derivatives
Keiichi Watanabe and Shin-ichi Ueji
pg 1386; DOI:
10.1039/b100182p
PDF
Regioselectivity and endo/exo selectivity in the cycloadditions of the phthalazinium dicyanomethanide 1,3-dipole with unsymmetrical alkene and alkyne dipolarophiles. Unexpected reversals of regiochemistry: a combined experimental and DFT theoretical study
Richard N. Butler Anthony G. Coyne Patrick McArdle Desmond Cunningham and Luke A. Burke
pg 1391; DOI:
10.1039/b101150m
PDF
The preparation of novel thiophene-based macrocyclic Mannich bases
Julie D. E. Chaffin John M. Barker and Patrick R. Huddleston
pg 1398; DOI:
10.1039/b007661i
PDF
Synthesis of new bis(tetrahydropyrrolo[3,4-b]carbazoles) with a functionalized diaryl spacer
Farokh Mehrabani and Ulf Pindur
pg 1406; DOI:
10.1039/b006899n
PDF
Palladium catalysed elaboration of codeine and morphine
Stephen G. Davies Christopher J. Goodwin Dirk Pyatt and Andrew D. Smith
pg 1413; DOI:
10.1039/b102581n
PDF
Design of potential new HIV protease inhibitors: enantioconvergent synthesis of new pyrrolidin-3-ol, and pyrrolidin-3-one peptide conjugates
Jérôme Courcambeck Frédéric Bihel Céline De Michelis Gilles Quéléver and Jean Louis Kraus
pg 1421; DOI:
10.1039/b101584m
PDF
Does water suppress the racemization and decomposition of amino acids?
Yuusaku Yokoyama Hidemasa Hikawa and Yasuoki Murakami
pg 1431; DOI:
10.1039/b102254g
PDF
Use of dissolving metals in the partial reduction of pyridines: formation of 2-alkyl-1,2-dihydropyridines
Timothy J. Donohoe Andrew J. McRiner Madeleine Helliwell and Peter Sheldrake
pg 1435; DOI:
10.1039/b101662h
PDF
Stereoselectivity of cyclisations viaN-acyliminium ions to form pyrido[2,3:3,4]pyrrolo[2,1-a]isoindole, -isoquinoline and -benz[c]azepine ring systems
Abood A. Bahajaj John M. Vernon and Giles D. Wilson
pg 1446; DOI:
10.1039/b009316p
PDF
Coordination of (-N-sulfonylaminoalkyl)phosphines and their analogous arsines to PdII and PtII. Application of the Pd-complexes as chiral catalysts in asymmetric hydrosilylation of 1,3-dienes
Magnus Gustafsson Karl-Erik Bergqvist and Torbjörn Frejd
pg 1452; DOI:
10.1039/b101464l
PDF
Synthesis of -hydroxy and -oxospiranes through ruthenium(II)-catalyzed ring-closing metathesis
Pompiliu S. Aburel Christian Rømming Kuangbiao Ma and Kjell Undheim
pg 1458; DOI:
10.1039/b101462p
PDF

Issue 13


Professor C. Robin Ganellin FRS
Professor C. Robin Ganellin
pg 13-vii; DOI:
10.1039/b101382n
PDF
Perkin 1 Abstracts: Solid Phase Organic Synthesis
Fabrice Anizon Jennifer Delaney Andrew Gunn Hassan Mamdani Catherine McCusker Fiona McKerlie and Tanya Wildman
pg 13-ix; DOI:
10.1039/b104302c
PDF
Preparative biotransformations
Stanley M. Roberts
pg 1475; DOI:
10.1039/b101682m
PDF
Chiral pyridylimidazolines: synthesis, arene ruthenium complexes and application in asymmetric catalysis
Adam J. Davenport David L. Davies John Fawcett and David R. Russell
pg 1500; DOI:
10.1039/b103175a
PDF
The scope and limitation of the [1,4]-Sbenzyl participation and debenzylation in the stereochemically controlled synthesis of substituted thiolanes
Jason Eames Nikolai Kuhnert and Stuart Warren
pg 1504; DOI:
10.1039/b102737a
PDF
Rearrangement of 18-iodo- and 20-iodopregnanes mediated by iodosyl derivatives
Daniel Nicoletti Alberto A. Ghini Ricardo F. Baggio M. Teresa Garland and Gerardo Burton
pg 1511; DOI:
10.1039/b102688g
PDF
Aziridination of cyclic dienes with enantiopure 3-acetoxyaminoquinazolin-4(3H)-ones
Robert S. Atkinson and Christopher K. Meades
pg 1518; DOI:
10.1039/b102592a
PDF
[11C]/(13C)Carbon monoxide in palladium-mediated synthesis of imides
Farhad Karimi Tor Kihlberg and Bengt Långström
pg 1528; DOI:
10.1039/b102524b
PDF
Serial synthesis of oxa[3.n]cyclophanes and homooxacalix[n]arenes via reductive coupling of arenedialdehydes, and their X-ray structures
Naoki Komatsu and Takefumi Chishiro
pg 1532; DOI:
10.1039/b102031p
PDF
Highly effective and recyclable chiral auxiliaries: a study of the synthesis and use of three 4-isopropyl-5,5-diaryloxazolidin-2-ones
Karen Alexander (née Gillon) Stuart Cook Colin L. Gibson and Alan R. Kennedy
pg 1538; DOI:
10.1039/b102020j
PDF
Biosynthesis of polyoxypeptin A: novel amino acid 3-hydroxy-3-methylproline derived from isoleucine
Kazuo Umezawa Yoko Ikeda Osamu Kawase Hiroshi Naganawa and Shinichi Kondo
pg 1550; DOI:
10.1039/b101942m
PDF
Synthesis of pentenoic acid analogs as potential anti-influenza agents
Scott C. Mauldin William J. Hornback and John E. Munroe
pg 1554; DOI:
10.1039/b101702k
PDF
C-Alkylation of hydroxyarenes by Michael reaction
Henryk Krawczyk and Ryszard Bodalski
pg 1559; DOI:
10.1039/b101210j
PDF
Synthesis of a new analogue of BINOL based on a homodimer of substituted 1-hydroxypyrazole
Øystein Rist and Mikael Begtrup
pg 1566; DOI:
10.1039/b010126p
PDF
Conversion of alkanenitriles to amidines and carboxylic acids mediated by a cobalt(II)–ketoxime system
Maximilian N. Kopylovich Vadim Yu. Kukushkin M. Fátima C. Guedes da Silva Matti Haukka João J. R. Fraústo da Silva and Armando J. L. Pombeiro
pg 1569; DOI:
10.1039/b101337h
PDF

Issue 14


Perkin 1 Abstracts: Natural Product Synthesis
Andrew Gunn Jacqueline E. Milne Marcel de Puit and Duncan McArthur
pg 14-xv; DOI:
10.1039/b105193h
PDF
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis
Gideon Grogan Alexis Carstairs Ian Jackson Denise McIntyre Alan Watt Sabine Flitsch and Nicholas Turner
pg 14-ix; DOI:
10.1039/b105469b
PDF
2-Chloro-1,1-dimethyl-1H-cycloprop[e]azulene, the first cyclopropa-fused azulene
Alan D. Payne and Dieter Wege
pg 1579; DOI:
10.1039/b104346n
PDF
Diastereocontrolled Strecker reaction using (S)-5-phenylmorpholin-2-one
Laurence M. Harwood Michael G. B. Drew David J. Hughes and Richard J. Vickers
pg 1581; DOI:
10.1039/b104052a
PDF
Isogalactofagomine lactam. A neutral nanomolar galactosidase inhibitor
Helmer Søhoel Xifu Liang and Mikael Bols
pg 1584; DOI:
10.1039/b103831c
PDF
Preparation of tetraalkylformamidinium salts and related species as precursors to stable carbenes
Roger W. Alder Michael E. Blake Simone Bufali Craig P. Butts A. Guy Orpen Jan Schütz and Stuart J. Williams
pg 1586; DOI:
10.1039/b104110j
PDF
Electrochemical oxidation of aspidofractinine-type alkaloids: Formation of kopsine, kopsidine, kopsinitarine and bisindole derivatives
Toh-Seok Kam Tuck-Meng Lim and Guan-Huat Tan
pg 1594; DOI:
10.1039/b103962h
PDF
Synthesis of nonpolar peptide nucleic acid monomers containing fluoroaromatics
Norio Shibata Biplab Kumar Das Hiroshi Honjo and Yoshio Takeuchi
pg 1605; DOI:
10.1039/b103170h
PDF
C-Glycosylation of tri-O-benzyl-2-deoxy-D-glucose: synthesis of naphthyl-substituted 3,6-dioxabicyclo[3.2.2]nonanes
Margaret A. Brimble and Timothy J. Brenstrum
pg 1612; DOI:
10.1039/b102807n
PDF
Synthesis of a 2-deoxyglucosyl analogue of medermycin
Margaret A. Brimble and Timothy J. Brenstrum
pg 1624; DOI:
10.1039/b103080a
PDF
Scope and limitations in sulfur ylide mediated catalytic asymmetric aziridination of imines: use of phenyldiazomethane, diazoesters and diazoacetamides
Varinder K. Aggarwal Marco Ferrara Christopher J. O'Brien Alison Thompson Ray V. H. Jones and Robin Fieldhouse
pg 1635; DOI:
10.1039/b102578n
PDF
Synthesis of dithiaporphyrin-based singlet–singlet energy transfer systems
Duraisamy Kumaresan Neeraj Agarwal and Mangalampalli Ravikanth
pg 1644; DOI:
10.1039/b102349g
PDF
A general and highly regio and stereoselective method for the synthesis of (E)-2-(2-arylvinyl)-3,1-benzoxathiin-4-ones through palladium–copper catalysis
Bidisha Nandi and Nitya G. Kundu
pg 1649; DOI:
10.1039/b102306n
PDF
The first example of a new type of acyclic, achiral nucleoside analogue: 1-[3-hydroxy-2-(hydroxymethyl)prop-1-enyl]thymine
Daniel Sejer Pedersen Thomas Boesen Anne B. Eldrup Benedikte Kiær Christian Madsen Ulla Henriksen and Otto Dahl
pg 1656; DOI:
10.1039/b101759o
PDF
Synthesis of 6-substituted purin-2-ones with potential cytokinin activity
Geir Andresen Aud Berglen Eriksen Bjørn Dalhus Lise-Lotte Gundersen and Frode Rise
pg 1662; DOI:
10.1039/b101327k
PDF
Design and preparation of serine–threonine protein phosphatase inhibitors based upon the nodularin and microcystin toxin structures. Part 3
Kerri L. Webster Antony B. Maude Michael E. O'Donnell Amit P. Mehrotra and David Gani
pg 1673; DOI:
10.1039/b100401h
PDF
Serine–threonine protein phosphatase inhibitors derived from nodularin: role of the 2-methyl and 3-diene groups in the Adda residue and the effect of macrocyclic conformational restraint
Michael E. O'Donnell Jonathan Sanvoisin and David Gani
pg 1696; DOI:
10.1039/b100402f
PDF
A generic medium throughput activity assay procedure for serine–threonine protein phosphatases using 14C-labelled N-acetyl-Arg-Arg-Ala-Thr(P)-Val-Ala
Jonathan Sanvoisin John R. Pollard Pantea Hormozdiari Walter H. J. Ward and David Gani
pg 1709; DOI:
10.1039/b100403o
PDF
Gal-conjugated anti-rhinovirus agents: chemo-enzymatic syntheses and testing of anti-Gal binding
Yongsheng Chen Wei Zhang Xi Chen Jianqiang Wang and Peng George Wang
pg 1716; DOI:
10.1039/b100356i
PDF

Emanuela Erba Donato Pocar and Pasqualina Trimarco
pg 1723; DOI:
10.1039/b008531f
PDF

Issue 15


Perkin 1 Abstracts: Solid Phase Organic Synthesis
Fabrice Anizon Jennifer Delaney Andrew Gunn Hassan Mamdani Catherine McCusker Fiona McKerlie and Tanya Wildman
pg 15-vii; DOI:
10.1039/b105192j
PDF
Catalytic asymmetric processes
Heather Tye and Paul J. Comina
pg 1729; DOI:
10.1039/a900862d
PDF
Bio-organic synthesis of a newly isolated peptide metastin, metastasis suppressor gene KiSS-1 processing product
Osamu Nishimura Masato Suenaga Takao Yamada Takashi Itoh Nobuyuki Koyama Mitsuhiro Wakimasu Tetsuya Ohtaki Chieko Kitada and Masahiko Fujino
pg 1748; DOI:
10.1039/b104948h
PDF
Unsymmetrically substituted furoxans. Part 18. Smiles rearrangement in furoxan systems and in related furazans
Donatella Boschi Giovanni Sorba Massimo Bertinaria Roberta Fruttero Rosella Calvino and Alberto Gasco
pg 1751; DOI:
10.1039/b104845g
PDF
Intramolecular azomethine ylide cycloaddition reactions to give octahydroindoles
Iain Coldham Katherine M. Crapnell Jonathan D. Moseley and Rémi Rabot
pg 1758; DOI:
10.1039/b104390k
PDF
First efficient synthesis of ()-erythro-roccellic acid
Sivaprakasam Mangaleswaran and Narshinha P. Argade
pg 1764; DOI:
10.1039/b104105n
PDF
Stereoselective syntheses of 1H-imidazo[2,1-a]isoindole-2,5(3H,9bH)-diones
Alan R. Katritzky Yong-Jiang Xu Hai-Ying He and Peter J. Steel
pg 1767; DOI:
10.1039/b104060j
PDF
The first efficient method for the intramolecular trapping of benzynes by phenols: a new approach to xanthenes
David W. Knight and Paul B. Little
pg 1771; DOI:
10.1039/b103834f
PDF
endo/exo Facial selectivities in cycloaddition reactions of substituted 1,2,3-triazolium-1-methanides, unstabilised 1,3-dipoles, with some alkene dipolarophiles: models for 1,2,3-triazolium-1-aminides: new tetracyclic pyrrolo[1,2-c][1,2,3]benzotriazole structures: azolium 1,3-dipoles
R. N. Butler and Leonie M. Wallace
pg 1778; DOI:
10.1039/b103759p
PDF
Atropisomeric -methyl substituted analogues of 4-(dimethylamino)pyridine: synthesis and evaluation as acyl transfer catalysts
Alan C. Spivey Adrian Maddaford David P. Leese and Alison J. Redgrave
pg 1785; DOI:
10.1039/b103385a
PDF
Azafulvenium methides: new extended dipolar systems
Oliver B. Sutcliffe Richard C. Storr Thomas L. Gilchrist and Paul Rafferty
pg 1795; DOI:
10.1039/b103250j
PDF
Xanthen-9-ylidene protecting groups in glycerol chemistry
Colin B. Reese and Hongbin Yan
pg 1807; DOI:
10.1039/b102923c
PDF
Intramolecular cycloadditions of N-alkenoyl aryl azides
Luisa Garanti Giorgio Molteni and Gianluigi Broggini
pg 1816; DOI:
10.1039/b102686k
PDF
Novel synthetic routes to nitrogen-bridged tricyclic derivatives of pyrrolo[2,1,5-cd]indolizine and pyrrolo[2,1,5-de]quinolizine derived from 2-acyl-N-(acylmethyl)pyridinium halides
Jiaxin Hu Xin Jiang Ting He Jian Zhou Yuefei Hu and Hongwen Hu
pg 1820; DOI:
10.1039/b102449n
PDF
A regio- and stereo-selective synthesis of 2-hydroxy-3-methylochromycinone in three steps from 2-bromo-5-acetoxy-1,4-naphthoquinone and 1-acetoxy-3,3-dimethyl-5-vinylcyclohexa-1,5-diene
Tomas Rozek John H. Bowie Simon M. Pyke Brian W. Skelton and Allan H. White
pg 1826; DOI:
10.1039/b101756j
PDF
Asymmetric synthesis of (+)-loline, a pyrrolizidine alkaloid from rye grass and tall fescue
Paul R. Blakemore Sung-Kee Kim Volker K. Schulze James D. White and Alexandre F. T. Yokochi
pg 1831; DOI:
10.1039/b103936a
PDF

Issue 16


Perkin 1 Abstracts: Biocatalysis in Organic Synthesis
Gideon Grogan Alexis Carstairs Ian Jackson Denise McIntyre Alan Watt Sabine Flitsch and Nicholas Turner
pg 16-vii; DOI:
10.1039/b106521c
PDF
Perkin 1 Abstracts: Natural Product Synthesis
Andrew Gunn Jacqueline E. Milne Marcel de Puit and Duncan McArthur
pg 16-xiii; DOI:
10.1039/b106740k
PDF
A concise and efficient stereoselective synthesis of protected (2R,1S,2S)-2-(carboxycyclopropyl)glycine (D-CCG-I)
Debendra K. Mohapatra
pg 1851; DOI:
10.1039/b105503h
PDF
Synthesis of 2-heteroaryl-3-hydroxypyridines by ring expansion reactions of 2-acylfurans with ammonia
Richard W. J. Chubb Martin R. Bryce and Brian Tarbit
pg 1853; DOI:
10.1039/b105228b
PDF
A conformationally locked tricyclic nucleoside. Synthesis, crystal structure and incorporation into oligonucleotides
Jacob Ravn Niels Thorup and Poul Nielsen
pg 1855; DOI:
10.1039/b104438a
PDF
Carotenoids and related polyenes. Part 6. Stereoselective synthesis of astaxanthin analogues and their antioxidant activities
Yumiko Yamano Yuki Sato Yasuko Watanabe Koshi Namikawa Wataru Miki and Masayoshi Ito
pg 1862; DOI:
10.1039/b104338m
PDF
Synthesis of novel all-cis-functionalized cyclopropane template-assembled collagen models
Shoko Yamazaki Mari Sakamoto Michiko Suzuri Masamitsu Doi Takashi Nakazawa and Yuji Kobayashi
pg 1870; DOI:
10.1039/b103887g
PDF
Direct synthesis of Fmoc-protected amino acids using organozinc chemistry: application to polymethoxylated phenylalanines and 4-oxoamino acids
Hervé J. C. Deboves Christian A. G. N. Montalbetti and Richard F. W. Jackson
pg 1876; DOI:
10.1039/b103832j
PDF
Stereoselective Baeyer–Villiger oxidation of some bridged bicyclic diketones
Eugenius Butkus and Sigitas Stonius
pg 1885; DOI:
10.1039/b103564a
PDF
A new route to polyoxygenate C and D rings of steroids by oxidation of a 8,14-diene steroid with the methyltrioxorhenium–H2O2–urea system
Donato Sica Domenica Musumeci Franco Zollo and Simona De Marino
pg 1889; DOI:
10.1039/b103389c
PDF
Trapping highly reactive dipolarophiles. Exploiting the mechanism associated with the azomethine ylide strategy for -lactam synthesis
Giles A. Brown Kirsty M. Anderson Jonathan M. Large Denis Planchenault Dominique Urban Neil J. Hales and Timothy Gallagher
pg 1897; DOI:
10.1039/b103271m
PDF
Synthesis, structure, and reactivity of (tropon-2-ylimino)arsorane and in situ generation of its stiborane and -bismuthorane analogues: reactions with heterocumulenes and an activated acetylene giving heteroazulenes
Makoto Nitta Yuhki Mitsumoto and Hiroyuki Yamamoto
pg 1901; DOI:
10.1039/b103098c
PDF
Synthesis and properties of 2-nitrosoadenosine
Martin J. Wanner and Gerrit-Jan Koomen
pg 1908; DOI:
10.1039/b102897a
PDF
Enantioselective synthesis of -hydroxy amines and aziridines using asymmetric transfer hydrogenation of -amino ketones
Aparecida M. Kawamoto and Martin Wills
pg 1916; DOI:
10.1039/b102895m
PDF
Chemical consequences of fluorine substitution. Part 1. Experimental and theoretical results on Diels–Alder reactions of - and -fluorostyrenes
Thomas Ernet Andreas H. Maulitz Ernst-Ulrich Würthwein and Günter Haufe
pg 1929; DOI:
10.1039/b102684b
PDF
Ultrasound-accelerated synthesis of 3,4-dihydropyrimidin-2(1H)-ones with ceric ammonium nitrate
Jhillu S. Yadav Basi V. Subba Reddy Kasireddy Bhaskar Reddy Kavuda Sarita Raj and Attaluri R. Prasad
pg 1939; DOI:
10.1039/b102565c
PDF
The syntheses of three highly unsaturated marine lipid hydrocarbons
Anne Kristin Holmeide Lars Skattebøl and Magne Sydnes
pg 1942; DOI:
10.1039/b101889m
PDF
Ketoester methacrylate resin, secondary amine clean-up in the presence of primary amines
Zhanru Yu Sonia Alesso David Pears Paul A. Worthington Richard W. A. Luke and Mark Bradley
pg 1947; DOI:
10.1039/b101395p
PDF
One-pot synthesis of unsymmetrical biaryls from suitably functionalized 2H-pyran-2-ones through carbanion-induced ring-transformation reactions
Vishnu J. Ram Pratibha Srivastava Nidhi Agarwal Ashoke Sharon and Prakas R. Maulik
pg 1953; DOI:
10.1039/b009725j
PDF
A novel system for the preparation of orphan receptor ligand peptides
Osamu Nishimura Nobuyuki Koyama Takashi Itoh Masato Suenaga Takeo Moriya Masanori Miwa Yoko Tanaka Chieko Kitada and Masahiko Fujino
pg 1960; DOI:
10.1039/b009566o
PDF

Issue 17


Perkin 1 Abstracts: Solid Phase Organic Synthesis
Fabrice Anizon Jennifer Delaney Andrew Gunn Hassan Mamdani Catherine McCusker Fiona McKerlie and Tanya Wildman
pg 17-vii; DOI:
10.1039/b106738a
PDF
Generation and reactivity of -metalated vinyl ethers
Richard W. Friesen
pg 1969; DOI:
10.1039/b104589j
PDF
-Allyl cation cyclisations initiated by electrocyclic ring-opening of gem-dihalocyclopropanes: application to the first total syntheses of the crinine-type alkaloids maritinamine and epi-maritinamine
Martin G. Banwell Joanne E. Harvey and Katrina A. Jolliffe
pg 2002; DOI:
10.1039/b106369n
PDF
Is N-acetylornithine aminotransferase the real N-succinyl-LL-diaminopimelate aminotransferase in Escherichia coli and Mycobacterium smegmatis?
Russell J. Cox and Paul S. H. Wang
pg 2006; DOI:
10.1039/b106146c
PDF
Oxidations of 3-alkenyltetronic acids with dimethyldioxirane (DMD) and air: regioselectivity and formation of a spirotricyclic hemiketal endoperoxide lactone
Rainer Schobert Sven Siegfried Jochen Weingärtner and Mark Nieuwenhuyzen
pg 2009; DOI:
10.1039/b104227k
PDF
Cyclic ureas as ortho directing substituents
Jon-Paul Meigh Mercedes Álvarez and John A. Joule
pg 2012; DOI:
10.1039/b105420c
PDF
Synthesis and in vitro enzyme activity of aza, oxa and thia derivatives of bacterial cell wall biosynthesis intermediates
Russell J. Cox and Paul S. H. Wang
pg 2022; DOI:
10.1039/b105117m
PDF
Acid- or base-promoted photostimulated homolytic tert-butylation of pyridines and thiophenes
Byeong Hyo Kim Insik Jeon Tae Hee Han Hae Jin Park and Young Moo Jun
pg 2035; DOI:
10.1039/b104906m
PDF
Chiral synthons from carvone. Part 50. Enantiospecific approaches to both enantiomers of bicyclo[4.3.0]nonane-3,8-dione derivatives
A. Srikrishna and T. Jagadeeswar Reddy
pg 2040; DOI:
10.1039/b104253j
PDF
An alternative approach to the synthesis of a recombinant galanin-like peptide (GALP)
Takashi Itoh Nobuyuki Koyama Masanori Miwa Masato Suenaga Tetsuya Ohtaki Chieko Kitada Osamu Nishimura and Masahiko Fujino
pg 2047; DOI:
10.1039/b103835b
PDF
Friedel–Crafts reactions of a sulfonyl-substituted vinylic epoxide with various aromatics
Svante Brandänge Jan-Erling Bäckvall and Hans Leijonmarck
pg 2051; DOI:
10.1039/b103582g
PDF
Influence of ring size on the outcome of sulfide contraction reactions with thiolactams. Isolation of bicyclic ketene S,N-acetals and thioisomnchnones
Joseph P. Michael Charles B. de Koning Christiaan W. van der Westhuyzen and Manuel A. Fernandes
pg 2055; DOI:
10.1039/b103560f
PDF
Synthesis of glycero amino acid-based surfactants. Part 1. Enzymatic preparation of rac-1-O-(N-acetyl-L-aminoacyl)glycerol derivatives
Carmen Morán María Rosa Infante and Pere Clapés
pg 2063; DOI:
10.1039/b103132p
PDF
Synthesis of imines, diimines and macrocyclic diimines as possible ligands, in aqueous solution
Alina Simion Cristian Simion Tadeshige Kanda Satoko Nagashima Yoshiharu Mitoma Tomoko Yamada Keisuke Mimura and Masashi Tashiro
pg 2071; DOI:
10.1039/b102749m
PDF
An efficient approach to (E)--methyl Baylis–Hillman adducts via indium-mediated allylation of aldehydes in aqueous media
Joo Hwan Cha Ae Nim Pae Kyung Il Il Choi Yong Seo Cho Hun Yeong Koh and Eun Lee
pg 2079; DOI:
10.1039/b102532p
PDF
Highly peri- and stereoselective intramolecular photocycloaddition and cyclisation of N-(1-naphthylethyl)prop-2-enamides
Shigeo Kohmoto Yoshiyuki Miyaji Masaru Tsuruoka Keiki Kishikawa Makoto Yamamoto and Kazutoshi Yamada
pg 2082; DOI:
10.1039/b100678i
PDF
Medium-sized cyclophanes. Part 58. Synthesis and conformational studies of [2.n]metacyclophan-1-enes and [n.1]metacyclophanes
Takehiko Yamato Koji Fujita and Hirohisa Tsuzuki
pg 2089; DOI:
10.1039/b010075g
PDF
Isolation, structure and synthesis of mahafacyclin B, a cyclic heptapeptide from the latex of Jatropha mahafalensis
Carine Baraguey Alain Blond Florine Cavelier Jean-Louis Pousset Bernard Bodo and Catherine Auvin-Guette
pg 2098; DOI:
10.1039/b008538n
PDF

Issue 18


Perkin 1 Abstracts: Biocatalysis in Organic Synthesis
Gideon Grogan Alexis Carstairs Ian Jackson Denise McIntyre Alan Watt Sabine Flitsch and Nicholas Turner
pg 18-ix; DOI:
10.1039/b107562b
PDF
Perkin 1 Abstracts: Natural Product Synthesis
Andrew Gunn Jacqueline E. Milne Marcel de Puit and Duncan McArthur
pg 18-xv; DOI:
10.1039/b107661m
PDF
Protecting groups
Krzysztof Jarowicki and Philip Kocienski
pg 2109; DOI:
10.1039/b103282h
PDF
Garner's aldehyde
Xifu Liang Jens Andersch and Mikael Bols
pg 2136; DOI:
10.1039/b101054i
PDF
First highly stereoselective synthesis of (+)-dihydrosesamin, a trisubstituted tetrahydrofuran-type of lignan, by using highly erythro-selective aldol condensation
Satoshi Yamauchi Teruhisa Tanaka and Yoshiro Kinoshita
pg 2158; DOI:
10.1039/b105419h
PDF
Functionalised bicyclic alcohols by enantioselective -deprotonation–rearrangement of meso-epoxides
David M. Hodgson Iain D. Cameron Martin Christlieb Rebecca Green Gary P. Lee and Lesley A. Robinson
pg 2161; DOI:
10.1039/b105369h
PDF
DISAL glycosyl donors for efficient glycosylations under acidic conditions: Application to solid-phase oligosaccharide synthesis
Lars Petersen and Knud J. Jensen
pg 2175; DOI:
10.1039/b105872j
PDF
Double intramolecular hetero Diels–Alder reactions of ,-unsaturated hydrazones as 1-azadienes: a new route to 2,2-bipyridines
Nicholas Bushby Christopher J. Moody David A. Riddick and Ian R. Waldron
pg 2183; DOI:
10.1039/b105409k
PDF
A chemoenzymatic synthesis of the carbobicyclic core associated with CP-225,917 and CP-263,114 (phomoidrides A and B)
Martin G. Banwell Kenneth J. McRae and Anthony C. Willis
pg 2194; DOI:
10.1039/b105376k
PDF
Studies related to carba-pyranoses: a strategy for the synthesis of -1,3-glycosidically linked aminomonocarba-disaccharides
David S. Larsen Roger J. Lins Richard J. Stoodley and Nicholas S. Trotter
pg 2204; DOI:
10.1039/b105374b
PDF
Synthesis of ellipticine by reaction of 1-(4-methoxybenzyl)indole-2,3-dicarboxylic anhydride with (3-bromo-4-pyridyl)triisopropoxytitanium
Yasuyoshi Miki Hiroko Hachiken and Norihide Yanase
pg 2213; DOI:
10.1039/b105116b
PDF
The first stereospecific synthesis of L-tetrahydrodipicolinic acid; a key intermediate of diaminopimelate metabolism
Jennifer F. Caplan Andrew Sutherland and John C. Vederas
pg 2217; DOI:
10.1039/b105091p
PDF
One-step iodination of the diazocyclopentadien-2-ylcarbonyl group—a new and convenient preparation of effective radiolabelled photoaffinity probes
Elena L. Vodovozova Ekaterina V. Tsibizova and Julian G. Molotkovsky
pg 2221; DOI:
10.1039/b104945n
PDF
A highly efficient, stereoselective oxyfunctionalization of unactivated carbons in steroids with dimethyldioxirane
Takashi Iida Takeru Yamaguchi Ryusei Nakamori Masahiro Hikosaka Nariyasu Mano Junichi Goto and Toshio Nambara
pg 2229; DOI:
10.1039/b104938k
PDF
Synthesis of a thiophene analogue of kuanoniamine A
Yvette A. Jackson Seon A. Hepburn and William F. Reynolds
pg 2237; DOI:
10.1039/b104710h
PDF
Allene synthesis by an asymmetric Baylis–Hillman style reaction on vinylphosphine oxides
David J. Fox Jonathan A. Medlock Richard Vosser and Stuart Warren
pg 2240; DOI:
10.1039/b104436m
PDF
Intramolecular [2+2] photocycloadditions as an approach towards the right-hand side of solanoeclepin A
Richard H. Blaauw Jorg C. J. Benningshof Angeline E. van Ginkel Jan H. van Maarseveen and Henk Hiemstra
pg 2250; DOI:
10.1039/b104165g
PDF
[2 + 2] Cycloaddition reaction of cycloheptatriene with dichloroketene. A novel and efficient synthetic strategy for the synthesis of 2-hydroxyazulene
Ryuji Yokoyama Shunji Ito Masataka Watanabe Nobuyuki Harada Chizuko Kabuto and Noboru Morita
pg 2257; DOI:
10.1039/b104164a
PDF
Highly selective one-pot conversion of THP and MOM ethers to acetates by indium triiodide-catalysed deprotection and subsequent transesterification by ethyl acetate
Brindaban C. Ranu and Alakananda Hajra
pg 2262; DOI:
10.1039/b104055n
PDF
Chemoselectivity in reactions of an -diazo--diketone with some conjugative double-bond systems
Jiaxi Xu Qihan Zhang Liangbi Chen and Hui Chen
pg 2266; DOI:
10.1039/b103173m
PDF
Synthesis and thermal transformation of stable monocyclic 4-thiabenzenes
Hiroshi Shimizu Noriaki Kudo Tadashi Kataoka and Mikio Hori
pg 2269; DOI:
10.1039/b102806p
PDF
Oxidative radical cyclizations of malonate enolates induced by the ferrocenium ion – a remarkable influence of enolate counterion and additives
Ullrich Jahn and Philip Hartmann
pg 2277; DOI:
10.1039/b102211n
PDF
Regio- and stereoselective synthesis of fluoroalkadienes using -fluoroalkenyliodonium salt
Masanori Yoshida Dai Nagahara Tsuyoshi Fukuhara Norihiko Yoneda and Shoji Hara
pg 2283; DOI:
10.1039/b101836l
PDF
An efficient synthesis of julibrosides related to neosaponin
Yuguo Du Meimei Zhang and Fanzuo Kong
pg 2289; DOI:
10.1039/b009955o
PDF
Efficient formation of lipophilic dihydroxotin(IV) porphyrins and bis-porphyrins
Maxwell J. Crossley Pall Thordarson and Richard A.-S. Wu
pg 2294; DOI:
10.1039/b104846p
PDF

Issue 19


Perkin 1 Abstracts: Solid Phase Organic Synthesis
Jennifer Delaney Andrew Gunn Hassan Mamdani and Tanya Wildman
pg 19-ix; DOI:
10.1039/b107265j
PDF
Saturated oxygen heterocycles
Mark C. Elliott and Eve Williams
pg 2303; DOI:
10.1039/b007290g
PDF
Novel and facile catalytic synthesis of 2,4-dioxopyrido[2,3-d]pyrimidine derivatives in water
Noé Rosas Pankaj Sharma Cecilio Alvarez Armando Cabrera Rodrigo Ramírez Alejandro Delgado and Henri Arzoumanian
pg 2341; DOI:
10.1039/b101374m
PDF
Enantiospecific syntheses of pseudopterosin aglycones. Part 1. Synthesis of the putative aglycone of pseudopterosin G–J via an AABABC annulation strategy
Robert Chow Philip J. Kocienski Alexander Kuhl Jean-Yves LeBrazidec Kenneth Muir and Paul Fish
pg 2344; DOI:
10.1039/b102960f
PDF
Enantiospecific syntheses of pseudopterosin aglycones. Part 2. Synthesis of pseudopterosin K–L aglycone and pseudopterosin A–F aglycone via a BBABAC annulation strategy
Philip J. Kocienski Alessandro Pontiroli and Liu Qun
pg 2356; DOI:
10.1039/b102961b
PDF
Unusual stereoselectivity in the alkylation of pyroglutamate ester urethanes
Jean-Damien Charrier James E. S. Duffy Peter B. Hitchcock and Douglas W. Young
pg 2367; DOI:
10.1039/b106451g
PDF
Synthesis of epibatidine isomers: endo-5- and 6- (6-chloro-3-pyridyl-2-azabicyclo[2.2.1]heptanes
Caroline D. Cox John R. Malpass John Gordon and Alan Rosen
pg 2372; DOI:
10.1039/b106212n
PDF
A concise C-glycosyl amino acid synthesis by alkenyl C-glycoside–vinyloxazolidine cross-metathesis. Synthesis of glycosyl serine, asparagine and hydroxynorvaline isosteres
Alessandro Dondoni Pier Paolo Giovannini and Alberto Marra
pg 2380; DOI:
10.1039/b106029p
PDF
An improved, versatile synthesis of the GABAC antagonists (1,2,5,6-tetrahydropyridin-4-yl)methylphosphinic acid (TPMPA) and (piperidin-4-yl)methylphosphinic acid (P4MPA)
Jane R. Hanrahan Kenneth N. Mewett Mary Chebib Peter M. Burden and Graham A. R. Johnston
pg 2389; DOI:
10.1039/b105989k
PDF
Three-component synthesis of (E)-,-unsaturated amides of the piperine family
Rainer Schobert Sven Siegfried and Gary J. Gordon
pg 2393; DOI:
10.1039/b105745f
PDF
Simple and selective one-pot replacement of the N-methyl group of tertiary amines by quaternization and demethylation with sodium sulfide or potassium thioacetate: an application to the synthesis of pergolide
Luigi Anastasia Giuliana Cighetti and Pietro Allevi
pg 2398; DOI:
10.1039/b104843k
PDF
A practical protocol for the synthesis of 3-hydroxy-4,5-disubstituted pyridine derivatives from acyclic compounds
Luigi Anastasia Mario Anastasia and Pietro Allevi
pg 2404; DOI:
10.1039/b105478n
PDF
Synthesis of bis[1,2]dithiolo[1,4]thiazine imines from Hnig's base
Stanislav A. Amelichev Susana Barriga Lidia S. Konstantinova Tatjana B. Markova Oleg A. Rakitin Charles W. Rees and Tomás Torroba
pg 2409; DOI:
10.1039/b105243h
PDF
Synthesis and stereochemistry of new tetraspiro-1,3-dioxanes
Dorina Opris Ion Grosu Loïc Toupet Gérard Plé Anamaria Terec Sorin Mager and Luminita Muntean
pg 2413; DOI:
10.1039/b104604g
PDF
Synthesis of 6,7-dehydroartemisinic acid
Lai-King Sy and Geoffrey D. Brown
pg 2421; DOI:
10.1039/b104471k
PDF
Retinoids and related compounds. Part 26. Synthesis of (11Z)-8,18-propano- and methano-retinals and conformational study of the rhodopsin chromophore
Akimori Wada Masako Tsutsumi Yuka Inatomi Hiroo Imai Yoshinori Shichida and Masayoshi Ito
pg 2430; DOI:
10.1039/b104394n
PDF
Synthesis and catalytic properties of p-acylthio(phenylacetylene)n substituted chiral manganese salen complexes
Morten Nielsen and Kurt V. Gothelf
pg 2440; DOI:
10.1039/b104103g
PDF
Stereoselective synthesis of a set of two functionalized (E)-alkene dipeptide isosteres of L-amino acid-L-Glu and L-amino acid-D-Glu
Shinya Oishi Hirokazu Tamamura Masaki Yamashita Yoshihiko Odagaki Nobuyuki Hamanaka Akira Otaka and Nobutaka Fujii
pg 2445; DOI:
10.1039/b103833h
PDF
Selective radical-chain epimerisation at electron-rich chiral tertiary C–H centres using thiols as protic polarity-reversal catalysts
Hai-Shan Dang Brian P. Roberts and Derek A. Tocher
pg 2452; DOI:
10.1039/b103558b
PDF
Novel phosphitylating reagents containing a phosphorus–fluorine bond and their application in efficient synthesis of phosphorofluoridates and phosphorofluoridothionates
Wojciech Dbkowski and Izabela Tworowska
pg 2462; DOI:
10.1039/b103082p
PDF
Studies on polycyclic fluoroazaarenes: synthesis of trans-9-fluoro- and -11-fluoro 3,4-dihydroxy-3,4-dihydrobenz[c]acridines as potential proximate carcinogenic metabolites of fluorobenz[c]acridine
Dipanjan Pan Gandhi K. Kar Jayanta K. Ray Jyh-Ming Lin Shantu Amin Suchada Chantrapromma and Hoong-Kun Fun
pg 2470; DOI:
10.1039/b102750f
PDF
The photochemical reactions of nitrogen-rich mesoionic 1,3-diphenyltetrazolium heterocycles and related compounds
Shuki Araki Hiromi Hattori Koji Ogawa Masashi Kuzuya Tomoko Inoue Hatsuo Yamamura and Masao Kawai
pg 2476; DOI:
10.1039/b009526p
PDF
Preparation and synthetic utility of 3-(benzotriazol-1-ylmethyl)areno- and -hetareno[b]thiophenes
Alan R. Katritzky Vladimir Y. Vvedensky and Dmytro O. Tymoshenko
pg 2483; DOI:
10.1039/b008612f
PDF

Issue 20


Perkin 1 Abstracts: Biocatalysis in Organic Synthesis
Gideon Grogan Alexis Carstairs Ian Jackson Denise McIntyre Alan Watt Sabine Flitsch and Nicholas Turner
pg 20-xi; DOI:
10.1039/b108606p
PDF
Perkin 1 Abstracts: Natural Product Synthesis
Andrew Gunn Jacqueline E. Milne Marcel de Puit and Duncan McArthur
pg 20-xvi; DOI:
10.1039/b108756h
PDF
Synthesis of aromatic heterocycles
Thomas L. Gilchrist
pg 2491; DOI:
10.1039/a904578c
PDF
Rapid assembly of anti,anti-1,2,3-triol motifs via stereoselective addition of organometallics to aldehydes obtained from (R,R,S,R)-2,3-butane diacetal protected butanetetraol derivatives
Darren J. Dixon Lars Krause and Steven V. Ley
pg 2516; DOI:
10.1039/b105118k
PDF
Highly stereocontrolled reduction of an alkynyl ketone possessing a 1,3-dithianyl moiety using oxazaborolidine–BH3
Makoto Shimizu Yoshiyuki Ikari and Akinobu Wakabayashi
pg 2519; DOI:
10.1039/b107604c
PDF
Lewis-acid catalysed arylation of the hydroxyamino sugar moiety of the natural product SB-219383
John M. Berge Catherine S. V. Houge-Frydrych and Richard L. Jarvest
pg 2521; DOI:
10.1039/b105965n
PDF
Synthesis of a conformationally rigid scyllo-inositol polymer as a novel chelating ligand
Tae-Hyun Kim and Andrew B. Holmes
pg 2524; DOI:
10.1039/b105105a
PDF
Transition metal complexes as linkers for solid phase synthesis: chromium carbonyl complexes as linkers for arenes
Alex C. Comely Susan E. Gibson (née Thomas) Neil J. Hales and Mark A. Peplow
pg 2526; DOI:
10.1039/b106582n
PDF
Facile synthesis of 6-cyano-9-substituted-9H-purines and their ring expansion to 8-(arylamino)-4-imino-3-methylpyrimidino[5,4-d]pyrimidines
Amal Al-Azmi Brian L. Booth Robert A. Carpenter Alice Carvalho Elodie Marrelec Robin G. Pritchard and M. Fernanda J. R. P. Proença
pg 2532; DOI:
10.1039/b106539b
PDF
Ring fused 1,2,5-thiadiazoles from oximes and trithiazyl trichloride
Charles W. Rees and Tai-Yuen Yue
pg 2538; DOI:
10.1039/b106384g
PDF
Synthesis of spiro-indanes by cycloaddition strategy
Sambasivarao Kotha and Ethirajan Manivannan
pg 2543; DOI:
10.1039/b106280h
PDF
Polyaromatic amines. Part 2. Synthesis of 4,4,4-tris(N-aryl-N-phenylamino)triphenylamine, N,N-bis[4-(N-aryl-N-phenylamino)phenyl]tolylamine and N,N,N,N-tetraaryl-o-phenylenediamine derivatives
M. John Plater and Toby Jackson
pg 2548; DOI:
10.1039/b106273p
PDF
The synthesis and evaluation of o-phenylenediamine derivatives as fluorescent probes for nitric oxide detection
M. John Plater Iain Greig Miep H. Helfrich and StuartH. Ralston
pg 2553; DOI:
10.1039/b105953j
PDF
A general -cyanoformylation using -litho--ethoxyacrylonitrile: application to the syntheses of new 6-cyano-2,4-bis(phenylthio)- and 4-cyano-2,6-bis(phenylthio)hepta-2,4,6-trienals
Mitsuhiro Yoshimatsu Sachiko Yamaguchi and Yoshiaki Matsubara
pg 2560; DOI:
10.1039/b105894k
PDF
Diazoketones as precursors in -lactam synthesis. New insights into the mechanism of the photochemically induced Staudinger reaction
Michael R. Linder Wolfgang U. Frey and Joachim Podlech
pg 2566; DOI:
10.1039/b105748k
PDF
Efficient and convenient entry to -hydroxy--trifluoromethyl--substituted ketones and 2,6-disubstituted 4-trifluoromethylpyridines based on the reaction of trifluoromethyl ketones with enamines or imines
Kazumasa Funabiki Akie Isomura Yoshihiro Yamaguchi Wataru Hashimoto Kei Matsunaga Katsuyoshi Shibata and Masaki Matsui
pg 2578; DOI:
10.1039/b105636k
PDF
Vilsmeier–Haack reaction of tertiary alcohols: formation of functionalised pyridines and naphthyridines
Ajith Dain Thomas and Chitoorthekkathil V. Asokan
pg 2583; DOI:
10.1039/b105634b
PDF
Synthesis of dihydrobenzazaphosphole ligands via an intramolecular cyclisation reaction
Wilson Leung Sarah Cosway Raymond H. V. Jones Hannah McCann and Martin Wills
pg 2588; DOI:
10.1039/b105495n
PDF
Optimisation of substitution at the 2- and 5- positions of 3,4-dialkoxythiophenes via the Mannich reaction: the influences of steric crowding, electrophile reactivity and temperature
Joan Halfpenny Phillip B. Rooney and Zachary S. Sloman
pg 2595; DOI:
10.1039/b105476g
PDF
Synthesis and evaluation of a broad range of chiral sulfides for asymmetric sulfur ylide epoxidation of aldehydes
Varinder K. Aggarwal Rémy Angelaud Dominique Bihan Paul Blackburn Robin Fieldhouse Silvia J. Fonquerna Gair D. Ford George Hynd Elfyn Jones Ray V. H. Jones Philippe Jubault Matthew J. Palmer Paul D. Ratcliffe and Harry Adams
pg 2604; DOI:
10.1039/b105416n
PDF
Diastereoselective synthesis of 2-alkylated 4-silyloxyproline esters
Tatsunori Sato Satomi Kawasaki Nobuo Oda Shôko Yagi Serry A. A. El Bialy Jun'ichi Uenishi Masashige Yamauchi and Masazumi Ikeda
pg 2623; DOI:
10.1039/b105238c
PDF
-Aminophosphonic compounds derived from methyl 1-dimethoxyphosphoryl-2-succinimidocyclohex-3-ene-1-carboxylates
Nathalie Defacqz Roland Touillaux Alex Cordi and Jacqueline Marchand-Brynaert
pg 2632; DOI:
10.1039/b105111n
PDF
Reusable solid-phase supports for oligonucleotides and antisense therapeutics
Richard T. Pon Shuyuan Yu Zhiqiang Guo Ranjit Deshmukh and Yogesh S. Sanghvi
pg 2638; DOI:
10.1039/b105089n
PDF
Synthetic studies toward the kempane diterpenes. Diels–Alder additions to bicyclic dienes
Chunjian Liu Guanglin Bao and D. Jean Burnell
pg 2644; DOI:
10.1039/b104924k
PDF
Synthetic studies toward the kempane diterpenes. Approaches to the assembly of the ring system
Guanglin Bao Chunjian Liu and D. Jean Burnell
pg 2657; DOI:
10.1039/b104986k
PDF
The synthesis and structural characterisation of some azo-containing phosphine chalcogenides and comparison to non-phosphorus-containing analogues
Mark J. Alder Vanessa M. Bates Wendy I. Cross Kevin R. Flower and Robin G. Pritchard
pg 2669; DOI:
10.1039/b104918f
PDF
Stereochemistry of enacyloxins. Part 3. (12S,17R,18S,19R)-Absolute configuration of enacyloxins, a series of antibiotics from Frateuria sp. W-315
Ryo Takeuchi Hiromasa Kiyota Manabu Yaosaka Toshihiko Watanabe Keijiro Enari Takeyoshi Sugiyama and Takayuki Oritani
pg 2676; DOI:
10.1039/b104341m
PDF
Optimisation of the allylsilane approach to C-10 deoxo carba analogues of dihydroartemisinin: synthesis and in vitro antimalarial activity of new, metabolically stable C-10 analogues
Paul M. O'Neill Matthew Pugh Andrew V. Stachulski Stephen A. Ward Jill Davies and B. Kevin Park
pg 2682; DOI:
10.1039/b104340b
PDF
Epimerization of peptide nucleic acids analogs during solid-phase synthesis: optimization of the coupling conditions for increasing the optical purity
Roberto Corradini Stefano Sforza Arnaldo Dossena Gerardo Palla Raniero Rocchi Ferdinando Filira Flavia Nastri and Rosangela Marchelli
pg 2690; DOI:
10.1039/b104146k
PDF
Stereocontrolled construction of rigid tricyclic bis(-amino acid) derivatives by Ru(II)-catalyzed cascade and Diels–Alder reactions
Jon Efskind Christian Römming and Kjell Undheim
pg 2697; DOI:
10.1039/b103254m
PDF
Reactions of 1-(2-alkoxyphenyl)alkaniminyl radicals
Rino Leardini Hamish McNab Matteo Minozzi Daniele Nanni David Reed and Andrew G. Wright
pg 2704; DOI:
10.1039/b103181n
PDF
Aldol-type condensation reactions of lithium eneselenolates generated from selenoamides with aldehydes
Toshiaki Murai Akiko Suzuki and Shinzi Kato
pg 2711; DOI:
10.1039/b100198l
PDF
Molecular recognition of xanthine alkaloids: First synthetic receptors for theobromine and a series of new receptors for caffeine
Shyamaprosad Goswami Ajit Kumar Mahapatra and Reshmi Mukherjee
pg 2717; DOI:
10.1039/b009319j
PDF

Issue 21


Perkin 1 Abstracts: Solid Phase Organic Synthesis
Jennifer Delaney Andrew Gunn and Tanya Wildman
pg 21-vii; DOI:
10.1039/b109264m
PDF
Recent developments in lanthanide mediated organic synthesis
Patrick G. Steel
pg 2727; DOI:
10.1039/a908189e
PDF
A novel approach to the synthesis of mono- and dipyrroloporphyrins
Ana M. G. Silva Maria A. F. Faustino Augusto C. Tomé Maria G. P. M. S. Neves Artur M. S. Silva and José A. S. Cavaleiro
pg 2752; DOI:
10.1039/b108783p
PDF
Reductive cyclization with baker's yeast of 4-alkyl-2-nitroacetanilides to 6-alkylbenzimidazoles and 1-hydroxy-2-methyl-6-alkylbenzimidazoles
Arturo Navarro-Ocaña Luís F. Olguín Hector Luna Manuel Jiménez-Estrada and Eduardo Bárzana
pg 2754; DOI:
10.1039/b107492j
PDF
Synthesis of (3R,6R)- and (3S,6R)-piperidinone PNA
Ask Püschl Thomas Boesen Tullia Tedeschi Otto Dahl and Peter E. Nielsen
pg 2757; DOI:
10.1039/b103901f
PDF
A bioisosteric oligosaccharide mimetic based on isofagomine-type monomers
Xifu Liang Bent O. Petersen Jens Ø. Duus and Mikael Bols
pg 2764; DOI:
10.1039/b103756k
PDF
Reactions of thiobenzoylketene S,N-acetals with silyl enol ethers of cyclic ketones in the presence of desilylating reagents: formation and desulfurization of thienolactams
Jong Seok Lee Dong Joon Lee Bo Sung Kim and Kyongtae Kim
pg 2774; DOI:
10.1039/b102922n
PDF
A novel synthesis of imidazoles via the cycloaddition of nitrile ylides to their imidoyl chloride precursors
Paul W. Groundwater Ian Garnett Andrew J. Morton Toqir Sharif Simon J. Coles Michael B. Hursthouse Miklos Nyerges Rosaleen J. Anderson David Bendell Alexander McKillop and Weimin Zhang
pg 2781; DOI:
10.1039/b104130b
PDF
Polyhalogenated heterocyclic compounds. Part 47. Syntheses of multi-substituted pyridine derivatives from pentafluoropyridine
Richard D. Chambers Philip R. Hoskin Graham Sandford Dmitrii S. Yufit and Judith A. K. Howard
pg 2788; DOI:
10.1039/b105950p
PDF
Reactive immunization elicits catalytic antibodies for polyester hydrolysis
Da-Wei Chen Robert J. Kubiak Jon A. Ashley and Kim D. Janda
pg 2796; DOI:
10.1039/b105412k
PDF
Diastereoselective Lewis acid mediated hydrophosphonylation of heterocyclic imines: a stereoselective approach towards -amino phosphonates
Imre Schlemminger Andreas Willecke Wolfgang Maison Rainer Koch Arne Lützen and Jürgen Martens
pg 2804; DOI:
10.1039/b101501j
PDF
Cycloaddition of nitrile imines to resin-bound enamines: a solid phase synthesis of 1,4-diarylpyrazoles
Andrew C. Donohue Sue Pallich and Tom D. McCarthy
pg 2817; DOI:
10.1039/b102913b
PDF
Synthesis of bisquaraine dyes. Novel homologues of 1,2-squaraines bearing symmetrical and unsymmetrical structures
Yutaka Hyodo Hiroyuki Nakazumi Shigeyuki Yagi and Kazuhisa Nakai
pg 2823; DOI:
10.1039/b104059f
PDF
Development of catalysts for the Baylis–Hillman reaction: the application of tetramethylguanidine and attempts to use a supported analogue
Nicholas E. Leadbeater and Cornelia van der Pol
pg 2831; DOI:
10.1039/b106267k
PDF
Convenient preparations of polysubstituted 3H-pyrroles promoted by SmI2
Xiaoliang Xu and Yongmin Zhang
pg 2836; DOI:
10.1039/b102268g
PDF
Synthesis and applications to asymmetric catalysis of a series of mono- and bis(diazaphospholidine) ligands
Donald Smyth Heather Tye Colin Eldred Nathaniel W. Alcock and Martin Wills
pg 2840; DOI:
10.1039/b106399p
PDF
Synthesis of (R)-{6-[O-methyl-N-(-methylbenzyl)hydroxyamino]benzene} chromium tricarbonyl via nucleophilic aromatic substitution of (6-fluorobenzene) chromium tricarbonyl
M. Rute G. da Costa M. João M. Curto Stephen G. Davies John Sanders and Fátima C. Teixeira
pg 2850; DOI:
10.1039/b107237b
PDF
Lithium–potassium superbases as key reagents for the base-catalysed isomerisation of some terpenoids
Annamaria Deagostino Paolo Balma Tivola Cristina Prandi and Paolo Venturello
pg 2856; DOI:
10.1039/b106906c
PDF
Intramolecular epoxidation in unsaturated ketones and oxaziridines
Alan Armstrong and Alistair G. Draffan
pg 2861; DOI:
10.1039/b107839a
PDF
The synthesis of 5-substituted proline derivatives and of 5-substituted pyrrole-2-carboxylates by 5-endo cyclisations featuring a method for effectively favouring these with respect to 5-exo cyclisations
David W. Knight Adele L. Redfern and Jeremy Gilmore
pg 2874; DOI:
10.1039/b106739g
PDF

Issue 22


Perkin 1 Abstracts: Natural Product Synthesis
Andrew Gunn Jacqueline E. Milne Marcel de Puit and Duncan McArthur
pg 22-xvii; DOI:
10.1039/b109682f
PDF
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis
Gideon Grogan Alexis Carstairs Ian Jackson Denise McIntyre Alan Watt Sabine Flitsch and Nicholas Turner
pg 22-xi; DOI:
10.1039/b109853p
PDF
Synthesis of heterocycles by radical cyclisation
W. Russell Bowman Martin O. Cloonan and Sussie L. Krintel
pg 2885; DOI:
10.1039/a909340k
PDF
Short synthesis of the optically active E-ring portion of (S)-camptothecin
S. Leue W. Miao A. Kanazawa Y. Génisson S. Garçon and A. E. Greene
pg 2903; DOI:
10.1039/b109071m
PDF
The reactions of diacetylenic ketones with nitrogen nucleophiles; facile preparation of alkynyl substituted pyrimidines and pyrazoles
Jack E. Baldwin Gareth J. Pritchard and Richard E. Rathmell
pg 2906; DOI:
10.1039/b108645f
PDF
Highly diastereoselective synthesis of -amino alcohols
Wim J. N. Meester Rudmer van Dijk Jan H. van Maarseveen Floris P. J. T. Rutjes Pedro H. H. Hermkens and Henk Hiemstra
pg 2909; DOI:
10.1039/b108254j
PDF
Asymmetric synthesis of N-diphenylphosphinoylamines by solvent-free enantioselective addition of dialkylzincs to N-diphenylphosphinoylimines
Itaru Sato Ryo Kodaka and Kenso Soai
pg 2912; DOI:
10.1039/b106775n
PDF
Novel synthesis of enantiomerically enriched 5-hydroxycyclohex-2-enone by enantioselective deprotonation strategy: application to the synthesis of inositol phosphatase inhibitor
Toshio Honda and Katsunori Endo
pg 2915; DOI:
10.1039/b107567p
PDF
Isolation and characterization of spirocaesalmin, a novel rearranged vouacapane diterpenoid from Caesalpinia minax Hance
Ren-Wang Jiang Shuang-Cheng Ma Paul P. H. But and Thomas C. W. Mak
pg 2920; DOI:
10.1039/b107473n
PDF
Conjugate addition of 6-membered hydrazine to chiral tert-butyl (E)-2-(p-tolylsulfinyl)cinnamates. Synthesis of (S)-celacinnine
Haruo Matsuyama Nobuhiro Itoh Aoi Matsumoto Nahoko Ohira Kenji Hara Masato Yoshida and Masahiko Iyoda
pg 2924; DOI:
10.1039/b107443c
PDF
Asymmetric synthesis of -amino acid scaffolds
Steven D. Bull Stephen G. Davies and Andrew D. Smith
pg 2931; DOI:
10.1039/b107440g
PDF
NMR characterization of lignins from transgenic poplars with suppressed caffeic acid O-methyltransferase activity
Jane M. Marita John Ralph Catherine Lapierre Lise Jouanin and Wout Boerjan
pg 2939; DOI:
10.1039/b107219f
PDF
Domino Michael–O-alkylation reaction: one-pot synthesis of 2,4-diacylhydrofuran derivatives and its application to antitumor naphthofuran synthesis
Hisahiro Hagiwara Kouji Sato Daisuke Nishino Takashi Hoshi Toshio Suzuki and Masayoshi Ando
pg 2946; DOI:
10.1039/b107180g
PDF
A new and efficient route to derivatives of (R)-4-hydroxycyclohex-2-enone
Libing Yu Ruzhou Zhang and Zhiqin Wang
pg 2958; DOI:
10.1039/b107085a
PDF
Synthesis and study of 4-hydroxymethyl-3-(alkylamino)acridines as models of a new class of DNA-intercalating–alkylating agents
Franck Charmantray Alain Duflos Jean Lhomme and Martine Demeunynck
pg 2962; DOI:
10.1039/b107055j
PDF
Diels–Alder reactions of alkyl 2H-azirine-3-carboxylates with furans
M. José Alves Nuno G. Azoia Jamie F. Bickley A. Gil Fortes Thomas L. Gilchrist and Ricardo Mendonça
pg 2969; DOI:
10.1039/b106985n
PDF
An efficient method for the one-pot construction of the 1H-naphtho[2,3-c]pyran-5,10-dione system
Kazuhiro Kobayashi Masaharu Uchida Tomokazu Uneda Keiichi Yoneda Miyuki Tanmatsu Osamu Morikawa and Hisatoshi Konishi
pg 2977; DOI:
10.1039/b106933k
PDF
The stereoselective synthesis of oxetanes; exploration of a new, Mitsunobu-style procedure for the cyclisation of 1,3-diols
Martin Christlieb John E. Davies Jason Eames Richard Hooley and Stuart Warren
pg 2983; DOI:
10.1039/b106851b
PDF
Pyrrolidinones derived from (S)-pyroglutamic acid. Part 3. -Aminopyrrolidinones
Philip W. H. Chan Ian F. Cottrell and Mark G. Moloney
pg 2997; DOI:
10.1039/b106782f
PDF
Pyrrolidinones derived from (S)-pyroglutamic acid. Part 4. , -Diaminopyrrolidinones
Philip W. H. Chan Ian F. Cottrell and Mark G. Moloney
pg 3007; DOI:
10.1039/b106783b
PDF
A new stereoselective route to the carbocyclic nucleoside cyclobut-A
Jagannath Panda Sarita Ghosh and Subrata Ghosh
pg 3013; DOI:
10.1039/b106542b
PDF
Expedient syntheses of naturally occurring ()-3-benzylphthalides and ()-3-aryl-8-hydroxy-3,4-dihydroisocoumarins: Structure revision of the ()-3-benzylphthalide isolated from Frullania falciloba
Raghao S. Mali Kantipudi N. Babu and Prakash G. Jagtap
pg 3017; DOI:
10.1039/b106268a
PDF
Novel cycloadditions of ortho-thioquinones with acyclic dienes: expeditious synthesis of 1,4-benzooxathiines
Vijay Nair Bini Mathew Siji Thomas Mariappanadar Vairamani and Sripadi Prabhakar
pg 3020; DOI:
10.1039/b106265b
PDF
[2+2]Photocycloaddition of 2-(dibenzylamino)ethyl 3-benzoylacrylate in a crystalline state: weak intermolecular interactions as important factors determining efficiency of the solid-state photoreaction
Tadashi Hasegawa Kaori Ikeda and Yuko Yamazaki
pg 3025; DOI:
10.1039/b105970j
PDF
Stereoselective synthesis of the pyrroloisoquinoline ring system
Steven M. Allin Stella L. James William P. Martin Timothy A. D. Smith and Mark R. J. Elsegood
pg 3029; DOI:
10.1039/b105402n
PDF
Putative metabolites of fulvestrant, an estrogen receptor downregulator. Improved glucuronidation using trichloroacetimidates
John R. Ferguson John R. Harding David A. Killick Keith W. Lumbard Feodor Scheinmann and Andrew V. Stachulski
pg 3037; DOI:
10.1039/b105397n
PDF
Manganese(III) acetate-mediated oxidative coupling of phenylhydrazines with benzene: a novel method for biaryl coupling
Ayhan S. Demir Ömer Reis and Emine Özgül-Karaaslan
pg 3042; DOI:
10.1039/b105119a
PDF
Absolute stereostructures of cell-adhesion inhibitors, macrosphelides C, E–G and I, produced by a Periconia species separated from an Aplysia sea hare
Takeshi Yamada Masashi Iritani Mitsunobu Doi Katsuhiko Minoura Tadayoshi Ito and Atsushi Numata
pg 3046; DOI:
10.1039/b104337b
PDF
2-(Lithiomethyl)-1-methylimidazole as a non-reactive bulk base and its novel mixed dimer with a chiral lithium amide in catalytic stereoselective deprotonation
Sten O. Nilsson Lill Daniel Pettersen Mohamed Amedjkouh and Per Ahlberg
pg 3054; DOI:
10.1039/b104336f
PDF
Reaction of phenylhydrazines with arenes in the presence of aluminium trichloride
Atsushi Ohwada Shigeru Nara Takeshi Sakamoto and Yasuo Kikugawa
pg 3064; DOI:
10.1039/b103802h
PDF
5-Amino-3-imino-1,2,6,7-tetracyano-3H-pyrrolizine: synthesis of alkylimino derivatives. X-Ray crystal and molecular structures of the hex-5-enyl, and Langmuir–Blodgett film of the octyl and octadecyl derivatives
Alberto Flamini Vincenzo Fares Aldo Capobianchi and Veronica Valentini
pg 3069; DOI:
10.1039/b103423p
PDF
Reactions of 4-methylchromene-2,7,8-trione with phosphonium ylides. Synthesis and evaluation of fused 1,3-dioxolocoumarins as antioxidants and antiinflammatories
Konstantina C. Fylaktakidou Daman R. Gautam Dimitra J. Hadjipavlou-Litina Christos A. Kontogiorgis Konstantinos E. Litinas and Demetrios N. Nicolaides
pg 3073; DOI:
10.1039/b103092m
PDF
Nucleoside carbonyl(di- and triphosphates)
Ivan B. Yanachkov James M. Stattel and George E. Wright
pg 3080; DOI:
10.1039/b102467c
PDF

Issue 23


Perkin 1 Abstracts: Solid Phase Organic Synthesis
Fabrice Anizon Jennifer Delaney Andrew Gunn Hassan Mamdani Catherine McCusker Fiona McKerlie and Tanya Wildman
pg 23-ix; DOI:
10.1039/b109854n
PDF
Supported catalysts and their applications in synthetic organic chemistry
Yolanda R. de Miguel Emilie Brulé and Robert G. Margue
pg 3085; DOI:
10.1039/b101948l
PDF
New access to 1,3-dialkyl-2,3-dihydro-2-imino-1H-imidazoles and their application to the first total synthesis of naamine B, a marine 2,3-dihydro-2-imino-1,3-dimethyl-1H-imidazole alkaloid
Ikuo Kawasaki Seikou Nakamura Satomi Yanagitani Akiko Kakuno Masayuki Yamashita and Shunsaku Ohta
pg 3095; DOI:
10.1039/b108762b
PDF
Biosynthesis of fluoroacetate and 4-fluorothreonine in Streptomyces cattleya. Incorporation of oxygen-18 from [2-2H,2-18O]-glycerol and the role of serine metabolites in fluoroacetaldehyde biosynthesis
Christoph Schaffrath Cormac D. Murphy John T. G. Hamilton and David O'Hagan
pg 3100; DOI:
10.1039/b108720g
PDF
Orthogonal N,N-deprotection strategies of -amino esters
Steven D. Bull Stephen G. Davies Peter M. Kelly Massimo Gianotti and Andrew D. Smith
pg 3106; DOI:
10.1039/b106389h
PDF
Asymmetric synthesis of -haloaryl -amino acid derivatives
Steven D. Bull Stephen G. Davies Santiago Delgado-Ballester Peter M. Kelly Luke J. Kotchie Massimo Gianotti Mario Laderas and Andrew D. Smith
pg 3112; DOI:
10.1039/b108573p
PDF
A simple access to 3,6-branched oligosaccharides: Synthesis of a glycopeptide derivative that relates to Lycium barbarum L.
Yuguo Du Meimei Zhang Feng Yang and Guofeng Gu
pg 3122; DOI:
10.1039/b108399f
PDF
Synthesis of new chiral and nonchiral N2O2 and N2S2 tetradentate ligands and their metal complexes
Franck Mevellec Sylvain Collet David Deniaud Alain Reliquet and Jean-Claude Meslin
pg 3128; DOI:
10.1039/b108210h
PDF
Rearrangement of 1,4,5,6-tetrahalo-7,7-dimethoxybicyclo[2.2.1]hept-5-en-2-ones to phenolic derivatives
Faiz Ahmed Khan Jyotirmayee Dash Dheeraj Jain and B. Prabhudas
pg 3132; DOI:
10.1039/b108152g
PDF
Synthesis and self-aggregation of zinc chlorophylls possessing an -hydroxyalkyl group: effect of distance between interactive hydroxy group and chlorin moiety on aggregation
Shiki Yagai and Hitoshi Tamiaki
pg 3135; DOI:
10.1039/b107902f
PDF
Azatriquinanes. Part 4. The chemistry of azatriquinenamine and its bromination products
Manuel Lera Alexander J. Blake Claire Wilson and Mark Mascal
pg 3145; DOI:
10.1039/b107707d
PDF
6-Substituted 2-azabicyclo[2.2.1]hept-5-enes by nitrogen-directed radical rearrangement: synthesis of an epibatidine analogue with high binding affinity at the nicotinic acetylcholine receptor
David M. Hodgson Christopher R. Maxwell Richard Wisedale Ian R. Matthews Kate J. Carpenter Anthony H. Dickenson and Susan Wonnacott
pg 3150; DOI:
10.1039/b107414h
PDF
Additions of stabilised and semi-stabilised sulfur ylides to tosyl protected imines: are they under kinetic or thermodynamic control?
Varinder K. Aggarwal Jonathan P. H. Charmant Cinzia Ciampi Jonathan M. Hornby Christopher J. O'Brien George Hynd and Richard Parsons
pg 3159; DOI:
10.1039/b107275g
PDF
Michael addition of thiols, carbon nucleophiles and amines to dehydroamino acid and dehydropeptide derivatives
Paula M. T. Ferreira Hernâni L. S. Maia Luís S. Monteiro and Joana Sacramento
pg 3167; DOI:
10.1039/b106487h
PDF
Antitumour polycyclic acridines. Part 9. Synthesis of 7H-pyrido[4,3,2-kl]acridines with basic side chains
Michael J. Ellis and Malcolm F. G. Stevens
pg 3174; DOI:
10.1039/b106324n
PDF
Antitumour polycyclic acridines. Part 10. Synthesis of penta- and hexa-cyclic heteroaromatic systems by radical cyclisations of substituted 9-anilinoacridines
Michael J. Ellis and Malcolm F. G. Stevens
pg 3180; DOI:
10.1039/b106327h
PDF
Novel organic-solvent-free aziridination of olefins: Chloramine-T–I2 system under phase-transfer catalysis conditions
Daisuke Kano Satoshi Minakata and Mitsuo Komatsu
pg 3186; DOI:
10.1039/b104940m
PDF
Intramolecular aldol-type condensation between side chains of naphthoquinones: biomimetic synthesis of 1,6- and 1,8-dihydroxyanthraquinones
Hidemitsu Uno Akane Masumoto Erina Honda Yumi Nagamachi Youtarou Yamaoka and Noboru Ono
pg 3189; DOI:
10.1039/b104789m
PDF
Peptido-organic Diels–Alder reactions on hydrophilic resin: scope for combinatorial chemistry
Anette Graven and Morten Meldal
pg 3198; DOI:
10.1039/b103765j
PDF
Reactions of N-benzyl-pyridinium or -isoquinolinium ylides with ethyl 3-fluoro-3-(fluoroalkyl)acrylates to give fluoroalkyl-substituted indolizine and pyrrolo[2,1-a]isoquinoline derivatives
Weimin Peng and Shizheng Zhu
pg 3204; DOI:
10.1039/b103586j
PDF

Issue 24


Perkin 1 Abstracts: Biocatalysis in Organic Synthesis
Gideon Grogan Alexis Carstairs Ian Jackson Denise McIntyre Alan Watt Sabine Flitsch and Nicholas Turner
pg 24-xvii; DOI:
10.1039/b110714n
PDF
Organic syntheses through free-radical annulations and related cascade sequences
Andrew J. McCarroll and John C. Walton
pg 3215; DOI:
10.1039/b105234a
PDF
Formation of adamantan-1-ols by the reactions of adamantanes with 2,3-dichloro-5,6-dicyano-p-benzoquinone (DDQ) in trifluoromethanesulfonic acid
Kiyoshi Tanemura Tsuneo Suzuki Yoko Nishida Koko Satsumabayashi and Takaaki Horaguchi
pg 3230; DOI:
10.1039/b109548j
PDF
The synthesis of pyrano[2,3-b]quinoxalines related to molybdopterin
Ben Bradshaw Andrew Dinsmore David Collison C. David Garner and John A. Joule
pg 3232; DOI:
10.1039/b108576j
PDF
Synthesis of the organic ligand of the molybdenum cofactor, in protected form
Ben Bradshaw Andrew Dinsmore Wadi Ajana David Collison C. David Garner and John A. Joule
pg 3239; DOI:
10.1039/b108579b
PDF
Synthesis of conformationally constrained amino acid and peptide derivatives
Patrick D. Bailey Neill Bannister Marine Bernad Sophie Blanchard and Andrew N. Boa
pg 3245; DOI:
10.1039/b108872f
PDF
Norlignan biosynthesis in Asparagus officinalis L.: the norlignan originates from two non-identical phenylpropane units
Shiro Suzuki Toshiaki Umezawa and Mikio Shimada
pg 3252; DOI:
10.1039/b107949b
PDF
Efficient synthesis of pyridines via a sequential solventless aldol condensation and Michael addition
Gareth W. V. Cave and Colin L. Raston
pg 3258; DOI:
10.1039/b107302h
PDF
Palladium-catalyzed cyanation of bromocalix[4]arenes at the upper rim
Hideaki Hioki Rumi Nakaoka Aya Maruyama and Mitsuaki Kodama
pg 3265; DOI:
10.1039/b109083f
PDF
Dilithiation of arenetricarbonylchromium(0) complexes with enantioselective quench: application to chiral biaryl synthesis
Yen-Ling Tan Andrew J. P. White David A. Widdowson René Wilhelm and David J. Williams
pg 3269; DOI:
10.1039/b108807f
PDF
Conjugate additions of organocuprates to a 3-methylene-6-isopropyldiketopiperazine acceptor for the asymmetric synthesis of homochiral -amino acids
Steven D. Bull Stephen G. Davies A. Christopher Garner and Michael D. O'Shea
pg 3281; DOI:
10.1039/b108621a
PDF
Dioxygenase-catalysed mono-, di- and tri-oxygenation of dialkyl sulfides and thioacetals: chemoenzymatic synthesis of enantiopure cis-diol sulfoxides
Derek R. Boyd Narain D. Sharma Simon A. Haughey John F. Malone AlistairW. T. King Brian T. McMurray André Alves-Areias Christopher C. R. Allen Robert Holt and Howard Dalton
pg 3288; DOI:
10.1039/b108620k
PDF
A rational approach to calix[n]furan precursors
Valérie Bénéteau Otto Meth-Cohn and Charles W. Rees
pg 3297; DOI:
10.1039/b108402j
PDF
A novel stereoselective synthesis of N-heterocycles by intramolecular hydrovinylation
Ulrich Bothe Hans Christian Rudbeck David Tanner and Mogens Johannsen
pg 3305; DOI:
10.1039/b108310d
PDF
Rearrangement of ammonium ylides produced by intramolecular reaction of catalytically generated metal carbenoids. Part 1. Synthesis of cyclic amines
J. Stephen Clark Paul B. Hodgson Michael D. Goldsmith and Leslie J. Street
pg 3312; DOI:
10.1039/b108179a
PDF
Rearrangement of ammonium ylides produced by intramolecular reaction of catalytically generated metal carbenoids. Part 2. Stereoselective synthesis of bicyclic amines
J. Stephen Clark Paul B. Hodgson Michael D. Goldsmith Alexander J. Blake Paul A. Cooke and Leslie J. Street
pg 3325; DOI:
10.1039/b108182a
PDF
Carotenoids and related polyenes. Part 7. Total synthesis of crassostreaxanthin B applying the stereoselective rearrangement of tetrasubstituted epoxides
Chisato Tode Yumiko Yamano and Masayoshi Ito
pg 3338; DOI:
10.1039/b108037g
PDF
Synthesis of chiral cis- and trans-furo[3,2-c][2]benzoxocines from D-glucose by regioselective 8-endo aryl radical cyclisation
Aniruddha Nandi Ranjan Mukhopadhyay and Partha Chattopadhyay
pg 3346; DOI:
10.1039/b107886k
PDF
Novel diphenylphosphine derivatives of 2,2-bithiophene, 2,2:5,2-terthiophene, 2-(2-thienyl)pyridine and 2,6-di-2-thienylpyridine. Crystal structures of 5,5-bis(diphenylphosphino)-2,2-bithiophene, diphenyl{5-[6-(diphenylphosphino)-2-pyridyl]-2-thienyl}phosphine and 2,6-bis[5-(diphenylphosphino)-2-thienyl]pyridine
John S. Field Raymond J. Haines Elena I. Lakoba and M. Hal Sosabowski
pg 3352; DOI:
10.1039/b107389n
PDF
Size discrimination in intramolecular complexation of modified -cyclodextrins: a preparative and nuclear magnetic resonance study
Julia S. Lock Bruce L. May Philip Clements John Tsanaktsidis Christopher J. Easton and Stephen F. Lincoln
pg 3361; DOI:
10.1039/b107324a
PDF
Synthesis of nucleic-acid base containing norbornene derivatives as monomers for ring-opening-metathesis–polymerization
R. Gareth Davies Vernon C. Gibson Michael B. Hursthouse Mark E. Light Edward L. Marshall Michael North David A. Robson Ian Thompson Andrew J. P. White David J. Williams and Paul J. Williams
pg 3365; DOI:
10.1039/b107139d
PDF
Nitrogen-containing heterocycles: 1,3-dipolar cycloaddition of stabilized nitrones with alkynes; primary cycloadducts, first and second generation rearrangement processes
Frances Heaney Julie Fenlon Colm O'Mahony Patrick McArdle and Desmond Cunningham
pg 3382; DOI:
10.1039/b106832f
PDF
On the scope and limitations of the Heck reaction of upper rim tetraiodocalix[4]arenes
Nikolai Kuhnert and Adam Le-Gresley
pg 3393; DOI:
10.1039/b106535c
PDF
Polyhalogenated BEDT-TTF through chlorination (SO2Cl2, Cl2) and fluorination (Selectfluor, XeF2) of 5,6-dihydro[1,3]dithiolo[4,5-b][1,4]dithiin-2-one
Olivier J. Dautel and Marc Fourmigué
pg 3399; DOI:
10.1039/b106144p
PDF
Facile attachment of functional moieties to crosslinked polystyrene beads via robust linkages: Suzuki reactions using polymer-supported boronic acids
Roger J. Kell Philip Hodge Mohammad Nisar and Richard T. Williams
pg 3403; DOI:
10.1039/b103760a
PDF
Synthesis of geminal bis(hydroxymethyl)pyrrolidine and pyrrolizidine imino sugars
Frank Schieweck and Hans-Josef Altenbach
pg 3409; DOI:
10.1039/b007607o
PDF