Perkin 1 Abstracts: Solid Phase Organic Synthesis Catherine McCusker Tanya Wildman and Fiona McKerlie pg 1-ix; DOI: 10.1039/b009122g |
Applications of stoichiometric transition metal complexes in organic synthesis Anthony J. Fletcher and Steven D. R. Christie pg 1; DOI: 10.1039/b002281k |
A new synthetic approach to porphyrin-![]() Vinich Promarak and Paul L. Burn pg 14; DOI: 10.1039/b007389j |
An approach to the synthesis of 5,5-trans-fused lactam analogues of ![]() Paul W. Smith Andrew R. Whittington Kevin N. Cobley Albert Jaxa-Chamiec and Harry Finch pg 21; DOI: 10.1039/b007286i |
Organophosphorus chemistry. Part 1. The synthesis of alkyl methylphosphonic acids Christopher M. Timperley Michael Bird Ian Holden and Robin M. Black pg 26; DOI: 10.1039/b007077g |
Picolyl-armed 1,3-alternate calix[4]areneazacrown ethers Jong Seung Kim Ok Jae Shon Wonbo Sim Sun Kyu Kim Moon Hwan Cho Jin-Gyu Kim Il-Hwan Suh and Dong Won Kim pg 31; DOI: 10.1039/b006801m |
Studies on the reactivity of N-(3-thienyl)carbamates Delphine Brugier Francis Outurquin and Claude Paulmier pg 37; DOI: 10.1039/b003580g |
Unexpected products from the formylation of N,N-dimethylanilines with 2-formamidopyridine in POCl3 Ying Cheng Peng Jiao David J. Williams and Otto-Meth Cohn pg 44; DOI: 10.1039/b006148o |
Cross-coupling reactions in Cinchona alkaloid chemistry: aryl-substituted and dimeric quinine, quinidine, as well as quincorine and quincoridine derivatives Jens Frackenpohl Wilfried M. Braje and H. Martin R. Hoffmann pg 47; DOI: 10.1039/b004693k |
TFA-catalyzed ring transformation of 4-hydroxycyclobutenone: A simple and general route for preparation of 3-substituted 4-aminofuran-2(5H![]() ![]() Jie Wang Xin Jiang Ming Chen Zongming Ge Yuefei Hu and Hongwen Hu pg 66; DOI: 10.1039/b004654j |
Parasite glycoconjugates. Part 11. Preparation of phosphodisaccharide synthetic probes, substrate analogues for the elongating ![]() Andrew J. Ross Irina A. Ivanova Michael A. J. Ferguson and Andrei V. Nikolaev pg 72; DOI: 10.1039/b004653l |
![]() Toshifumi Miyazawa Shin ![]() pg 82; DOI: 10.1039/b004183l |
Broadening of the substrate tolerance of ![]() Toshifumi Miyazawa Kayoko Tanaka Eiichi Ensatsu Ryoji Yanagihara and Takashi Yamada pg 87; DOI: 10.1039/b004180g |
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis Gideon Grogan Alexis Carstairs Ian Jackson Denise McIntyre Alan Watt Sabine Flitsch and Nicholas Turner pg 2-ix; DOI: 10.1039/b010107i |
Perkin 1 Abstracts: Natural Product Synthesis Jacqueline E. Milne Marcel de Puit and Duncan McAurthur pg 2-xv; DOI: 10.1039/b010200h |
Stoichiometric asymmetric processes Peter O ![]() pg 95; DOI: 10.1039/a907926b |
Ring-fused gem-dibromocyclopropanes as precursors to enantiomerically pure D- and L-series 3-deoxy- and 2-amino-2,3-dideoxyaldohexose derivatives Martin G. Banwell Wolfgang Ebenbeck and Alison J. Edwards pg 114; DOI: 10.1039/b008146i |
The chemistry of lithiated phosphine oxides: the stereoselective synthesis of alkene-4,5-diols Thomas Boesen Neil Feeder Martin D. Eastgate David J. Fox Jonathan A. Medlock Charles R. Tyzack and Stuart Warren pg 118; DOI: 10.1039/b008500f |
Cyclodimerization of indol-2-ylacetylenes. An example of intermolecular enyne–alkyne cycloaddition Daniele Passarella Alessandra Giardini Marisa Martinelli and Alessandra Silvani pg 127; DOI: 10.1039/b009154p |
General syntheses of 1-alkyltoxoflavin and 8-alkylfervenulin derivatives of biological significance by the regioselective alkylation of reumycin derivatives and the rates of transalkylation from 1-alkyltoxoflavins into nucleophiles Tomohisa Nagamatsu and Hirofumi Yamasaki pg 130; DOI: 10.1039/b007302o |
Scope and limitations of the [1,2]-alkylsulfanyl (SMe, SEt and SCH2Ph) and sulfanyl (SH) migration in the stereospecific synthesis of substituted tetrahydrofurans![]() Jason Eames Nikolai Kuhnert and Stuart Warren pg 138; DOI: 10.1039/b007284m |
Synthesis of 3-deazathiamine Daniel Hawksley David A. Griffin and Finian J. Leeper pg 144; DOI: 10.1039/b006962k |
Juli–Colonna stereoselective epoxidation of some ![]() ![]() ![]() Peter C. Ray and Stanley M. Roberts pg 149; DOI: 10.1039/b007100p |
Synthesis of thieno[2,3-b]quinoxalines from 2-haloquinoxalines Montserrat Armengol and John A. Joule pg 154; DOI: 10.1039/b008459j |
Synthesis of biphenylenes and tetraphenylenes using copper-catalyzed coupling of arylzinc intermediates S. M. Humayun Kabir Masashi Hasegawa Yoshiyuki Kuwatani Masato Yoshida Haruo Matsuyama and Masahiko Iyoda pg 159; DOI: 10.1039/b006375o |
Approaches to the synthesis of (+)- and (–)-epibatidine![]() M. Teresa Barros Christopher D. Maycock and M. Rita Ventura pg 166; DOI: 10.1039/b002980g |
Stereoselective synthesis of 24-alkyl-22-hydroxysterols based on chelation-controlled radical reactions Hajime Nagano Mikako Matsuda and Tomoko Yajima pg 174; DOI: 10.1039/b007139k |
Photoinduced [2+2] cycloadditions (the Paterno–Bchi reaction) of 1H-1-acetylindole-2,3-dione with alkenes Jie Xue Yan Zhang Tao Wu Hoong-Kun Fun and Jian-Hua Xu pg 183; DOI: 10.1039/b005576j |
Synthesis of naturally occurring phosphatidylinositol 3,4,5-trisphosphate [PtdIns(3,4,5)P3] and its diastereoisomers Piers R. J. Gaffney and Colin B. Reese pg 192; DOI: 10.1039/b007267m |
A conjugate addition–radical cyclisation approach to sesquiterpene-phenol natural products Barry S. Crombie Colin Smith Christalla Z. Varnavas and Timothy W. Wallace pg 206; DOI: 10.1039/b005617k |
Professor Christopher J. Moody![]() pg 3-vii; DOI: 10.1039/b009213o |
Perkin 1 Abstracts: Solid Phase Organic Synthesis Catherine McCusker Tanya Wildman Fiona McKerlie Andrew Gunn Hassan Mamdani Jennifer Delaney and Sabrice Anizon pg 3-ix; DOI: 10.1039/b100469g |
Unusual chemoselective addition of diisopropylzinc to 2,2![]() ![]() Shigehisa Tanji Takanori Shibata Itaru Sato and Kenso Soai pg 217; DOI: 10.1039/b009474i |
Observations on the samarium diiodide-promoted C–C fragmentation/ring expansion chemistry of some aliphatic 1,4-diketones D. Bradley G. Williams Kevin Blann and Cedric W. Holzapfel pg 219; DOI: 10.1039/b008110h |
A first synthesis of a phosphatidylcholine bearing docosahexaenoic and tetracosahexaenoic acids Naomichi Baba Md. Khorshed Alam Yoshihiro Mori Syed S. Haider Masatoshi Tanaka Shuhei Nakajima and Sakayu Shimizu pg 221; DOI: 10.1039/b007923p |
Selenium catalysed oxidations with aqueous hydrogen peroxide. Part I: epoxidation reactions in homogeneous solution Gerd-Jan ten Brink Bruno C. M. Fernandes Michiel C. A. van Vliet Isabel W. C. E. Arends and Roger A. Sheldon pg 224; DOI: 10.1039/b008198l |
Synthesis of espicufolin based on 6-endo ring closure of o-alkynoylnaphthols![]() Hidemitsu Uno Katsuji Sakamoto Erina Honda Kaori Fukuhara Noboru Ono Junya Tanaka and Masahiro Sakanaka pg 229; DOI: 10.1039/b007859j |
Synthesis and reactivity of ![]() ![]() ![]() Shin-ichi Watanabe Keiichirou Yamamoto Yukiko Itagaki Tatsunori Iwamura Tetsuo Iwama Tadashi Kataoka Genzoh Tanabe and Osamu Muraoka pg 239; DOI: 10.1039/b007715l |
Studies on the preparation of camphorylidene derivatives of ![]() David L. Gamble William P. Hems and Brian Ridge pg 248; DOI: 10.1039/b007659g |
Spirostanic analogues of teasterone. Synthesis, characterisation and biological activity of laxogenin, (23S![]() Martín A. Iglesias-Arteaga Roxana Pérez Gil Carlos S. Pérez Martínez and Francisco Coll Manchado pg 261; DOI: 10.1039/b007656m |
Stereocontrolled synthesis of (2S![]() James C. Anderson and Alice Flaherty pg 267; DOI: 10.1039/b007586h |
Regio- and stereoselectivity in the solvomercuriation and intramolecular alkoxymercuriation of cyclic unsaturated alcohols Yasuhisa Senda Satomi Takayanagi Tomomi Sudo and Hiroki Itoh pg 270; DOI: 10.1039/b006963i |
Synthesis, X-ray structures and chemistry of enantiomerically pure 10,11-dihydro-5-phenyl-5H-dibenzo[b,f![]() Paul Wyatt Stuart Warren Mary McPartlin and Tom Woodroffe pg 279; DOI: 10.1039/b006883g |
Synthesis of sugar-modified derivatives of the unusual nucleoside oxanosine and its carbocyclic analogs as potential inhibitors of HIV![]() Yoshio Saito Mariko Nakamura Tsuneya Ohno Chanya Chaicharoenpong Eiko Ichikawa Shosuke Yamamura Kuniki Kato and Kazuo Umezawa pg 298; DOI: 10.1039/b006763f |
Synthesis of novel analogues of the calicheamicin ![]() ![]() Stéphane Moutel and Jacques Prandi pg 305; DOI: 10.1039/b006113l |
Diethylamino(trimethyl)silane-mediated direct 1,4-addition of naked aldehydes to electron-deficient olefins Hisahiro Hagiwara Nao Komatsubara Hiroki Ono Tomoyuki Okabe Takashi Hoshi Toshio Suzuki Masayoshi Ando and Michiharu Kato pg 316; DOI: 10.1039/b005728m |
The thionophosphate–thiolophosphate![]() ![]() Veejendra K. Yadav Rengarajan Balamurugan Masood Parvez and Raghav Yamdagni pg 323; DOI: 10.1039/b003501g |
Perkin 1 Abstracts: Natural Product Synthesis Jacqueline E. Milne Marcel de Puit Andrew Gunn and Duncan McAurthur pg 4-xiii; DOI: 10.1039/b100677k |
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis Gideon Grogan Alexis Carstairs Ian Jackson Denise McIntyre Alan Watt Sabine Flitsch and Nicholas Turner pg 4-ix; DOI: 10.1039/b100781p |
The synthesis of thiols, selenols, sulfides, selenides, sulfoxides, selenoxides, sulfones and selenones David J. Procter pg 335; DOI: 10.1039/b002081h |
Indium triiodide catalysed one-step conversion of tetrahydropyranyl ethers to acetates with high selectivity Brindaban C. Ranu and Alakananda Hajra pg 355; DOI: 10.1039/b100014b |
A polymer-supported thionating reagent Steven V. Ley Andrew G. Leach and R. Ian Storer pg 358; DOI: 10.1039/b008814p |
Enantiospecific enzyme-catalysed resolution of novel N,N-disubstituted ![]() D. Jonathan Bennett Kirsteen I. Buchanan Andrew Cooke Ola Epemolu Niall M. Hamilton Edward J. Hutchinson and Ann Mitchell pg 362; DOI: 10.1039/b008000o |
The preparation and use of polyHIPE-grafted reactants to reduce alkyl halides under free-radical conditions Alexandre Chemin Anthony Mercier Hervé Deleuze Bernard Maillard and Olivier Mondain-Monval pg 366; DOI: 10.1039/b009318l |
Asymmetric synthesis of enantiomerically enriched atropisomeric amides by desymmetrisation of N,N-dialkylmesitamides![]() Jonathan Clayden Paul Johnson and Jennifer H. Pink pg 371; DOI: 10.1039/b008678i |
Selective vicarious nucleophilic amination of 3-nitropyridines Jan M. Bakke Harald Svensen and Raffaela Trevisan pg 376; DOI: 10.1039/b008660f |
Synthesis of the bis-spiroacetal moiety of the polyether antibiotic CP44,161 Paul R. Allen Margaret A. Brimble and Hishani Prabaharan pg 379; DOI: 10.1039/b008159k |
Titanium(IV) chloride, zirconium(IV) chloride or boron trichloride and phosphine-promoted Baylis–Hillman reaction of aldehydes with ![]() ![]() Min Shi Jian-Kang Jiang Shi-Cong Cui and Yan-Shu Feng pg 390; DOI: 10.1039/b008105l |
Transformations of selenadiazoliumyl-N-unsubstituted methanides (ylides) to new divinyl selenide derivatives and substituted 1,3,5-selenadiazines. Organoselenium systems from azolium 1,3-dipoles Richard N. Butler and Anthony Fox pg 394; DOI: 10.1039/b007974j |
Reactions involving fluoride ion. Part 47. Reactions of perfluorobicycloalkenes Richard D. Chambers and Takayuki Nakamura pg 398; DOI: 10.1039/b007825p |
Novel organosulfur donors containing hydroxy functionalities: synthesis of bis[2,2-bis(hydroxymethyl)propane-1,3-diyldithio]tetrathiafulvalene and related materials![]() Turan Ozturk Nezire Saygili Serife Ozkara Melanie Pilkington Craig R. Rice Deborah A. Tranter Figen Turksoy and John D. Wallis pg 407; DOI: 10.1039/b007660k |
Carbocyclic ring closure of hex-5-enopyranosides and pent-4-enofuranosides: a nitrile oxide approach John K. Gallos and Theocharis V. Koftis pg 415; DOI: 10.1039/b007654f |
Gas-phase pyrolysis of 4-amino-3-allylthio-1,2,4-triazoles: a new route to [1,3]thiazolo[3,2-b][1,2,4]triazoles Dale D. J. Cartwright Bernard A. J. Clark and Hamish McNab pg 424; DOI: 10.1039/b007638o |
Synthesis of a regio-isomer of kealiiquinone, a marine benzimidazole alkaloid Seikou Nakamura Naoki Tsuno Masayuki Yamashita Ikuo Kawasaki Shunsaku Ohta and Yoshitaka Ohishi pg 429; DOI: 10.1039/b007560o |
Alkoxydienylstannanes via metalation of ![]() ![]() ![]() Paolo Balma Tivola Anna Deagostino Cristina Prandi and Paolo Venturello pg 437; DOI: 10.1039/b007500k |
Selective metallation of thiophene and thiazole rings with magnesium amide base Manabu Shilai Yoshinori Kondo and Takao Sakamoto pg 442; DOI: 10.1039/b007376h |
The role of the ester group in determining the regiochemistry of selected ![]() ![]() Ernest W. Della and Paul A. Smith pg 445; DOI: 10.1039/b006691p |
Microwave-induced 1,3-dipolar intramolecular cycloadditions of N-substituted oximes, nitrones, and azomethine ylides for the chiral synthesis of functionalized nitrogen heterocycles Qian Cheng Wen Zhang Yoshimichi Tagami and Takayuki Oritani pg 452; DOI: 10.1039/b006000n |
Heterocycles of biological importance. Part 5. The formation of novel biologically active pyrimido[1,2-a]benzimidazoles from allenic nitriles and aminobenzimidazoles Peter Forche Asobo Helene Wahe Joseph Tanyi Mbafor Augustin Ephraim Nkengfack Zacharias Tanee Fomum Emmanuel Fondjo Sopbue and Dietrich Döpp pg 457; DOI: 10.1039/b005511p |
Investigation of arene–arene interaction in stereoselective MCPBA epoxidation Keiki Kishikawa Mamoru Naruse Shigeo Kohmoto Makoto Yamamoto and Kentaro Yamaguchi pg 462; DOI: 10.1039/b004098n |
The synthesis of cyclic peptides John N. Lambert Jeffrey P. Mitchell and Kade D. Roberts pg 471; DOI: 10.1039/b001942i |
Synthesis of novel 5-amino-6-ethoxy-2-alkylpyrimidine-4-carbonitriles Amal Al-Azmi Brian L. Booth Robin G. Pritchard and Fernanda J. R. P. Proença pg 485; DOI: 10.1039/b009804n |
Diastereoselective SmI2 mediated cascade radical cyclisations of methylenecyclopropane derivatives—syntheses of paeonilactone B and 6-epi-paeonilactone A Raymond J. Boffey William G. Whittingham and Jeremy D. Kilburn pg 487; DOI: 10.1039/b009513n |
Regiochemistry in alkylation, acylation and methoxycarbonylation of alkali salts from 2-substituted alkenylpropanedinitriles Hege Karlsen Pål H. Songe Lise Kristin Sunsby Lise Cathrine Hagen Per Kolsaker and Christian Rømming pg 497; DOI: 10.1039/b009175h |
Synthesis of novel pipecolic acid derivatives. Part 2. Addition of trimethylsilyl cyanide to 3,4,5,6-tetrahydropyridines Ole Westerhoff Arne Lützen Wolfgang Maison Marc Kosten and Jürgen Martens pg 508; DOI: 10.1039/b009112j |
Microchip-based synthesis and total analysis systems (SYNTAS): chemical microprocessing for generation and analysis of compound libraries Michael C. Mitchell Valerie Spikmans Andreas Manz and Andrew J. de Mello pg 514; DOI: 10.1039/b009037i |
Stereocontrolled synthesis of trifluoromethylated (E)- or (Z)-ynenyl sulfones via sequential transformations Yanchang Shen Guoping Wang and Jie Sun pg 519; DOI: 10.1039/b008849h |
Synthesis of trisphaeridine and norchelerythrine through palladium-catalyzed aryl–aryl coupling reactions Takashi Harayama Hisashi Akamatsu Kana Okamura Taeko Miyagoe Toshihiko Akiyama Hotoshi Abe and Yasuo Takeuchi pg 523; DOI: 10.1039/b008683p |
Synthesis and structure of 1-methyl-2,6-bis(electron-withdrawing group)-substituted selenabenzenes Eiji Honda Tatsunori Iwamura Shin-ichi Watanabe Tadashi Kataoka Osamu Muraoka and Genzoh Tanabe pg 529; DOI: 10.1039/b008562f |
Metabolites of the higher fungi. Part 32. Rosnecatrone, a phytotoxic bicyclo[4.1.0]hept-3-en-2-one from the fungus Rosellinia necatrix Prill Raymond L. Edwards Derek J. Maitland Ian J. Scowen Antonio J. T. De Sousa and Anthony J. S. Whalley pg 537; DOI: 10.1039/b008195g |
A strategy for chemical synthesis of selectively methyl-esterified oligomers of galacturonic acid Mads H. Clausen Malene R. Jørgensen Jesper Thorsen and Robert Madsen pg 543; DOI: 10.1039/b006981g |
Reaction of tetrafluoroethene oligomers. Part 17. Some reactions of (E/Z)-perfluoro-2,3-dimethylpenta-1,3-diene Graham D. Burns Paul L. Coe and Colan L. Andrews pg 552; DOI: 10.1039/b006825j |
Preparation of pyrimido[2,1-a]phthalazines and an aminopyrimido[2,1-a]isoindole by retro Diels–Alder reaction Pál Sohár Ferenc Miklós Antal Csámpai and Géza Stájer pg 558; DOI: 10.1039/b005008n |
Perkin 1 Abstracts: Natural Product Synthesis Andrew Gunn Jaqueline E. Milne Marcel de Puit and Duncan McArthur pg 6-xvii; DOI: 10.1039/b101363g |
Perkin 1 Abstracts: Solid Phase Organic Synthesis Fabrice Anizon Jennifer Delaney Andrew Gunn Hassan Mamdani Catherine McCusker Fiona McKerlie and Tanya Wildman pg 6-vii; DOI: 10.1039/b101365n |
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis Gideon Grogan Alexis Carstairs Ian Jackson Denise McIntyre Alan Watt Sabine Flitsch and Nicholas Turner pg 6-xii; DOI: 10.1039/b101581h |
Versatile route to 2,6-dideoxyamino sugars from non-sugar materials: Syntheses of vicenisamine and kedarosamine Yoshitaka Matsushima Takuya Nakayama Shigehiro Tohyama Tadashi Eguchi and Katsumi Kakinuma pg 569; DOI: 10.1039/b008878l |
Benzylic oxidation of aromatics with cerium(IV) triflate; synthetic scope and mechanistic insight Kenneth K. Laali Mark Herbert Brad Cushnyr Anand Bhatt and David Terrano pg 578; DOI: 10.1039/b008843i |
Cyclodextrins to limit substrate inhibition and alter substrate selectivity displayed by enzymes Christopher J. Easton Jason B. Harper Sarah J. Head Kitty Lee and Stephen F. Lincoln pg 584; DOI: 10.1039/b008339i |
Attempts to find a solution to the problem of atropisomer interconversion in 1,8-diarylnaphthalenes and 5,6-diarylacenaphthenes Melanie Steele Michael Watkinson and Andrew Whiting pg 588; DOI: 10.1039/b008319o |
The bisected s-trans conformation-controlled highly stereoselective addition of Grignard reagents to C-cyclopropylaldonitrone. An efficient synthesis of 1-phenyl-2-[(S![]() Yuji Kazuta Satoshi Shuto Hiroshi Abe and Akira Matsuda pg 599; DOI: 10.1039/b008230i |
Further evidence for the participation of primary carbon-centered free radicals in the antimalarial action of the qinghaosu (artemisinin) series of compounds Dong-Ye Wang Yu-Lin Wu Yikang Wu Jie Liang and Ying Li pg 605; DOI: 10.1039/b008145k |
Secondary mould metabolites. Part 59. Sesquiterpene illudanes: semi-synthesis of new illudins, structures and biological activity Alberto Arnone Lucio Merlini Gianluca Nasini Orso Vajna de Pava and Franco Zunino pg 610; DOI: 10.1039/b007633n |
Steroid-fullerene adducts from Diels–Alder reactions: characterization and the effect on the activity of Ca2+-ATPase Lian-Sheng Li Yun-Jin Hu Yikang Wu Yu-Lin Wu Jiachang Yue and Fuyu Yang pg 617; DOI: 10.1039/b007498p |
Pyrimidine annelated heterocycles—synthesis and cycloaddition of the first pyrimido[1,4]diazepine N-oxides Frances Heaney Cathriona Burke Desmond Cunningham and Patrick McArdle pg 622; DOI: 10.1039/b007163n |
Perkin 1 Abstracts: Solid Phase Organic Synthesis Fabrice Anizon Jennifer Delaney Andrew Gunn Hassan Mamdani Catherine McCusker Fiona McKerlie and Tanya Wildman pg 7-vii; DOI: 10.1039/b102280f |
Enantioselective synthesis of hydroxy ketones through cleavage and formation of acyloin linkage. Enzymatic kinetic resolution via C–C bond cleavage Ayhan S. Demir Martina Pohl Elena Janzen and Michael Müller pg 633; DOI: 10.1039/b100341k |
Multiple substitutions on (![]() Susan E. Gibson (née Thomas) Jonathan W. Steed and Surojit Sur pg 636; DOI: 10.1039/b009639n |
Regioselectivity of methylation of O-demethylangolensin [1-(2,4-dihydroxyphenyl)-2-(4-hydroxyphenyl)propan-1-one]. An expedient synthesis of angolensin Kristiina Wähälä Tuija Jokela Auli Salakka Seppo Kaltia and Markku Mesilaakso pg 642; DOI: 10.1039/b100778p |
Efficient 1,8- and 1,9-asymmetric inductions in the Grignard reaction of ![]() ![]() ![]() Masamitsu Date Yasufumi Tamai Tetsutaro Hattori Hideki Takayama Yoshinori Kamikubo and Sotaro Miyano pg 645; DOI: 10.1039/b100497m |
The pyridinium reduction route to alkaloids: a synthesis of ()-tashiromine Roderick W. Bates and Jutatip Boonsombat pg 654; DOI: 10.1039/b100407g |
Synthesis and absolute configuration of stellettadine A, a bisguanidinium alkaloid isolated from a marine sponge Stelletta sp. Hirosato Takikawa Dai Nozawa and Kenji Mori pg 657; DOI: 10.1039/b100206f |
Conversion of enamines, enamides and triazoles by trithiazyl trichloride into 1,2,5-thiadiazoles Charles W. Rees and Tai-Yuen Yue pg 662; DOI: 10.1039/b010140k |
The efficient, enantioselective synthesis of quinoxaline, pyrazine and 1,2,4-triazine substituted ![]() Robert M. Adlington Jack E. Baldwin David Catterick and Gareth J. Pritchard pg 668; DOI: 10.1039/b010134f |
The oxidative rearrangement of furan-2-carboximidamides: preparation and properties of 2-acylaminofurans Mária Bobo ![]() ![]() ![]() ![]() pg 680; DOI: 10.1039/b010010m |
Total synthesis and radiolabelling of an efficient rt-PA inhibitor: [11C] (Z,Z![]() Fabrice Siméon Franck Sobrio Fabienne Gourand and Louisa Barré pg 690; DOI: 10.1039/b009850g |
Novel bis(tetrahydropyrrolo[3,4-b]carbazoles) linked with aliphatic chains: synthesis and structural aspects Kerstin U. Meyer and Ulf Pindur pg 695; DOI: 10.1039/b009731o |
Attempts at asymmetric electrosynthesis of ![]() Sophie Goumain Hassan Oulyadi Philippe Jubault Christian Feasson and Jean-Charles Quirion pg 701; DOI: 10.1039/b008906k |
Utilization of industrial waste materials. Part 20. Stereoselective cycloaddition of silylenes and a disilene to an enantiomerically pure cyclic ketimine derived from an industrial waste material Nikolai Graf von Keyserlingk Jürgen Martens Detlev Ostendorf Wolfgang Saak and Manfred Weidenbruch pg 706; DOI: 10.1039/b008708o |
Synthesis and NMR characterisation of novel highly cyclised polyprenoid hydrocarbons from sediments Emmanuelle Grosjean Jacques Poinsot Armelle Charrié-Duhaut Stéphanie Tabuteau Pierre Adam Jean Trendel Philippe Schaeffer Jacques Connan Daniel Dessort and Pierre Albrecht pg 711; DOI: 10.1039/b008104n |
Aromatic azapentalenes: 1H- and (mesoionic) 2H-pyrrolotetrazoles. Part 1. Synthesis and spectral characteristics![]() Dietrich Moderhack Dirk Decker and Bernhard Holtmann pg 720; DOI: 10.1039/b007873p |
Aromatic azapentalenes: 1H- and (mesoionic) 2H-pyrrolotetrazoles. Part 2. Reaction with electrophiles Dietrich Moderhack Dirk Decker and Bernhard Holtmann pg 729; DOI: 10.1039/b007874n |
Pd(0)–Cu(I)-catalyzed cross-coupling of alkynylsilanes with triarylantimony(V) diacetates Suk-Ku Kang Hyung-Chul Ryu and Young-Taek Hong pg 736; DOI: 10.1039/b007800j |
Synthesis, characterization, and electrogenerated chemiluminescence of phenyl-substituted, phenyl-annulated, and spirofluorenyl-bridged oligothiophenes Ullrich Mitschke and Peter Bäuerle pg 740; DOI: 10.1039/b006553f |
Carbohydrate-derived dienes for intramolecular and asymmetric Diels–Alder reactions![]() Pilar Areces José Luis Jiménez Maria de la Cruz Pozo Emilio Román and José Antonio Serrano pg 754; DOI: 10.1039/b006078j |
Gran Magnusson Jan Kihlberg pg 767; DOI: 10.1039/b009690n |
Iodine and its interhalogen compounds: versatile reagents in carbohydrate chemistry. XIV. Glycosylated amino acid synthesis K. P. Ravindranathan Kartha Lluis Ballell Julia Bilke Michael McNeil and Robert A. Field pg 770; DOI: 10.1039/b009682m |
Synthesis of clustered xenotransplantation antagonists using palladium-catalyzed cross-coupling of prop-2-ynyl ![]() Bingcan Liu and René Roy pg 773; DOI: 10.1039/b101234g |
Synthesis of carba sugars from aldonolactones. Part IV. Stereospecific synthesis of carbaheptopyranoses by radical-induced carbocyclisation of 2,3-unsaturated octonolactones Sussi Holstein Wagner and Inge Lundt pg 780; DOI: 10.1039/b100708o |
Cyclizations versus rearrangements in the reactions of some epoxyolefins with Lewis acids![]() Lars Pettersson and Torbjörn Frejd pg 789; DOI: 10.1039/b010101j |
Stereoselective photochemical transformations of hexopyranosyl imides to highly functionalised heterocycles Swantje Thiering Carsten E. Sowa and Joachim Thiem pg 801; DOI: 10.1039/b010020j |
Carbopeptoids: peptides and diketopiperazines incorporating the anomeric centre of mannopyranose Daniel D. Long Richard J. Tennant-Eyles Juan C. Estevez Mark R. Wormald Raymond A. Dwek Martin D. Smith and George W. J. Fleet pg 807; DOI: 10.1039/b009940f |
Towards a modular approach for heparin synthesis Michael Haller and Geert-Jan Boons pg 814; DOI: 10.1039/b009845k |
Trivalent ![]() Thisbe K. Lindhorst Sven Kötter Ulrike Krallmann-Wenzel and Stefan Ehlers pg 823; DOI: 10.1039/b009786l |
Efficient stereoselective synthesis of 1-thio-![]() Henry N. Yu Chang-Chun Ling and David R. Bundle pg 832; DOI: 10.1039/b009626l |
Synthesis and structure–activity relationships of di- and trisaccharide inhibitors for Shiga-like toxin Type 1 Pavel I. Kitov and David R. Bundle pg 838; DOI: 10.1039/b009685g |
Studies on aluminium mediated asymmetric Friedel–Crafts hydroxyalkylation reactions of pyridinecarbaldehydes Aase Sejr Gothelf Tore Hansen and Karl Anker Jørgensen pg 854; DOI: 10.1039/b009669p |
Halogenation of pyrazoloquinolines and pyrazoloisoquinolines. Theoretical analysis of the regioreactivity and cross-coupling of 3-halogen derivatives![]() Jan Pawlas Jeremy Greenwood Per Vedsø Tommy Liljefors Palle Jakobsen Per Olaf Huusfeldt and Mikael Begtrup pg 861; DOI: 10.1039/b006435l |
Conformational selection of non-hydrolyzable glycomimetics: the conformation of N,N![]() José Luis Muñoz Alicia García-Herrero Juan Luis Asensio F.-Isabelle Auzennaeau F. Javier Cañada and Jesús Jiménez-Barbero pg 867; DOI: 10.1039/b006965p |
Synthesis of uronic acid-containing xylans found in wood and pulp Stefan Oscarson and Pär Svahnberg pg 873; DOI: 10.1039/b009670a |
Chemoenzymatic synthesis of derivatives of a T-cell-stimulating peptide which carry tumor-associated carbohydrate antigens Shaji K. George Björn Holm Celso A. Reis Tilo Schwientek Henrik Clausen and Jan Kihlberg pg 880; DOI: 10.1039/b009567m |
The p-methoxybenzyl ether as an in situ-removable carbohydrate-protecting group: a simple one-pot synthesis of the globotetraose tetrasaccharide Sumita Bhattacharyya Bengt G. Magnusson Ulf Wellmar and Ulf J. Nilsson pg 886; DOI: 10.1039/b009448j |
Investigation of the Lewis acid mediated stereoselective cyclization of cationic aminyl radicals leading to substituted pyrrolidines Åsa Sjöholm Martin Hemmerling Nicolas Pradeille and Peter Somfai pg 891; DOI: 10.1039/b009391m |
Synthesis and evaluation of anti-HIV activity of 3-azido-4-(hydroxymethyl)tetrahydrofuran derivatives containing 2-(thymin-1-yl)methyl, 2-(cytosin-1-yl)methyl or 2-(adenin-9-yl)methyl substituents – a new series of AZT analogues Anne G. Olsen Claus Nielsen and Jesper Wengel pg 900; DOI: 10.1039/b009109j |
Synthesis of 1-azagalactofagomine, a potent galactosidase inhibitor Henrik Helligsø Jensen and Mikael Bols pg 905; DOI: 10.1039/b007973l |
Studies on the C-alkylation and C-allylation of small peptides employing glycyl radical intermediates Peter Blakskjær Lone Pedersen and Troels Skrydstrup pg 910; DOI: 10.1039/b005468m |
Professor Ei-ichi Negishi![]() Professor Ei-ichi Negishi pg 9-xi; DOI: 10.1039/b009326m |
Perkin 1 Abstracts: Natural Product Synthesis Andrew Gunn Jacqueline E. Milne Marcel de Puit and Duncan McArthur pg 9-xxi; DOI: 10.1039/b102281b |
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis Gideon Grogan Alexis Carstairs Ian Jackson Denise McIntyre Alan Watt Sabine Flitsch and Nicholas Turner pg 9-xiii; DOI: 10.1039/b102587m |
Perkin 1 Abstracts: Solid Phase Organic Synthesis Fabrice Anizon Jennifer Delaney Andrew Gunn Hassan Mamdani Catherine McCusker Fiona McKerlie and Tanya Wildman pg 9-xxvi; DOI: 10.1039/b103258p |
The use of supercritical fluids in synthetic organic chemistry R. Scott Oakes Anthony A. Clifford and Christopher M. Rayner pg 917; DOI: 10.1039/b101219n |
exo-Glycals from glycosyl cyanides. First generation of C-glycosylmethylene carbenes from 2,5- and 2,6-anhydroaldose tosylhydrazones Marietta Tóth and László Somsák pg 942; DOI: 10.1039/b102963k |
Synthesis of N-acylaziridines from ![]() Virginia R. Ward Matthew A. Cooper and A. David Ward pg 944; DOI: 10.1039/b102468j |
Indium-mediated allylation reactions of ![]() Jeong Ah Shin Kyung Il Choi Ae Nim Pae Hun Yeong Koh Han-Young Kang and Yong Seo Cho pg 946; DOI: 10.1039/b101111l |
Unusually facile palladium catalysed oxidation of imidazolidines and oxazolidines Alexandre Alexakis Isabelle Aujard Julien Pytkowicz Sylvain Roland and Pierre Mangeney pg 949; DOI: 10.1039/b010089g |
Synthesis and characterisation of ![]() ![]() Amal Mansour and Moshe Portnoy pg 952; DOI: 10.1039/b009640g |
Indium metal as a reducing agent in organic synthesis Michael R. Pitts Justin R. Harrison and Christopher J. Moody pg 955; DOI: 10.1039/b101712h |
Synthesis of thieno[2,3-b]quinoxalines and pyrrolo[1,2-a]quinoxalines from 2-haloquinoxalines Montserrat Armengol and John A. Joule pg 978; DOI: 10.1039/b101458g |
Synthesis of bicyclic nucleosides by ring-closing metathesis Jacob Ravn and Poul Nielsen pg 985; DOI: 10.1039/b101364p |
Development and application of allyl, 2-sulfonylethyl and 2-thioethyl carbamate linkers for solid phase N-acyliminium ion chemistry Jan H. van Maarseveen Wim J. N. Meester Johan J. N. Veerman Chris G. Kruse Pedro H. H. Hermkens Floris P. J. T. Rutjes and Henk Hiemstra pg 994; DOI: 10.1039/b100998m |
Asymmetric cycloaddition of anthrone and maleimides catalyzed by C2-chiral pyrrolidines Kouhei Uemae Satoshi Masuda and Yukio Yamamoto pg 1002; DOI: 10.1039/b100961n |
Triterpenoid total synthesis. Part 6. Synthesis of testudinariols A and B, triterpene metabolites of the marine mollusc Pleurobrancus testudinarius Masao Yoshida Hirosato Takikawa and Kenji Mori pg 1007; DOI: 10.1039/b100777g |
Synthesis of trans-3,4-dihydroxy-3,4-dihydrophenanthro[3,2-b![]() ![]() Subodh Kumar pg 1018; DOI: 10.1039/b100345n |
Rhodium(II)-carbenoid C–H insertion reactions in the synthesis of ![]() ![]() ![]() Pompiliu S. Aburel Christian Rømming and Kjell Undheim pg 1024; DOI: 10.1039/b100179p |
An efficient synthesis of highly functionalized asymmetric porphyrins with organolithium reagents Xiangdong Feng and Mathias O. Senge pg 1030; DOI: 10.1039/b100012h |
Solvent and ligand effects on selective mono- and dilithiation of 1-(chlorophenyl)pyrroles and 1-(methoxyphenyl)pyrroles![]() Katalin Fogassy Krisztina Kovács György M. Keser ![]() ![]() pg 1039; DOI: 10.1039/b100008j |
Synthesis and nicotinic acetylcholine-binding properties of epibatidine homologues: homoepibatidine and dihomoepibatidine John R. Malpass David A. Hemmings Anna L. Wallis Stephen R. Fletcher and Shailendra Patel pg 1044; DOI: 10.1039/b010178h |
Stereocontrol in a one-pot procedure for anionic oxy-Cope rearrangement followed by intramolecular aldol reaction Alistair P. Rutherford Cameron S. Gibb Richard C. Hartley and Jonathan M. Goodman pg 1051; DOI: 10.1039/b010138i |
The reaction of 1-(2,4,6-trimethylphenyl)-1,2-dihydrophosphinine 1-oxides with dimethyl acetylenedicarboxylate; a [4+2] or a [2+2] cycloaddition? György Keglevich Ágnes GyöngyvérVaskó András Dobó Krisztina Ludányi and László T ![]() pg 1062; DOI: 10.1039/b010080n |
[2+2] Heterodimers of methyl phenanthrene-9-carboxylate and benzene Taehee Noh Hyun Yu Youngmee Jeong Kyungmoon Jeon and Sukjin Kang pg 1066; DOI: 10.1039/b009846i |
Thermal decomposition of tert-butyl ortho-(phenylsulfanyl)- and ortho-(phenylsulfonyl)phenyliminoxyperacetates: The reactivity of thio-substituted iminyl radicals Rino Leardini Hamish McNab Matteo Minozzi and Daniele Nanni pg 1072; DOI: 10.1039/b009843o |
Gas-phase cyclisation reactions of 1-(2-arylthiophenyl)alkaniminyl and 2-(aryliminomethyl)thiophenoxyl radicals Tim Creed Rino Leardini Hamish McNab Daniele Nanni Iain S. Nicolson and David Reed pg 1079; DOI: 10.1039/b009844m |
Synthesis of multifunctionalized phosphonic acid esters via opening of oxiranes and azetidinium salts with phosphoryl-substituted carbanions Agata Bakalarz-Jeziorna Jan Heli ![]() ![]() pg 1086; DOI: 10.1039/b009720i |
Synthesis and isomerization of arene oxide metabolites of phenanthrene, triphenylene, dibenz[a,c]anthracene and dibenz[a,h]anthracene Suresh K. Balani I. N. Brannigan Derek R. Boyd Narain D. Sharma Francis Hempenstall and Allison Smith pg 1091; DOI: 10.1039/b009712h |
Phenylboronic acid as a labile protective agent: the selective derivatisation of 1,2,3-triols Vijaya Bhaskar K. Peter J. Duggan David G. Humphrey Guy Y. Krippner Victoria McCarl and Daniel A. Offermann pg 1098; DOI: 10.1039/b009450l |
Substituted triazines and pyrimidines from 1,3,5-triazine and a lithium amidinate, alkyl- or 1-azaallyl W. Marco Boesveld Peter B. Hitchcock and Michael F. Lappert pg 1103; DOI: 10.1039/b008681i |
Synthesis and reactions of some optically active epoxides formally derived from tertiary allylic alcohols Jamie F. Bickley Adam T. Gillmore Stanley M. Roberts John Skidmore and Alexander Steiner pg 1109; DOI: 10.1039/b008275i |
Cryptoregiochemistry of a Brassica napus fatty acid desaturase (FAD3): a kinetic isotope effect study Christopher K. Savile Darwin W. Reed Dauenpen Meesapyodsuk Patrick S. Covello and Peter H. Buist pg 1116; DOI: 10.1039/b008111f |
Clavulanic acid biosynthesis; the final steps M. Fulston M. Davison S. W. Elson N. H. Nicholson J. W. Tyler and S. R. Woroniecki pg 1122; DOI: 10.1039/b007009m |
The reaction of 2-(tetrazol-5-yl)alkyl ketones and of 2-(tetrazol-5-yl)alkanoic acid derivatives with lead tetraacetate. A novel method of preparation of alk-2-ynyl ketones and alk-2-ynoic acid derivatives![]() József Fetter Ildikó Nagy Le Thanh Giang Mária Kajtár-Peredy Antal Rockenbauer László Korecz and Gábor Czira pg 1131; DOI: 10.1039/b005286h |
Synthesis of phosphorus- and selenium-containing macrocycles and their complexation with Pd(II)Cl2 J. L. Li J. B. Meng Y. M. Wang J. T. Wang and T. Matsuura pg 1140; DOI: 10.1039/b005045h |
Perkin 1 Abstracts: Natural Product Synthesis Andrew Gunn Jacqueline E. Milne Marcel de Puit and Duncan McArthur pg 10-xv; DOI: 10.1039/b103457j |
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis Gideon Grogan Alexis Carstairs Ian Jackson Denise McIntyre Alan Watt Sabine Flitsch and Nicholas Turner pg 10-ix; DOI: 10.1039/b103527b |
A simple entry into enantiopure hydrindanes, hydroisoquinolones and diquinanes from 3,10-dioxygenated dicyclopentadienes: Application to the synthesis of (+)-coronafacic acid and a formal synthesis of (+)-coriolin Goverdhan Mehta and D. Srinivasa Reddy pg 1153; DOI: 10.1039/b009307f |
Conversion of homochiral amines, ![]() ![]() Ayhan S. Demir Idris M. Akhmedov Özge ![]() ![]() ![]() pg 1162; DOI: 10.1039/b008317h |
Electrochemical and yeast-catalysed ring-opening of isoxazoles in the synthesis of analogues of the herbicide Grasp![]() Christopher J. Easton Graham A. Heath C. Merrîcc M. Hughes Connie K. Y. Lee G. Paul Savage Gregory W. Simpson Edward R. T. Tiekink George J. Vuckovic and Richard D. Webster pg 1168; DOI: 10.1039/b008081k |
Syntheses and X-ray crystal structures of derivatives of 2,2![]() ![]() ![]() Pier Lucio Anelli Marino Brocchetta (the late) Costantino Maffezzoni Paola Paoli Patrizia Rossi Fulvio Uggeri and Massimo Visigalli pg 1175; DOI: 10.1039/b009666k |
A stereochemically flexible approach to pyrrolidines based on 5-endo-trig iodocyclisations of homoallylic sulfonamides Andrew D. Jones David W. Knight and David E. Hibbs pg 1182; DOI: 10.1039/b008537p |
Convenient synthesis of optically active 1,2-diol monosulfonates and terminal epoxides via oxazaborolidine-catalyzed asymmetric borane reduction of ![]() Byung Tae Cho Weon Ki Yang and Ok Kyung Choi pg 1204; DOI: 10.1039/b010155i |
1,2-Bis[(2-dimethylamino-2-thioxo-1-phenylethylidene)hydrazino]ethane: a new tetradentate ligand for Ni2+ Jean-Damien Charrier David Deniaud Alain Reliquet and Jean-Claude Meslin pg 1212; DOI: 10.1039/b101030l |
A multinuclear NMR study of the restricted rotation in a bi-imidazole nucleoside![]() Jukka Mäki Karel D. Klika Rainer Sjöholm and Leif Kronberg pg 1216; DOI: 10.1039/b010182f |
Solvent-free bentonite-catalyzed condensation of malonic acid and aromatic aldehydes under microwave irradiation André Loupy Suk-Jin Song Sun-Mee Sohn Young-Mee Lee and Tae-Woo Kwon pg 1220; DOI: 10.1039/b009803p |
A novel and convenient method for synthesizing unsymmetrical N-benzyloxycarbonyl-protected 1-amino-1-arylalkylphosphonate mixed diesters Jiaxi Xu and Nanyan Fu pg 1223; DOI: 10.1039/b008340m |
Synthesis and reactions of N-(azulen-1-ylmethylene)arylamines![]() Alexandru C. Razus Carmen Nitu Simona Carvaci Liviu Birzan Stefan A. Razus Mihaela Pop and Laszlo Tarko pg 1227; DOI: 10.1039/b100007l |
Molybdenum(0) and tungsten(0) catalysts with enhanced reactivity for allylic substitution: regioselectivity and solvent effects![]() Andrei V. Malkov Ian R. Baxendale Darren J. Mansfield and Pavel Ko ![]() pg 1234; DOI: 10.1039/b100903f |
A new and efficient approach to the synthesis of 6-amidino-2-oxopurines Brian L. Booth Isabel M. Cabral Alice M. Dias A. Paula Freitas Ana M. Matos Beja M. Fernanda Proença and Manuela Ramos Silva pg 1241; DOI: 10.1039/b010224p |
The semi-pinacol rearrangement of homochiral epoxyalcohols catalysed by rare earth triflates Jamie F. Bickley Bernhardt Hauer Paula C. A. Pena Stanley M. Roberts and John Skidmore pg 1253; DOI: 10.1039/b101838h |
A novel utilization of trifluoromethanide as a base: a convenient synthesis of trimethylsilylacetylene Mitsuhiro Yoshimatsu and Masako Kuribayashi pg 1256; DOI: 10.1039/b101537k |
Enantioselective amino acid recognition using acyclic thiourea receptors Graham M. Kyne Mark E. Light Mike B. Hursthouse Javier de Mendoza and Jeremy D. Kilburn pg 1258; DOI: 10.1039/b102298a |
Regio- and stereo-selective dioxygenase-catalysed cis-dihydroxylation of fjord-region polycyclic arenes Derek R. Boyd Narain D. Sharma John S. Harrison Martina A. Kennedy Christopher C. R. Allen and David T. Gibson pg 1264; DOI: 10.1039/b101833g |
The azomethine ylide strategy for ![]() David Brown Giles A. Brown Sarah R. Martel Denis Planchenault Evelyn Turmes Kenneth E. Walsh Richard Wisedale Neil J. Hales Colin W. G. Fishwick and Timothy Gallagher pg 1270; DOI: 10.1039/b010046n |
The azomethine ylide strategy for ![]() Giles A. Brown Sarah R. Martel Richard Wisedale Jonathan P. H. Charmant Neil J. Hales Colin W. G. Fishwick and Timothy Gallagher pg 1281; DOI: 10.1039/b010050l |
Intermolecular addition of alkyl radicals to imines in the absence and in the presence of a Lewis acid Nis Halland and Karl Anker Jørgensen pg 1290; DOI: 10.1039/b101762o |
Metabolites of the higher fungi. Part 33. Grammicin, a novel bicyclic C7H6O4 furanopyranol from the fungus Xylariagrammica (Mont.) Fr. Raymond L. Edwards Derek J. Maitland Pattama Pittayakhajonwut and Anthony J. S. Whalley pg 1296; DOI: 10.1039/b101708j |
Synthesis of substituted hexa-3,5-dienoic acid methyl esters from conjugated dienones Rishan Lang Nongkhlaw Ridaphun Nongrum and Bekington Myrboh pg 1300; DOI: 10.1039/b101242h |
One-step synthesis of 5-acylisothiazoles from furans Jérôme Guillard Christelle Lamazzi Otto Meth-Cohn Charles W. Rees Andrew J. P. White and David J. Williams pg 1304; DOI: 10.1039/b101157j |
An efficient procedure for cleavage of aziridines with various thiols promoted by ZnCl2 Jie Wu Xue-Long Hou and Li-Xin Dai pg 1314; DOI: 10.1039/b100591j |
Ebenaceae extractives. Part 11. The synthesis of 7-methyljuglone. A re-examination Oliver C. Musgrave and Douglas Skoyles pg 1318; DOI: 10.1039/b009531l |
Binding interactions between 3-aryl-1,2,4-oxadiazol-5-ones and a trisimidazoline base Anja Reichert Roland Fröhlich Roderick Ferguson and Arno Kraft pg 1321; DOI: 10.1039/b009451j |
Steroidal guanidines as enantioselective receptors for N-acyl ![]() ![]() Laurence J. Lawless Adrian G. Blackburn Alan J. Ayling M. Nieves Pérez-Payán and Anthony P. Davis pg 1329; DOI: 10.1039/b009215k |
Perkin 1 Abstracts: Natural Product Synthesis Andrew Gunn Jacqueline E. Milne Marcel de Puit and Duncan McArthur pg 12-xvi; DOI: 10.1039/b104270j |
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis Gideon Grogan Alexis Carstairs Ian Jackson Denise McIntyre Alan Watt Sabine Flitsch and Nicholas Turner pg 12-ix; DOI: 10.1039/b104422m |
An operationally simple and fully regiocontrolled formal total synthesis of the montanine-type Amaryllidaceae alkaloid ()-pancracine Martin G. Banwell Alison J. Edwards Katrina A. Jolliffe and Michael Kemmler pg 1345; DOI: 10.1039/b102252k |
Improved catalytic procedures for the copper(I)-promoted reactions of ![]() Christopher Hunter Richard F. W. Jackson and Harshad K. Rami pg 1349; DOI: 10.1039/b102446a |
Synthesis and some properties of 7H-naphth[3,2,1-cd![]() Noritaka Abe Hiroyuki Fujii Kahei Takase and Tadayoshi Morita pg 1353; DOI: 10.1039/b101333p |
Reactions of 7H-naphth[3,2,1-cd![]() Noritaka Abe Hiroyuki Fujii Kahei Takase and Tadayoshi Morita pg 1359; DOI: 10.1039/b101332g |
Synthesis of novel Hg2+ receptors based on N-benzyloxyamide derivatives and their application to anion-selective electrodes Shin-ichi Sasaki Tsuyoshi Amano Satoru Ozawa Tomomi Masuyama Daniel Citterio Hideaki Hisamoto Hisao Hori and Koji Suzuki pg 1366; DOI: 10.1039/b008978h |
Neighboring group effect of pyridazine and pyrazine rings for ![]() Tomoshige Kobayashi Kiyomi Miki Behrooz Nikaeen and Akira Ohta pg 1372; DOI: 10.1039/b101330k |
Dimethyl sulfoxide as a co-solvent dramatically enhances the enantioselectivity in lipase-catalysed resolutions of 2-phenoxypropionic acyl derivatives Keiichi Watanabe and Shin-ichi Ueji pg 1386; DOI: 10.1039/b100182p |
Regioselectivity and endo/exo selectivity in the cycloadditions of the phthalazinium dicyanomethanide 1,3-dipole with unsymmetrical alkene and alkyne dipolarophiles. Unexpected reversals of regiochemistry: a combined experimental and DFT theoretical study Richard N. Butler Anthony G. Coyne Patrick McArdle Desmond Cunningham and Luke A. Burke pg 1391; DOI: 10.1039/b101150m |
The preparation of novel thiophene-based macrocyclic Mannich bases Julie D. E. Chaffin John M. Barker and Patrick R. Huddleston pg 1398; DOI: 10.1039/b007661i |
Synthesis of new bis(tetrahydropyrrolo[3,4-b]carbazoles) with a functionalized diaryl spacer Farokh Mehrabani and Ulf Pindur pg 1406; DOI: 10.1039/b006899n |
Palladium catalysed elaboration of codeine and morphine Stephen G. Davies Christopher J. Goodwin Dirk Pyatt and Andrew D. Smith pg 1413; DOI: 10.1039/b102581n |
Design of potential new HIV protease inhibitors: enantioconvergent synthesis of new pyrrolidin-3-ol, and pyrrolidin-3-one peptide conjugates Jérôme Courcambeck Frédéric Bihel Céline De Michelis Gilles Quéléver and Jean Louis Kraus pg 1421; DOI: 10.1039/b101584m |
Does water suppress the racemization and decomposition of amino acids? Yuusaku Yokoyama Hidemasa Hikawa and Yasuoki Murakami pg 1431; DOI: 10.1039/b102254g |
Use of dissolving metals in the partial reduction of pyridines: formation of 2-alkyl-1,2-dihydropyridines![]() Timothy J. Donohoe Andrew J. McRiner Madeleine Helliwell and Peter Sheldrake pg 1435; DOI: 10.1039/b101662h |
Stereoselectivity of cyclisations viaN-acyliminium ions to form pyrido[2![]() ![]() Abood A. Bahajaj John M. Vernon and Giles D. Wilson pg 1446; DOI: 10.1039/b009316p |
Coordination of (![]() Magnus Gustafsson Karl-Erik Bergqvist and Torbjörn Frejd pg 1452; DOI: 10.1039/b101464l |
Synthesis of ![]() ![]() Pompiliu S. Aburel Christian Rømming Kuangbiao Ma and Kjell Undheim pg 1458; DOI: 10.1039/b101462p |
Professor C. Robin Ganellin FRS![]() Professor C. Robin Ganellin pg 13-vii; DOI: 10.1039/b101382n |
Perkin 1 Abstracts: Solid Phase Organic Synthesis Fabrice Anizon Jennifer Delaney Andrew Gunn Hassan Mamdani Catherine McCusker Fiona McKerlie and Tanya Wildman pg 13-ix; DOI: 10.1039/b104302c |
Preparative biotransformations Stanley M. Roberts pg 1475; DOI: 10.1039/b101682m |
Chiral pyridylimidazolines: synthesis, arene ruthenium complexes and application in asymmetric catalysis Adam J. Davenport David L. Davies John Fawcett and David R. Russell pg 1500; DOI: 10.1039/b103175a |
The scope and limitation of the [1,4]-Sbenzyl participation and debenzylation in the stereochemically controlled synthesis of substituted thiolanes Jason Eames Nikolai Kuhnert and Stuart Warren pg 1504; DOI: 10.1039/b102737a |
Rearrangement of 18-iodo- and 20-iodopregnanes mediated by iodosyl derivatives![]() Daniel Nicoletti Alberto A. Ghini Ricardo F. Baggio M. Teresa Garland and Gerardo Burton pg 1511; DOI: 10.1039/b102688g |
Aziridination of cyclic dienes with enantiopure 3-acetoxyaminoquinazolin-4(3H)-ones Robert S. Atkinson and Christopher K. Meades pg 1518; DOI: 10.1039/b102592a |
[11C]/(13C)Carbon monoxide in palladium-mediated synthesis of imides Farhad Karimi Tor Kihlberg and Bengt Långström pg 1528; DOI: 10.1039/b102524b |
Serial synthesis of oxa[3.n]cyclophanes and homooxacalix[n]arenes via reductive coupling of arenedialdehydes, and their X-ray structures Naoki Komatsu and Takefumi Chishiro pg 1532; DOI: 10.1039/b102031p |
Highly effective and recyclable chiral auxiliaries: a study of the synthesis and use of three 4-isopropyl-5,5-diaryloxazolidin-2-ones Karen Alexander (née Gillon) Stuart Cook Colin L. Gibson and Alan R. Kennedy ![]() pg 1538; DOI: 10.1039/b102020j |
Biosynthesis of polyoxypeptin A: novel amino acid 3-hydroxy-3-methylproline derived from isoleucine Kazuo Umezawa Yoko Ikeda Osamu Kawase Hiroshi Naganawa and Shinichi Kondo pg 1550; DOI: 10.1039/b101942m |
Synthesis of pentenoic acid analogs as potential anti-influenza agents Scott C. Mauldin William J. Hornback and John E. Munroe pg 1554; DOI: 10.1039/b101702k |
C-Alkylation of hydroxyarenes by Michael reaction Henryk Krawczyk and Ryszard Bodalski pg 1559; DOI: 10.1039/b101210j |
Synthesis of a new analogue of BINOL based on a homodimer of substituted 1-hydroxypyrazole Øystein Rist and Mikael Begtrup pg 1566; DOI: 10.1039/b010126p |
Conversion of alkanenitriles to amidines and carboxylic acids mediated by a cobalt(II)–ketoxime system![]() Maximilian N. Kopylovich Vadim Yu. Kukushkin M. Fátima C. Guedes da Silva Matti Haukka João J. R. Fraústo da Silva and Armando J. L. Pombeiro pg 1569; DOI: 10.1039/b101337h |
Perkin 1 Abstracts: Natural Product Synthesis Andrew Gunn Jacqueline E. Milne Marcel de Puit and Duncan McArthur pg 14-xv; DOI: 10.1039/b105193h |
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis Gideon Grogan Alexis Carstairs Ian Jackson Denise McIntyre Alan Watt Sabine Flitsch and Nicholas Turner pg 14-ix; DOI: 10.1039/b105469b |
2-Chloro-1,1-dimethyl-1H-cycloprop[e]azulene, the first cyclopropa-fused azulene Alan D. Payne and Dieter Wege pg 1579; DOI: 10.1039/b104346n |
Diastereocontrolled Strecker reaction using (S)-5-phenylmorpholin-2-one Laurence M. Harwood Michael G. B. Drew David J. Hughes and Richard J. Vickers pg 1581; DOI: 10.1039/b104052a |
Isogalactofagomine lactam. A neutral nanomolar galactosidase inhibitor Helmer Søhoel Xifu Liang and Mikael Bols pg 1584; DOI: 10.1039/b103831c |
Preparation of tetraalkylformamidinium salts and related species as precursors to stable carbenes Roger W. Alder Michael E. Blake Simone Bufali Craig P. Butts A. Guy Orpen Jan Schütz and Stuart J. Williams pg 1586; DOI: 10.1039/b104110j |
Electrochemical oxidation of aspidofractinine-type alkaloids: Formation of kopsine, kopsidine, kopsinitarine and bisindole derivatives Toh-Seok Kam Tuck-Meng Lim and Guan-Huat Tan pg 1594; DOI: 10.1039/b103962h |
Synthesis of nonpolar peptide nucleic acid monomers containing fluoroaromatics Norio Shibata Biplab Kumar Das Hiroshi Honjo and Yoshio Takeuchi pg 1605; DOI: 10.1039/b103170h |
C-Glycosylation of tri-O-benzyl-2-deoxy-D-glucose: synthesis of naphthyl-substituted 3,6-dioxabicyclo[3.2.2]nonanes Margaret A. Brimble and Timothy J. Brenstrum pg 1612; DOI: 10.1039/b102807n |
Synthesis of a 2-deoxyglucosyl analogue of medermycin Margaret A. Brimble and Timothy J. Brenstrum pg 1624; DOI: 10.1039/b103080a |
Scope and limitations in sulfur ylide mediated catalytic asymmetric aziridination of imines: use of phenyldiazomethane, diazoesters and diazoacetamides Varinder K. Aggarwal Marco Ferrara Christopher J. O'Brien Alison Thompson Ray V. H. Jones and Robin Fieldhouse pg 1635; DOI: 10.1039/b102578n |
Synthesis of dithiaporphyrin-based singlet–singlet energy transfer systems Duraisamy Kumaresan Neeraj Agarwal and Mangalampalli Ravikanth pg 1644; DOI: 10.1039/b102349g |
A general and highly regio and stereoselective method for the synthesis of (E)-2-(2-arylvinyl)-3,1-benzoxathiin-4-ones through palladium–copper catalysis Bidisha Nandi and Nitya G. Kundu pg 1649; DOI: 10.1039/b102306n |
The first example of a new type of acyclic, achiral nucleoside analogue: 1-[3-hydroxy-2-(hydroxymethyl)prop-1-enyl]thymine Daniel Sejer Pedersen Thomas Boesen Anne B. Eldrup Benedikte Kiær Christian Madsen Ulla Henriksen and Otto Dahl pg 1656; DOI: 10.1039/b101759o |
Synthesis of 6-substituted purin-2-ones with potential cytokinin activity Geir Andresen Aud Berglen Eriksen Bjørn Dalhus Lise-Lotte Gundersen and Frode Rise pg 1662; DOI: 10.1039/b101327k |
Design and preparation of serine–threonine protein phosphatase inhibitors based upon the nodularin and microcystin toxin structures. Part 3 Kerri L. Webster Antony B. Maude Michael E. O'Donnell Amit P. Mehrotra and David Gani pg 1673; DOI: 10.1039/b100401h |
Serine–threonine protein phosphatase inhibitors derived from nodularin: role of the 2-methyl and 3-diene groups in the Adda residue and the effect of macrocyclic conformational restraint Michael E. O'Donnell Jonathan Sanvoisin and David Gani pg 1696; DOI: 10.1039/b100402f |
A generic medium throughput activity assay procedure for serine–threonine protein phosphatases using 14C-labelled N-acetyl-Arg-Arg-Ala-Thr(P)-Val-Ala Jonathan Sanvoisin John R. Pollard Pantea Hormozdiari Walter H. J. Ward and David Gani pg 1709; DOI: 10.1039/b100403o |
![]() Yongsheng Chen Wei Zhang Xi Chen Jianqiang Wang and Peng George Wang pg 1716; DOI: 10.1039/b100356i |
Emanuela Erba Donato Pocar and Pasqualina Trimarco pg 1723; DOI: 10.1039/b008531f |
Perkin 1 Abstracts: Solid Phase Organic Synthesis Fabrice Anizon Jennifer Delaney Andrew Gunn Hassan Mamdani Catherine McCusker Fiona McKerlie and Tanya Wildman pg 15-vii; DOI: 10.1039/b105192j |
Catalytic asymmetric processes Heather Tye and Paul J. Comina pg 1729; DOI: 10.1039/a900862d |
Bio-organic synthesis of a newly isolated peptide metastin, metastasis suppressor gene KiSS-1 processing product Osamu Nishimura Masato Suenaga Takao Yamada Takashi Itoh Nobuyuki Koyama Mitsuhiro Wakimasu Tetsuya Ohtaki Chieko Kitada and Masahiko Fujino pg 1748; DOI: 10.1039/b104948h |
Unsymmetrically substituted furoxans. Part 18. Smiles rearrangement in furoxan systems and in related furazans Donatella Boschi Giovanni Sorba Massimo Bertinaria Roberta Fruttero Rosella Calvino and Alberto Gasco pg 1751; DOI: 10.1039/b104845g |
Intramolecular azomethine ylide cycloaddition reactions to give octahydroindoles Iain Coldham Katherine M. Crapnell Jonathan D. Moseley and Rémi Rabot pg 1758; DOI: 10.1039/b104390k |
First efficient synthesis of ()-erythro-roccellic acid Sivaprakasam Mangaleswaran and Narshinha P. Argade pg 1764; DOI: 10.1039/b104105n |
Stereoselective syntheses of 1H-imidazo[2,1-a]isoindole-2,5(3H,9bH)-diones Alan R. Katritzky Yong-Jiang Xu Hai-Ying He and Peter J. Steel pg 1767; DOI: 10.1039/b104060j |
The first efficient method for the intramolecular trapping of benzynes by phenols: a new approach to xanthenes David W. Knight and Paul B. Little pg 1771; DOI: 10.1039/b103834f |
endo/exo Facial selectivities in cycloaddition reactions of substituted 1,2,3-triazolium-1-methanides, unstabilised 1,3-dipoles, with some alkene dipolarophiles: models for 1,2,3-triazolium-1-aminides: new tetracyclic pyrrolo[1,2-c][1,2,3]benzotriazole structures: azolium 1,3-dipoles R. N. Butler and Leonie M. Wallace pg 1778; DOI: 10.1039/b103759p |
Atropisomeric ![]() Alan C. Spivey Adrian Maddaford David P. Leese and Alison J. Redgrave pg 1785; DOI: 10.1039/b103385a |
Azafulvenium methides: new extended dipolar systems Oliver B. Sutcliffe Richard C. Storr Thomas L. Gilchrist and Paul Rafferty pg 1795; DOI: 10.1039/b103250j |
Xanthen-9-ylidene protecting groups in glycerol chemistry Colin B. Reese and Hongbin Yan pg 1807; DOI: 10.1039/b102923c |
Intramolecular cycloadditions of N-alkenoyl aryl azides Luisa Garanti Giorgio Molteni and Gianluigi Broggini pg 1816; DOI: 10.1039/b102686k |
Novel synthetic routes to nitrogen-bridged tricyclic derivatives of pyrrolo[2,1,5-cd]indolizine and pyrrolo[2,1,5-de]quinolizine derived from 2-acyl-N-(acylmethyl)pyridinium halides Jiaxin Hu Xin Jiang Ting He Jian Zhou Yuefei Hu and Hongwen Hu pg 1820; DOI: 10.1039/b102449n |
A regio- and stereo-selective synthesis of 2-hydroxy-3-methylochromycinone in three steps from 2-bromo-5-acetoxy-1,4-naphthoquinone and 1-acetoxy-3,3-dimethyl-5-vinylcyclohexa-1,5-diene Tomas Rozek John H. Bowie Simon M. Pyke Brian W. Skelton and Allan H. White pg 1826; DOI: 10.1039/b101756j |
Asymmetric synthesis of (+)-loline, a pyrrolizidine alkaloid from rye grass and tall fescue Paul R. Blakemore Sung-Kee Kim Volker K. Schulze James D. White and Alexandre F. T. Yokochi pg 1831; DOI: 10.1039/b103936a |
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis Gideon Grogan Alexis Carstairs Ian Jackson Denise McIntyre Alan Watt Sabine Flitsch and Nicholas Turner pg 16-vii; DOI: 10.1039/b106521c |
Perkin 1 Abstracts: Natural Product Synthesis Andrew Gunn Jacqueline E. Milne Marcel de Puit and Duncan McArthur pg 16-xiii; DOI: 10.1039/b106740k |
A concise and efficient stereoselective synthesis of protected (2R,1![]() ![]() Debendra K. Mohapatra pg 1851; DOI: 10.1039/b105503h |
Synthesis of 2-heteroaryl-3-hydroxypyridines by ring expansion reactions of 2-acylfurans with ammonia Richard W. J. Chubb Martin R. Bryce and Brian Tarbit pg 1853; DOI: 10.1039/b105228b |
A conformationally locked tricyclic nucleoside. Synthesis, crystal structure and incorporation into oligonucleotides Jacob Ravn Niels Thorup and Poul Nielsen pg 1855; DOI: 10.1039/b104438a |
Carotenoids and related polyenes. Part 6. Stereoselective synthesis of astaxanthin analogues and their antioxidant activities Yumiko Yamano Yuki Sato Yasuko Watanabe Koshi Namikawa Wataru Miki and Masayoshi Ito pg 1862; DOI: 10.1039/b104338m |
Synthesis of novel all-cis-functionalized cyclopropane template-assembled collagen models Shoko Yamazaki Mari Sakamoto Michiko Suzuri Masamitsu Doi Takashi Nakazawa and Yuji Kobayashi pg 1870; DOI: 10.1039/b103887g |
Direct synthesis of Fmoc-protected amino acids using organozinc chemistry: application to polymethoxylated phenylalanines and 4-oxoamino acids Hervé J. C. Deboves Christian A. G. N. Montalbetti and Richard F. W. Jackson pg 1876; DOI: 10.1039/b103832j |
Stereoselective Baeyer–Villiger oxidation of some bridged bicyclic diketones Eugenius Butkus and Sigitas Ston ![]() pg 1885; DOI: 10.1039/b103564a |
A new route to polyoxygenate C and D rings of steroids by oxidation of a ![]() Donato Sica Domenica Musumeci Franco Zollo and Simona De Marino pg 1889; DOI: 10.1039/b103389c |
Trapping highly reactive dipolarophiles. Exploiting the mechanism associated with the azomethine ylide strategy for ![]() Giles A. Brown Kirsty M. Anderson Jonathan M. Large Denis Planchenault Dominique Urban Neil J. Hales and Timothy Gallagher pg 1897; DOI: 10.1039/b103271m |
Synthesis, structure, and reactivity of (tropon-2-ylimino)arsorane and in situ generation of its stiborane and -bismuthorane analogues: reactions with heterocumulenes and an activated acetylene giving heteroazulenes Makoto Nitta Yuhki Mitsumoto and Hiroyuki Yamamoto pg 1901; DOI: 10.1039/b103098c |
Synthesis and properties of 2-nitrosoadenosine Martin J. Wanner and Gerrit-Jan Koomen pg 1908; DOI: 10.1039/b102897a |
Enantioselective synthesis of ![]() ![]() Aparecida M. Kawamoto and Martin Wills pg 1916; DOI: 10.1039/b102895m |
Chemical consequences of fluorine substitution. Part 1. Experimental and theoretical results on Diels–Alder reactions of ![]() ![]() Thomas Ernet Andreas H. Maulitz Ernst-Ulrich Würthwein and Günter Haufe pg 1929; DOI: 10.1039/b102684b |
Ultrasound-accelerated synthesis of 3,4-dihydropyrimidin-2(1H)-ones with ceric ammonium nitrate Jhillu S. Yadav Basi V. Subba Reddy Kasireddy Bhaskar Reddy Kavuda Sarita Raj and Attaluri R. Prasad pg 1939; DOI: 10.1039/b102565c |
The syntheses of three highly unsaturated marine lipid hydrocarbons Anne Kristin Holmeide Lars Skattebøl and Magne Sydnes pg 1942; DOI: 10.1039/b101889m |
Ketoester methacrylate resin, secondary amine clean-up in the presence of primary amines Zhanru Yu Sonia Alesso David Pears Paul A. Worthington Richard W. A. Luke and Mark Bradley pg 1947; DOI: 10.1039/b101395p |
One-pot synthesis of unsymmetrical biaryls from suitably functionalized 2H-pyran-2-ones through carbanion-induced ring-transformation reactions Vishnu J. Ram Pratibha Srivastava Nidhi Agarwal Ashoke Sharon and Prakas R. Maulik pg 1953; DOI: 10.1039/b009725j |
A novel system for the preparation of orphan receptor ligand peptides Osamu Nishimura Nobuyuki Koyama Takashi Itoh Masato Suenaga Takeo Moriya Masanori Miwa Yoko Tanaka Chieko Kitada and Masahiko Fujino pg 1960; DOI: 10.1039/b009566o |
Perkin 1 Abstracts: Solid Phase Organic Synthesis Fabrice Anizon Jennifer Delaney Andrew Gunn Hassan Mamdani Catherine McCusker Fiona McKerlie and Tanya Wildman pg 17-vii; DOI: 10.1039/b106738a |
Generation and reactivity of ![]() Richard W. Friesen pg 1969; DOI: 10.1039/b104589j |
![]() Martin G. Banwell Joanne E. Harvey and Katrina A. Jolliffe pg 2002; DOI: 10.1039/b106369n |
Is N-acetylornithine aminotransferase the real N-succinyl-LL-diaminopimelate aminotransferase in Escherichia coli and Mycobacterium smegmatis? Russell J. Cox and Paul S. H. Wang pg 2006; DOI: 10.1039/b106146c |
Oxidations of 3-alkenyltetronic acids with dimethyldioxirane (DMD) and air: regioselectivity and formation of a spirotricyclic hemiketal endoperoxide lactone Rainer Schobert Sven Siegfried Jochen Weingärtner and Mark Nieuwenhuyzen pg 2009; DOI: 10.1039/b104227k |
Cyclic ureas as ortho directing substituents Jon-Paul Meigh Mercedes Álvarez and John A. Joule pg 2012; DOI: 10.1039/b105420c |
Synthesis and in vitro enzyme activity of aza, oxa and thia derivatives of bacterial cell wall biosynthesis intermediates Russell J. Cox and Paul S. H. Wang pg 2022; DOI: 10.1039/b105117m |
Acid- or base-promoted photostimulated homolytic tert-butylation of pyridines and thiophenes Byeong Hyo Kim Insik Jeon Tae Hee Han Hae Jin Park and Young Moo Jun pg 2035; DOI: 10.1039/b104906m |
Chiral synthons from carvone. Part 50. Enantiospecific approaches to both enantiomers of bicyclo[4.3.0]nonane-3,8-dione derivatives A. Srikrishna and T. Jagadeeswar Reddy pg 2040; DOI: 10.1039/b104253j |
An alternative approach to the synthesis of a recombinant galanin-like peptide (GALP) Takashi Itoh Nobuyuki Koyama Masanori Miwa Masato Suenaga Tetsuya Ohtaki Chieko Kitada Osamu Nishimura and Masahiko Fujino pg 2047; DOI: 10.1039/b103835b |
Friedel–Crafts reactions of a sulfonyl-substituted vinylic epoxide with various aromatics Svante Brandänge Jan-Erling Bäckvall and Hans Leijonmarck pg 2051; DOI: 10.1039/b103582g |
Influence of ring size on the outcome of sulfide contraction reactions with thiolactams. Isolation of bicyclic ketene S,N-acetals and thioisomnchnones Joseph P. Michael Charles B. de Koning Christiaan W. van der Westhuyzen and Manuel A. Fernandes pg 2055; DOI: 10.1039/b103560f |
Synthesis of glycero amino acid-based surfactants. Part 1. Enzymatic preparation of rac-1-O-(N![]() Carmen Morán María Rosa Infante and Pere Clapés pg 2063; DOI: 10.1039/b103132p |
Synthesis of imines, diimines and macrocyclic diimines as possible ligands, in aqueous solution Alina Simion Cristian Simion Tadeshige Kanda Satoko Nagashima Yoshiharu Mitoma Tomoko Yamada Keisuke Mimura and Masashi Tashiro pg 2071; DOI: 10.1039/b102749m |
An efficient approach to (E)-![]() Joo Hwan Cha Ae Nim Pae Kyung Il Il Choi Yong Seo Cho Hun Yeong Koh and Eun Lee pg 2079; DOI: 10.1039/b102532p |
Highly peri- and stereoselective intramolecular photocycloaddition and cyclisation of N-(1-naphthylethyl)prop-2-enamides Shigeo Kohmoto Yoshiyuki Miyaji Masaru Tsuruoka Keiki Kishikawa Makoto Yamamoto and Kazutoshi Yamada pg 2082; DOI: 10.1039/b100678i |
Medium-sized cyclophanes. Part 58. Synthesis and conformational studies of [2.n]metacyclophan-1-enes and [n.1]metacyclophanes Takehiko Yamato Koji Fujita and Hirohisa Tsuzuki pg 2089; DOI: 10.1039/b010075g |
Isolation, structure and synthesis of mahafacyclin B, a cyclic heptapeptide from the latex of Jatropha mahafalensis Carine Baraguey Alain Blond Florine Cavelier Jean-Louis Pousset Bernard Bodo and Catherine Auvin-Guette pg 2098; DOI: 10.1039/b008538n |
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis Gideon Grogan Alexis Carstairs Ian Jackson Denise McIntyre Alan Watt Sabine Flitsch and Nicholas Turner pg 18-ix; DOI: 10.1039/b107562b |
Perkin 1 Abstracts: Natural Product Synthesis Andrew Gunn Jacqueline E. Milne Marcel de Puit and Duncan McArthur pg 18-xv; DOI: 10.1039/b107661m |
Protecting groups Krzysztof Jarowicki and Philip Kocienski pg 2109; DOI: 10.1039/b103282h |
Garner's aldehyde Xifu Liang Jens Andersch and Mikael Bols pg 2136; DOI: 10.1039/b101054i |
First highly stereoselective synthesis of (+)-dihydrosesamin, a trisubstituted tetrahydrofuran-type of lignan, by using highly erythro-selective aldol condensation Satoshi Yamauchi Teruhisa Tanaka and Yoshiro Kinoshita pg 2158; DOI: 10.1039/b105419h |
Functionalised bicyclic alcohols by enantioselective ![]() David M. Hodgson Iain D. Cameron Martin Christlieb Rebecca Green Gary P. Lee and Lesley A. Robinson pg 2161; DOI: 10.1039/b105369h |
DISAL glycosyl donors for efficient glycosylations under acidic conditions: Application to solid-phase oligosaccharide synthesis Lars Petersen and Knud J. Jensen pg 2175; DOI: 10.1039/b105872j |
Double intramolecular hetero Diels–Alder reactions of ![]() ![]() ![]() Nicholas Bushby Christopher J. Moody David A. Riddick and Ian R. Waldron pg 2183; DOI: 10.1039/b105409k |
A chemoenzymatic synthesis of the carbobicyclic core associated with CP-225,917 and CP-263,114 (phomoidrides A and B) Martin G. Banwell Kenneth J. McRae and Anthony C. Willis pg 2194; DOI: 10.1039/b105376k |
Studies related to carba-pyranoses: a strategy for the synthesis of ![]() David S. Larsen Roger J. Lins Richard J. Stoodley and Nicholas S. Trotter pg 2204; DOI: 10.1039/b105374b |
Synthesis of ellipticine by reaction of 1-(4-methoxybenzyl)indole-2,3-dicarboxylic anhydride with (3-bromo-4-pyridyl)triisopropoxytitanium Yasuyoshi Miki Hiroko Hachiken and Norihide Yanase pg 2213; DOI: 10.1039/b105116b |
The first stereospecific synthesis of L-tetrahydrodipicolinic acid; a key intermediate of diaminopimelate metabolism Jennifer F. Caplan Andrew Sutherland and John C. Vederas pg 2217; DOI: 10.1039/b105091p |
One-step iodination of the diazocyclopentadien-2-ylcarbonyl group—a new and convenient preparation of effective radiolabelled photoaffinity probes Elena L. Vodovozova Ekaterina V. Tsibizova and Julian G. Molotkovsky pg 2221; DOI: 10.1039/b104945n |
A highly efficient, stereoselective oxyfunctionalization of unactivated carbons in steroids with dimethyldioxirane Takashi Iida Takeru Yamaguchi Ryusei Nakamori Masahiro Hikosaka Nariyasu Mano Junichi Goto and Toshio Nambara pg 2229; DOI: 10.1039/b104938k |
Synthesis of a thiophene analogue of kuanoniamine A Yvette A. Jackson Seon A. Hepburn and William F. Reynolds pg 2237; DOI: 10.1039/b104710h |
Allene synthesis by an asymmetric Baylis–Hillman style reaction on vinylphosphine oxides David J. Fox Jonathan A. Medlock Richard Vosser and Stuart Warren pg 2240; DOI: 10.1039/b104436m |
Intramolecular [2+2] photocycloadditions as an approach towards the right-hand side of solanoeclepin A Richard H. Blaauw Jorg C. J. Benningshof Angeline E. van Ginkel Jan H. van Maarseveen and Henk Hiemstra pg 2250; DOI: 10.1039/b104165g |
[2 + 2] Cycloaddition reaction of cycloheptatriene with dichloroketene. A novel and efficient synthetic strategy for the synthesis of 2-hydroxyazulene Ryuji Yokoyama Shunji Ito Masataka Watanabe Nobuyuki Harada Chizuko Kabuto and Noboru Morita pg 2257; DOI: 10.1039/b104164a |
Highly selective one-pot conversion of THP and MOM ethers to acetates by indium triiodide-catalysed deprotection and subsequent transesterification by ethyl acetate Brindaban C. Ranu and Alakananda Hajra pg 2262; DOI: 10.1039/b104055n |
Chemoselectivity in reactions of an ![]() ![]() Jiaxi Xu Qihan Zhang Liangbi Chen and Hui Chen pg 2266; DOI: 10.1039/b103173m |
Synthesis and thermal transformation of stable monocyclic ![]() Hiroshi Shimizu Noriaki Kudo Tadashi Kataoka and Mikio Hori pg 2269; DOI: 10.1039/b102806p |
Oxidative radical cyclizations of malonate enolates induced by the ferrocenium ion – a remarkable influence of enolate counterion and additives Ullrich Jahn and Philip Hartmann pg 2277; DOI: 10.1039/b102211n |
Regio- and stereoselective synthesis of fluoroalkadienes using ![]() Masanori Yoshida Dai Nagahara Tsuyoshi Fukuhara Norihiko Yoneda and Shoji Hara pg 2283; DOI: 10.1039/b101836l |
An efficient synthesis of julibrosides related to neosaponin Yuguo Du Meimei Zhang and Fanzuo Kong pg 2289; DOI: 10.1039/b009955o |
Efficient formation of lipophilic dihydroxotin(IV) porphyrins and bis-porphyrins Maxwell J. Crossley Pall Thordarson and Richard A.-S. Wu pg 2294; DOI: 10.1039/b104846p |
Perkin 1 Abstracts: Solid Phase Organic Synthesis Jennifer Delaney Andrew Gunn Hassan Mamdani and Tanya Wildman pg 19-ix; DOI: 10.1039/b107265j |
Saturated oxygen heterocycles Mark C. Elliott and Eve Williams pg 2303; DOI: 10.1039/b007290g |
Novel and facile catalytic synthesis of 2,4-dioxopyrido[2,3-d]pyrimidine derivatives in water Noé Rosas Pankaj Sharma Cecilio Alvarez Armando Cabrera Rodrigo Ramírez Alejandro Delgado and Henri Arzoumanian pg 2341; DOI: 10.1039/b101374m |
Enantiospecific syntheses of pseudopterosin aglycones. Part 1. Synthesis of the putative aglycone of pseudopterosin G–J via an A![]() ![]() Robert Chow Philip J. Kocienski Alexander Kuhl Jean-Yves LeBrazidec Kenneth Muir and Paul Fish pg 2344; DOI: 10.1039/b102960f |
Enantiospecific syntheses of pseudopterosin aglycones. Part 2. Synthesis of pseudopterosin K–L aglycone and pseudopterosin A–F aglycone via a B![]() ![]() Philip J. Kocienski Alessandro Pontiroli and Liu Qun pg 2356; DOI: 10.1039/b102961b |
Unusual stereoselectivity in the alkylation of pyroglutamate ester urethanes Jean-Damien Charrier James E. S. Duffy Peter B. Hitchcock and Douglas W. Young pg 2367; DOI: 10.1039/b106451g |
Synthesis of epibatidine isomers: endo-5- and 6- (6![]() ![]() Caroline D. Cox John R. Malpass John Gordon and Alan Rosen pg 2372; DOI: 10.1039/b106212n |
A concise C-glycosyl amino acid synthesis by alkenyl C-glycoside–vinyloxazolidine cross-metathesis. Synthesis of glycosyl serine, asparagine and hydroxynorvaline isosteres Alessandro Dondoni Pier Paolo Giovannini and Alberto Marra pg 2380; DOI: 10.1039/b106029p |
An improved, versatile synthesis of the GABAC antagonists (1,2,5,6-tetrahydropyridin-4-yl)methylphosphinic acid (TPMPA) and (piperidin-4-yl)methylphosphinic acid (P4MPA) Jane R. Hanrahan Kenneth N. Mewett Mary Chebib Peter M. Burden and Graham A. R. Johnston pg 2389; DOI: 10.1039/b105989k |
Three-component synthesis of (E)-![]() ![]() Rainer Schobert Sven Siegfried and Gary J. Gordon pg 2393; DOI: 10.1039/b105745f |
Simple and selective one-pot replacement of the N-methyl group of tertiary amines by quaternization and demethylation with sodium sulfide or potassium thioacetate: an application to the synthesis of pergolide Luigi Anastasia Giuliana Cighetti and Pietro Allevi pg 2398; DOI: 10.1039/b104843k |
A practical protocol for the synthesis of 3-hydroxy-4,5-disubstituted pyridine derivatives from acyclic compounds Luigi Anastasia ![]() pg 2404; DOI: 10.1039/b105478n |
Synthesis of bis[1,2]dithiolo[1,4]thiazine imines from Hnig's base Stanislav A. Amelichev Susana Barriga Lidia S. Konstantinova Tatjana B. Markova Oleg A. Rakitin Charles W. Rees and Tomás Torroba pg 2409; DOI: 10.1039/b105243h |
Synthesis and stereochemistry of new tetraspiro-1,3-dioxanes Dorina Opris Ion Grosu Loïc Toupet Gérard Plé Anamaria Terec Sorin Mager and Luminita Muntean pg 2413; DOI: 10.1039/b104604g |
Synthesis of 6,7-dehydroartemisinic acid Lai-King Sy and Geoffrey D. Brown pg 2421; DOI: 10.1039/b104471k |
Retinoids and related compounds. Part 26. Synthesis of (11Z)-8,18-propano- and methano-retinals and conformational study of the rhodopsin chromophore Akimori Wada Masako Tsutsumi Yuka Inatomi Hiroo Imai Yoshinori Shichida and Masayoshi Ito pg 2430; DOI: 10.1039/b104394n |
Synthesis and catalytic properties of p-acylthio(phenylacetylene)n substituted chiral manganese salen complexes Morten Nielsen and Kurt V. Gothelf pg 2440; DOI: 10.1039/b104103g |
Stereoselective synthesis of a set of two functionalized (E)-alkene dipeptide isosteres of L-amino acid-L-Glu and L-amino acid-D-Glu Shinya Oishi Hirokazu Tamamura Masaki Yamashita Yoshihiko Odagaki Nobuyuki Hamanaka Akira Otaka and Nobutaka Fujii pg 2445; DOI: 10.1039/b103833h |
Selective radical-chain epimerisation at electron-rich chiral tertiary C–H centres using thiols as protic polarity-reversal catalysts Hai-Shan Dang Brian P. Roberts and Derek A. Tocher ![]() pg 2452; DOI: 10.1039/b103558b |
Novel phosphitylating reagents containing a phosphorus–fluorine bond and their application in efficient synthesis of phosphorofluoridates and phosphorofluoridothionates Wojciech D ![]() pg 2462; DOI: 10.1039/b103082p |
Studies on polycyclic fluoroazaarenes: synthesis of trans-9-fluoro- and -11-fluoro 3,4-dihydroxy-3,4-dihydrobenz[c]acridines as potential proximate carcinogenic metabolites of fluorobenz[c]acridine Dipanjan Pan Gandhi K. Kar Jayanta K. Ray Jyh-Ming Lin Shantu Amin Suchada Chantrapromma ![]() pg 2470; DOI: 10.1039/b102750f |
The photochemical reactions of nitrogen-rich mesoionic 1,3-diphenyltetrazolium heterocycles and related compounds Shuki Araki Hiromi Hattori Koji Ogawa Masashi Kuzuya Tomoko Inoue Hatsuo Yamamura and Masao Kawai pg 2476; DOI: 10.1039/b009526p |
Preparation and synthetic utility of 3-(benzotriazol-1-ylmethyl)areno- and -hetareno[b]thiophenes Alan R. Katritzky Vladimir Y. Vvedensky and Dmytro O. Tymoshenko pg 2483; DOI: 10.1039/b008612f |
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis Gideon Grogan Alexis Carstairs Ian Jackson Denise McIntyre Alan Watt Sabine Flitsch and Nicholas Turner pg 20-xi; DOI: 10.1039/b108606p |
Perkin 1 Abstracts: Natural Product Synthesis Andrew Gunn Jacqueline E. Milne Marcel de Puit and Duncan McArthur pg 20-xvi; DOI: 10.1039/b108756h |
Synthesis of aromatic heterocycles Thomas L. Gilchrist pg 2491; DOI: 10.1039/a904578c |
Rapid assembly of anti,anti-1,2,3-triol motifs via stereoselective addition of organometallics to aldehydes obtained from (R![]() ![]() Darren J. Dixon Lars Krause and Steven V. Ley pg 2516; DOI: 10.1039/b105118k |
Highly stereocontrolled reduction of an alkynyl ketone possessing a 1,3-dithianyl moiety using oxazaborolidine–BH3 Makoto Shimizu Yoshiyuki Ikari and Akinobu Wakabayashi pg 2519; DOI: 10.1039/b107604c |
Lewis-acid catalysed arylation of the hydroxyamino sugar moiety of the natural product SB-219383 John M. Berge Catherine S. V. Houge-Frydrych and Richard L. Jarvest pg 2521; DOI: 10.1039/b105965n |
Synthesis of a conformationally rigid scyllo-inositol polymer as a novel chelating ligand Tae-Hyun Kim and Andrew B. Holmes pg 2524; DOI: 10.1039/b105105a |
Transition metal complexes as linkers for solid phase synthesis: chromium carbonyl complexes as linkers for arenes Alex C. Comely Susan E. Gibson (née Thomas) Neil J. Hales and Mark A. Peplow pg 2526; DOI: 10.1039/b106582n |
Facile synthesis of 6-cyano-9-substituted-9H-purines and their ring expansion to 8-(arylamino)-4-imino-3-methylpyrimidino[5,4-d]pyrimidines Amal Al-Azmi Brian L. Booth Robert A. Carpenter Alice Carvalho Elodie Marrelec Robin G. Pritchard and M. Fernanda J. R. P. Proença pg 2532; DOI: 10.1039/b106539b |
Ring fused 1,2,5-thiadiazoles from oximes and trithiazyl trichloride Charles W. Rees and Tai-Yuen Yue pg 2538; DOI: 10.1039/b106384g |
Synthesis of spiro-indanes by cycloaddition strategy Sambasivarao Kotha and Ethirajan Manivannan pg 2543; DOI: 10.1039/b106280h |
Polyaromatic amines. Part 2. Synthesis of 4,4![]() ![]() ![]() ![]() M. John Plater and Toby Jackson pg 2548; DOI: 10.1039/b106273p |
The synthesis and evaluation of o-phenylenediamine derivatives as fluorescent probes for nitric oxide detection M. John Plater Iain Greig Miep H. Helfrich and StuartH. Ralston pg 2553; DOI: 10.1039/b105953j |
A general ![]() ![]() ![]() Mitsuhiro Yoshimatsu Sachiko Yamaguchi and Yoshiaki Matsubara pg 2560; DOI: 10.1039/b105894k |
Diazoketones as precursors in ![]() Michael R. Linder Wolfgang U. Frey and Joachim Podlech pg 2566; DOI: 10.1039/b105748k |
Efficient and convenient entry to ![]() ![]() ![]() Kazumasa Funabiki Akie Isomura Yoshihiro Yamaguchi Wataru Hashimoto Kei Matsunaga Katsuyoshi Shibata and Masaki Matsui pg 2578; DOI: 10.1039/b105636k |
Vilsmeier–Haack reaction of tertiary alcohols: formation of functionalised pyridines and naphthyridines Ajith Dain Thomas and Chitoorthekkathil V. Asokan pg 2583; DOI: 10.1039/b105634b |
Synthesis of dihydrobenzazaphosphole ligands via an intramolecular cyclisation reaction Wilson Leung Sarah Cosway Raymond H. V. Jones Hannah McCann and Martin Wills pg 2588; DOI: 10.1039/b105495n |
Optimisation of substitution at the 2- and 5- positions of 3,4-dialkoxythiophenes via the Mannich reaction: the influences of steric crowding, electrophile reactivity and temperature Joan Halfpenny Phillip B. Rooney and Zachary S. Sloman pg 2595; DOI: 10.1039/b105476g |
Synthesis and evaluation of a broad range of chiral sulfides for asymmetric sulfur ylide epoxidation of aldehydes Varinder K. Aggarwal Rémy Angelaud Dominique Bihan Paul Blackburn Robin Fieldhouse Silvia J. Fonquerna Gair D. Ford George Hynd Elfyn Jones Ray V. H. Jones Philippe Jubault Matthew J. Palmer Paul D. Ratcliffe and Harry Adams pg 2604; DOI: 10.1039/b105416n |
Diastereoselective synthesis of 2-alkylated 4-silyloxyproline esters Tatsunori Sato Satomi Kawasaki Nobuo Oda Shôko Yagi Serry A. A. El Bialy Jun'ichi Uenishi Masashige Yamauchi and Masazumi Ikeda pg 2623; DOI: 10.1039/b105238c |
![]() Nathalie Defacqz Roland Touillaux Alex Cordi and Jacqueline Marchand-Brynaert pg 2632; DOI: 10.1039/b105111n |
Reusable solid-phase supports for oligonucleotides and antisense therapeutics Richard T. Pon Shuyuan Yu Zhiqiang Guo Ranjit Deshmukh and Yogesh S. Sanghvi pg 2638; DOI: 10.1039/b105089n |
Synthetic studies toward the kempane diterpenes. Diels–Alder additions to bicyclic dienes Chunjian Liu Guanglin Bao and D. Jean Burnell pg 2644; DOI: 10.1039/b104924k |
Synthetic studies toward the kempane diterpenes. Approaches to the assembly of the ring system Guanglin Bao Chunjian Liu and D. Jean Burnell pg 2657; DOI: 10.1039/b104986k |
The synthesis and structural characterisation of some azo-containing phosphine chalcogenides and comparison to non-phosphorus-containing analogues Mark J. Alder Vanessa M. Bates Wendy I. Cross Kevin R. Flower and Robin G. Pritchard pg 2669; DOI: 10.1039/b104918f |
Stereochemistry of enacyloxins. Part 3. (12![]() ![]() ![]() ![]() Ryo Takeuchi Hiromasa Kiyota Manabu Yaosaka Toshihiko Watanabe Keijiro Enari Takeyoshi Sugiyama and Takayuki Oritani pg 2676; DOI: 10.1039/b104341m |
Optimisation of the allylsilane approach to C-10 deoxo carba analogues of dihydroartemisinin: synthesis and in vitro antimalarial activity of new, metabolically stable C-10 analogues Paul M. O'Neill Matthew Pugh Andrew V. Stachulski Stephen A. Ward Jill Davies and B. Kevin Park pg 2682; DOI: 10.1039/b104340b |
Epimerization of peptide nucleic acids analogs during solid-phase synthesis: optimization of the coupling conditions for increasing the optical purity Roberto Corradini Stefano Sforza Arnaldo Dossena Gerardo Palla Raniero Rocchi Ferdinando Filira Flavia Nastri and Rosangela Marchelli pg 2690; DOI: 10.1039/b104146k |
Stereocontrolled construction of rigid tricyclic bis(![]() Jon Efskind Christian Römming and Kjell Undheim pg 2697; DOI: 10.1039/b103254m |
Reactions of 1-(2-alkoxyphenyl)alkaniminyl radicals Rino Leardini Hamish McNab Matteo Minozzi Daniele Nanni David Reed and Andrew G. Wright pg 2704; DOI: 10.1039/b103181n |
Aldol-type condensation reactions of lithium eneselenolates generated from selenoamides with aldehydes Toshiaki Murai Akiko Suzuki and Shinzi Kato pg 2711; DOI: 10.1039/b100198l |
Molecular recognition of xanthine alkaloids: First synthetic receptors for theobromine and a series of new receptors for caffeine Shyamaprosad Goswami Ajit Kumar Mahapatra and Reshmi Mukherjee pg 2717; DOI: 10.1039/b009319j |
Perkin 1 Abstracts: Solid Phase Organic Synthesis Jennifer Delaney Andrew Gunn and Tanya Wildman pg 21-vii; DOI: 10.1039/b109264m |
Recent developments in lanthanide mediated organic synthesis Patrick G. Steel pg 2727; DOI: 10.1039/a908189e |
A novel approach to the synthesis of mono- and dipyrroloporphyrins Ana M. G. Silva Maria A. F. Faustino Augusto C. Tomé Maria G. P. M. S. Neves Artur M. S. Silva and José A. S. Cavaleiro pg 2752; DOI: 10.1039/b108783p |
Reductive cyclization with baker's yeast of 4-alkyl-2-nitroacetanilides to 6-alkylbenzimidazoles and 1-hydroxy-2-methyl-6-alkylbenzimidazoles Arturo Navarro-Ocaña Luís F. Olguín Hector Luna Manuel Jiménez-Estrada and Eduardo Bárzana pg 2754; DOI: 10.1039/b107492j |
Synthesis of (3R,6R)- and (3S,6R)-piperidinone PNA Ask Püschl Thomas Boesen Tullia Tedeschi Otto Dahl and Peter E. Nielsen pg 2757; DOI: 10.1039/b103901f |
A bioisosteric oligosaccharide mimetic based on isofagomine-type monomers Xifu Liang Bent O. Petersen Jens Ø. Duus and Mikael Bols pg 2764; DOI: 10.1039/b103756k |
Reactions of thiobenzoylketene S,N-acetals with silyl enol ethers of cyclic ketones in the presence of desilylating reagents: formation and desulfurization of thienolactams Jong Seok Lee Dong Joon Lee Bo Sung Kim and Kyongtae Kim pg 2774; DOI: 10.1039/b102922n |
A novel synthesis of imidazoles via the cycloaddition of nitrile ylides to their imidoyl chloride precursors Paul W. Groundwater Ian Garnett Andrew J. Morton Toqir Sharif Simon J. Coles Michael B. Hursthouse Miklos Nyerges Rosaleen J. Anderson David Bendell Alexander McKillop and Weimin Zhang pg 2781; DOI: 10.1039/b104130b |
Polyhalogenated heterocyclic compounds. Part 47. Syntheses of multi-substituted pyridine derivatives from pentafluoropyridine Richard D. Chambers Philip R. Hoskin Graham Sandford Dmitrii S. Yufit and Judith A. K. Howard pg 2788; DOI: 10.1039/b105950p |
Reactive immunization elicits catalytic antibodies for polyester hydrolysis Da-Wei Chen Robert J. Kubiak Jon A. Ashley and Kim D. Janda pg 2796; DOI: 10.1039/b105412k |
Diastereoselective Lewis acid mediated hydrophosphonylation of heterocyclic imines: a stereoselective approach towards ![]() Imre Schlemminger Andreas Willecke Wolfgang Maison Rainer Koch Arne Lützen and Jürgen Martens pg 2804; DOI: 10.1039/b101501j |
Cycloaddition of nitrile imines to resin-bound enamines: a solid phase synthesis of 1,4-diarylpyrazoles Andrew C. Donohue Sue Pallich and Tom D. McCarthy pg 2817; DOI: 10.1039/b102913b |
Synthesis of bisquaraine dyes. Novel homologues of 1,2-squaraines bearing symmetrical and unsymmetrical structures Yutaka Hyodo Hiroyuki Nakazumi Shigeyuki Yagi and Kazuhisa Nakai pg 2823; DOI: 10.1039/b104059f |
Development of catalysts for the Baylis–Hillman reaction: the application of tetramethylguanidine and attempts to use a supported analogue Nicholas E. Leadbeater and Cornelia van der Pol pg 2831; DOI: 10.1039/b106267k |
Convenient preparations of polysubstituted 3H-pyrroles promoted by SmI2 Xiaoliang Xu and Yongmin Zhang pg 2836; DOI: 10.1039/b102268g |
Synthesis and applications to asymmetric catalysis of a series of mono- and bis(diazaphospholidine) ligands Donald Smyth Heather Tye Colin Eldred Nathaniel W. Alcock and Martin Wills pg 2840; DOI: 10.1039/b106399p |
Synthesis of (R)-{![]() ![]() ![]() M. Rute G. da Costa M. João M. Curto Stephen G. Davies John Sanders and Fátima C. Teixeira pg 2850; DOI: 10.1039/b107237b |
Lithium–potassium superbases as key reagents for the base-catalysed isomerisation of some terpenoids Annamaria Deagostino Paolo Balma Tivola Cristina Prandi and Paolo Venturello pg 2856; DOI: 10.1039/b106906c |
Intramolecular epoxidation in unsaturated ketones and oxaziridines Alan Armstrong and Alistair G. Draffan pg 2861; DOI: 10.1039/b107839a |
The synthesis of 5-substituted proline derivatives and of 5-substituted pyrrole-2-carboxylates by 5-endo cyclisations featuring a method for effectively favouring these with respect to 5-exo cyclisations David W. Knight Adele L. Redfern and Jeremy Gilmore pg 2874; DOI: 10.1039/b106739g |
Perkin 1 Abstracts: Natural Product Synthesis Andrew Gunn Jacqueline E. Milne Marcel de Puit and Duncan McArthur pg 22-xvii; DOI: 10.1039/b109682f |
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis Gideon Grogan Alexis Carstairs Ian Jackson Denise McIntyre Alan Watt Sabine Flitsch and Nicholas Turner pg 22-xi; DOI: 10.1039/b109853p |
Synthesis of heterocycles by radical cyclisation W. Russell Bowman Martin O. Cloonan and Sussie L. Krintel pg 2885; DOI: 10.1039/a909340k |
Short synthesis of the optically active E-ring portion of (S)-camptothecin S. Leue W. Miao A. Kanazawa Y. Génisson S. Garçon and A. E. Greene pg 2903; DOI: 10.1039/b109071m |
The reactions of diacetylenic ketones with nitrogen nucleophiles; facile preparation of alkynyl substituted pyrimidines and pyrazoles Jack E. Baldwin Gareth J. Pritchard and Richard E. Rathmell pg 2906; DOI: 10.1039/b108645f |
Highly diastereoselective synthesis of ![]() Wim J. N. Meester Rudmer van Dijk Jan H. van Maarseveen Floris P. J. T. Rutjes Pedro H. H. Hermkens and Henk Hiemstra pg 2909; DOI: 10.1039/b108254j |
Asymmetric synthesis of N-diphenylphosphinoylamines by solvent-free enantioselective addition of dialkylzincs to N-diphenylphosphinoylimines Itaru Sato Ryo Kodaka and Kenso Soai pg 2912; DOI: 10.1039/b106775n |
Novel synthesis of enantiomerically enriched 5-hydroxycyclohex-2-enone by enantioselective deprotonation strategy: application to the synthesis of inositol phosphatase inhibitor Toshio Honda and Katsunori Endo pg 2915; DOI: 10.1039/b107567p |
Isolation and characterization of spirocaesalmin, a novel rearranged vouacapane diterpenoid from Caesalpinia minax Hance Ren-Wang Jiang Shuang-Cheng Ma Paul P. H. But and Thomas C. W. Mak pg 2920; DOI: 10.1039/b107473n |
Conjugate addition of 6-membered hydrazine to chiral tert-butyl (E)-2-(p-tolylsulfinyl)cinnamates. Synthesis of (S)-celacinnine Haruo Matsuyama Nobuhiro Itoh Aoi Matsumoto Nahoko Ohira Kenji Hara Masato Yoshida and Masahiko Iyoda pg 2924; DOI: 10.1039/b107443c |
Asymmetric synthesis of ![]() Steven D. Bull Stephen G. Davies and Andrew D. Smith pg 2931; DOI: 10.1039/b107440g |
NMR characterization of lignins from transgenic poplars with suppressed caffeic acid O-methyltransferase activity Jane M. Marita John Ralph Catherine Lapierre Lise Jouanin and Wout Boerjan pg 2939; DOI: 10.1039/b107219f |
Domino Michael–O-alkylation reaction: one-pot synthesis of 2,4-diacylhydrofuran derivatives and its application to antitumor naphthofuran synthesis Hisahiro Hagiwara Kouji Sato Daisuke Nishino Takashi Hoshi Toshio Suzuki and Masayoshi Ando pg 2946; DOI: 10.1039/b107180g |
A new and efficient route to derivatives of (R)-4-hydroxycyclohex-2-enone Libing Yu Ruzhou Zhang and Zhiqin Wang pg 2958; DOI: 10.1039/b107085a |
Synthesis and study of 4-hydroxymethyl-3-(alkylamino)acridines as models of a new class of DNA-intercalating–alkylating agents Franck Charmantray Alain Duflos Jean Lhomme and Martine Demeunynck pg 2962; DOI: 10.1039/b107055j |
Diels–Alder reactions of alkyl 2H-azirine-3-carboxylates with furans M. José Alves Nuno G. Azoia Jamie F. Bickley A. Gil Fortes Thomas L. Gilchrist and Ricardo Mendonça pg 2969; DOI: 10.1039/b106985n |
An efficient method for the one-pot construction of the 1H-naphtho[2,3-c]pyran-5,10-dione system Kazuhiro Kobayashi Masaharu Uchida Tomokazu Uneda Keiichi Yoneda Miyuki Tanmatsu Osamu Morikawa and Hisatoshi Konishi pg 2977; DOI: 10.1039/b106933k |
The stereoselective synthesis of oxetanes; exploration of a new, Mitsunobu-style procedure for the cyclisation of 1,3-diols Martin Christlieb John E. Davies Jason Eames Richard Hooley and Stuart Warren pg 2983; DOI: 10.1039/b106851b |
Pyrrolidinones derived from (S)-pyroglutamic acid. Part 3. ![]() Philip W. H. Chan Ian F. Cottrell and Mark G. Moloney pg 2997; DOI: 10.1039/b106782f |
Pyrrolidinones derived from (S)-pyroglutamic acid. Part 4. ![]() ![]() Philip W. H. Chan Ian F. Cottrell and Mark G. Moloney pg 3007; DOI: 10.1039/b106783b |
A new stereoselective route to the carbocyclic nucleoside cyclobut-A Jagannath Panda Sarita Ghosh and Subrata Ghosh pg 3013; DOI: 10.1039/b106542b |
Expedient syntheses of naturally occurring ()-3-benzylphthalides and ()-3-aryl-8-hydroxy-3,4-dihydroisocoumarins: Structure revision of the ()-3-benzylphthalide isolated from Frullania falciloba Raghao S. Mali Kantipudi N. Babu and Prakash G. Jagtap pg 3017; DOI: 10.1039/b106268a |
Novel cycloadditions of ortho-thioquinones with acyclic dienes: expeditious synthesis of 1,4-benzooxathiines Vijay Nair Bini Mathew Siji Thomas Mariappanadar Vairamani and Sripadi Prabhakar pg 3020; DOI: 10.1039/b106265b |
[2+2]Photocycloaddition of 2-(dibenzylamino)ethyl 3-benzoylacrylate in a crystalline state: weak intermolecular interactions as important factors determining efficiency of the solid-state photoreaction Tadashi Hasegawa Kaori Ikeda and Yuko Yamazaki pg 3025; DOI: 10.1039/b105970j |
Stereoselective synthesis of the pyrroloisoquinoline ring system Steven M. Allin Stella L. James William P. Martin Timothy A. D. Smith and Mark R. J. Elsegood pg 3029; DOI: 10.1039/b105402n |
Putative metabolites of fulvestrant, an estrogen receptor downregulator. Improved glucuronidation using trichloroacetimidates John R. Ferguson John R. Harding David A. Killick Keith W. Lumbard Feodor Scheinmann and Andrew V. Stachulski pg 3037; DOI: 10.1039/b105397n |
Manganese(III) acetate-mediated oxidative coupling of phenylhydrazines with benzene: a novel method for biaryl coupling Ayhan S. Demir Ömer Reis and Emine Özgül-Karaaslan pg 3042; DOI: 10.1039/b105119a |
Absolute stereostructures of cell-adhesion inhibitors, macrosphelides C, E–G and I, produced by a Periconia species separated from an Aplysia sea hare Takeshi Yamada Masashi Iritani Mitsunobu Doi Katsuhiko Minoura Tadayoshi Ito and Atsushi Numata pg 3046; DOI: 10.1039/b104337b |
2-(Lithiomethyl)-1-methylimidazole as a non-reactive bulk base and its novel mixed dimer with a chiral lithium amide in catalytic stereoselective deprotonation Sten O. Nilsson Lill Daniel Pettersen Mohamed Amedjkouh and Per Ahlberg pg 3054; DOI: 10.1039/b104336f |
Reaction of phenylhydrazines with arenes in the presence of aluminium trichloride Atsushi Ohwada Shigeru Nara Takeshi Sakamoto and Yasuo Kikugawa pg 3064; DOI: 10.1039/b103802h |
5-Amino-3-imino-1,2,6,7-tetracyano-3H-pyrrolizine: synthesis of alkylimino derivatives. X-Ray crystal and molecular structures of the hex-5-enyl, and Langmuir–Blodgett film of the octyl and octadecyl derivatives Alberto Flamini Vincenzo Fares Aldo Capobianchi and Veronica Valentini pg 3069; DOI: 10.1039/b103423p |
Reactions of 4-methylchromene-2,7,8-trione with phosphonium ylides. Synthesis and evaluation of fused 1,3-dioxolocoumarins as antioxidants and antiinflammatories Konstantina C. Fylaktakidou Daman R. Gautam Dimitra J. Hadjipavlou-Litina Christos A. Kontogiorgis Konstantinos E. Litinas and Demetrios N. Nicolaides pg 3073; DOI: 10.1039/b103092m |
Nucleoside carbonyl(di- and triphosphates) Ivan B. Yanachkov James M. Stattel and George E. Wright pg 3080; DOI: 10.1039/b102467c |
Perkin 1 Abstracts: Solid Phase Organic Synthesis Fabrice Anizon Jennifer Delaney Andrew Gunn Hassan Mamdani Catherine McCusker Fiona McKerlie and Tanya Wildman pg 23-ix; DOI: 10.1039/b109854n |
Supported catalysts and their applications in synthetic organic chemistry Yolanda R. de Miguel Emilie Brulé and Robert G. Margue pg 3085; DOI: 10.1039/b101948l |
New access to 1,3-dialkyl-2,3-dihydro-2-imino-1H-imidazoles and their application to the first total synthesis of naamine B, a marine 2,3-dihydro-2-imino-1,3-dimethyl-1H-imidazole alkaloid Ikuo Kawasaki Seikou Nakamura Satomi Yanagitani Akiko Kakuno Masayuki Yamashita and Shunsaku Ohta pg 3095; DOI: 10.1039/b108762b |
Biosynthesis of fluoroacetate and 4-fluorothreonine in Streptomyces cattleya. Incorporation of oxygen-18 from [2-2H,2-18O]-glycerol and the role of serine metabolites in fluoroacetaldehyde biosynthesis Christoph Schaffrath Cormac D. Murphy John T. G. Hamilton and David O'Hagan pg 3100; DOI: 10.1039/b108720g |
Orthogonal N,N-deprotection strategies of ![]() Steven D. Bull Stephen G. Davies Peter M. Kelly Massimo Gianotti and Andrew D. Smith pg 3106; DOI: 10.1039/b106389h |
Asymmetric synthesis of ![]() ![]() Steven D. Bull Stephen G. Davies Santiago Delgado-Ballester Peter M. Kelly Luke J. Kotchie Massimo Gianotti Mario Laderas and Andrew D. Smith pg 3112; DOI: 10.1039/b108573p |
A simple access to 3,6-branched oligosaccharides: Synthesis of a glycopeptide derivative that relates to Lycium barbarum L. Yuguo Du Meimei Zhang Feng Yang and Guofeng Gu pg 3122; DOI: 10.1039/b108399f |
Synthesis of new chiral and nonchiral N2O2 and N2S2 tetradentate ligands and their metal complexes Franck Mevellec Sylvain Collet David Deniaud Alain Reliquet and Jean-Claude Meslin pg 3128; DOI: 10.1039/b108210h |
Rearrangement of 1,4,5,6-tetrahalo-7,7-dimethoxybicyclo[2.2.1]hept-5-en-2-ones to phenolic derivatives Faiz Ahmed Khan Jyotirmayee Dash Dheeraj Jain and B. Prabhudas pg 3132; DOI: 10.1039/b108152g |
Synthesis and self-aggregation of zinc chlorophylls possessing an ![]() Shiki Yagai and Hitoshi Tamiaki pg 3135; DOI: 10.1039/b107902f |
Azatriquinanes. Part 4. The chemistry of azatriquinenamine and its bromination products Manuel Lera Alexander J. Blake Claire Wilson and Mark Mascal pg 3145; DOI: 10.1039/b107707d |
6-Substituted 2-azabicyclo[2.2.1]hept-5-enes by nitrogen-directed radical rearrangement: synthesis of an epibatidine analogue with high binding affinity at the nicotinic acetylcholine receptor David M. Hodgson Christopher R. Maxwell Richard Wisedale Ian R. Matthews Kate J. Carpenter Anthony H. Dickenson and Susan Wonnacott pg 3150; DOI: 10.1039/b107414h |
Additions of stabilised and semi-stabilised sulfur ylides to tosyl protected imines: are they under kinetic or thermodynamic control? Varinder K. Aggarwal Jonathan P. H. Charmant Cinzia Ciampi Jonathan M. Hornby Christopher J. O'Brien George Hynd and Richard Parsons pg 3159; DOI: 10.1039/b107275g |
Michael addition of thiols, carbon nucleophiles and amines to dehydroamino acid and dehydropeptide derivatives Paula M. T. Ferreira Hernâni L. S. Maia Luís S. Monteiro and Joana Sacramento pg 3167; DOI: 10.1039/b106487h |
Antitumour polycyclic acridines. Part 9. Synthesis of 7H-pyrido[4,3,2-kl]acridines with basic side chains Michael J. Ellis and Malcolm F. G. Stevens pg 3174; DOI: 10.1039/b106324n |
Antitumour polycyclic acridines. Part 10. Synthesis of penta- and hexa-cyclic heteroaromatic systems by radical cyclisations of substituted 9-anilinoacridines Michael J. Ellis and Malcolm F. G. Stevens pg 3180; DOI: 10.1039/b106327h |
Novel organic-solvent-free aziridination of olefins: Chloramine-T–I2 system under phase-transfer catalysis conditions Daisuke Kano Satoshi Minakata and Mitsuo Komatsu pg 3186; DOI: 10.1039/b104940m |
Intramolecular aldol-type condensation between side chains of naphthoquinones: biomimetic synthesis of 1,6- and 1,8-dihydroxyanthraquinones Hidemitsu Uno Akane Masumoto Erina Honda Yumi Nagamachi Youtarou Yamaoka and Noboru Ono pg 3189; DOI: 10.1039/b104789m |
Peptido-organic Diels–Alder reactions on hydrophilic resin: scope for combinatorial chemistry Anette Graven and Morten Meldal pg 3198; DOI: 10.1039/b103765j |
Reactions of N-benzyl-pyridinium or -isoquinolinium ylides with ethyl 3-fluoro-3-(fluoroalkyl)acrylates to give fluoroalkyl-substituted indolizine and pyrrolo[2,1-a]isoquinoline derivatives Weimin Peng and Shizheng Zhu pg 3204; DOI: 10.1039/b103586j |
Perkin 1 Abstracts: Biocatalysis in Organic Synthesis Gideon Grogan Alexis Carstairs Ian Jackson Denise McIntyre Alan Watt Sabine Flitsch and Nicholas Turner pg 24-xvii; DOI: 10.1039/b110714n |
Organic syntheses through free-radical annulations and related cascade sequences Andrew J. McCarroll and John C. Walton pg 3215; DOI: 10.1039/b105234a |
Formation of adamantan-1-ols by the reactions of adamantanes with 2,3-dichloro-5,6-dicyano-p-benzoquinone (DDQ) in trifluoromethanesulfonic acid Kiyoshi Tanemura Tsuneo Suzuki Yoko Nishida Koko Satsumabayashi and Takaaki Horaguchi pg 3230; DOI: 10.1039/b109548j |
The synthesis of pyrano[2,3-b]quinoxalines related to molybdopterin Ben Bradshaw Andrew Dinsmore David Collison C. David Garner and John A. Joule pg 3232; DOI: 10.1039/b108576j |
Synthesis of the organic ligand of the molybdenum cofactor, in protected form Ben Bradshaw Andrew Dinsmore Wadi Ajana David Collison C. David Garner and John A. Joule pg 3239; DOI: 10.1039/b108579b |
Synthesis of conformationally constrained amino acid and peptide derivatives Patrick D. Bailey Neill Bannister Marine Bernad Sophie Blanchard and Andrew N. Boa pg 3245; DOI: 10.1039/b108872f |
Norlignan biosynthesis in Asparagus officinalis L.: the norlignan originates from two non-identical phenylpropane units Shiro Suzuki Toshiaki Umezawa and Mikio Shimada pg 3252; DOI: 10.1039/b107949b |
Efficient synthesis of pyridines via a sequential solventless aldol condensation and Michael addition Gareth W. V. Cave and Colin L. Raston pg 3258; DOI: 10.1039/b107302h |
Palladium-catalyzed cyanation of bromocalix[4]arenes at the upper rim Hideaki Hioki Rumi Nakaoka Aya Maruyama and Mitsuaki Kodama pg 3265; DOI: 10.1039/b109083f |
Dilithiation of arenetricarbonylchromium(0) complexes with enantioselective quench: application to chiral biaryl synthesis Yen-Ling Tan Andrew J. P. White David A. Widdowson René Wilhelm and David J. Williams pg 3269; DOI: 10.1039/b108807f |
Conjugate additions of organocuprates to a 3-methylene-6-isopropyldiketopiperazine acceptor for the asymmetric synthesis of homochiral ![]() Steven D. Bull Stephen G. Davies A. Christopher Garner and Michael D. O'Shea pg 3281; DOI: 10.1039/b108621a |
Dioxygenase-catalysed mono-, di- and tri-oxygenation of dialkyl sulfides and thioacetals: chemoenzymatic synthesis of enantiopure cis-diol sulfoxides Derek R. Boyd Narain D. Sharma Simon A. Haughey John F. Malone AlistairW. T. King Brian T. McMurray André Alves-Areias Christopher C. R. Allen Robert Holt and Howard Dalton pg 3288; DOI: 10.1039/b108620k |
A rational approach to calix[n]furan precursors Valérie Bénéteau Otto Meth-Cohn and Charles W. Rees pg 3297; DOI: 10.1039/b108402j |
A novel stereoselective synthesis of N-heterocycles by intramolecular hydrovinylation Ulrich Bothe Hans Christian Rudbeck David Tanner and Mogens Johannsen pg 3305; DOI: 10.1039/b108310d |
Rearrangement of ammonium ylides produced by intramolecular reaction of catalytically generated metal carbenoids. Part 1. Synthesis of cyclic amines J. Stephen Clark Paul B. Hodgson Michael D. Goldsmith and Leslie J. Street pg 3312; DOI: 10.1039/b108179a |
Rearrangement of ammonium ylides produced by intramolecular reaction of catalytically generated metal carbenoids. Part 2. Stereoselective synthesis of bicyclic amines J. Stephen Clark Paul B. Hodgson Michael D. Goldsmith Alexander J. Blake Paul A. Cooke and Leslie J. Street pg 3325; DOI: 10.1039/b108182a |
Carotenoids and related polyenes. Part 7. Total synthesis of crassostreaxanthin B applying the stereoselective rearrangement of tetrasubstituted epoxides Chisato Tode Yumiko Yamano and Masayoshi Ito pg 3338; DOI: 10.1039/b108037g |
Synthesis of chiral cis- and trans-furo[3,2-c][2]benzoxocines from D-glucose by regioselective 8-endo aryl radical cyclisation Aniruddha Nandi Ranjan Mukhopadhyay and Partha Chattopadhyay pg 3346; DOI: 10.1039/b107886k |
Novel diphenylphosphine derivatives of 2,2![]() ![]() ![]() ![]() ![]() ![]() ![]() ![]() ![]() ![]() ![]() ![]() John S. Field Raymond J. Haines Elena I. Lakoba and M. Hal Sosabowski pg 3352; DOI: 10.1039/b107389n |
Size discrimination in intramolecular complexation of modified ![]() Julia S. Lock Bruce L. May Philip Clements John Tsanaktsidis Christopher J. Easton and Stephen F. Lincoln pg 3361; DOI: 10.1039/b107324a |
Synthesis of nucleic-acid base containing norbornene derivatives as monomers for ring-opening-metathesis–polymerization R. Gareth Davies Vernon C. Gibson Michael B. Hursthouse Mark E. Light Edward L. Marshall Michael North David A. Robson Ian Thompson Andrew J. P. White David J. Williams and Paul J. Williams pg 3365; DOI: 10.1039/b107139d |
Nitrogen-containing heterocycles: 1,3-dipolar cycloaddition of stabilized nitrones with alkynes; primary cycloadducts, first and second generation rearrangement processes Frances Heaney Julie Fenlon Colm O'Mahony Patrick McArdle and Desmond Cunningham pg 3382; DOI: 10.1039/b106832f |
On the scope and limitations of the Heck reaction of upper rim tetraiodocalix[4]arenes Nikolai Kuhnert and Adam Le-Gresley pg 3393; DOI: 10.1039/b106535c |
Polyhalogenated BEDT-TTF through chlorination (SO2Cl2, Cl2) and fluorination (Selectfluor, XeF2) of 5,6-dihydro[1,3]dithiolo[4,5-b][1,4]dithiin-2-one Olivier J. Dautel and Marc Fourmigué pg 3399; DOI: 10.1039/b106144p |
Facile attachment of functional moieties to crosslinked polystyrene beads via robust linkages: Suzuki reactions using polymer-supported boronic acids Roger J. Kell Philip Hodge Mohammad Nisar and Richard T. Williams pg 3403; DOI: 10.1039/b103760a |
Synthesis of geminal bis(hydroxymethyl)pyrrolidine and pyrrolizidine imino sugars Frank Schieweck and Hans-Josef Altenbach pg 3409; DOI: 10.1039/b007607o |